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Found 3 Enz. Inhib. hit(s) with Target = 'Taste receptor type 2 member 8' and Ligand = 'BDBM210973'
TargetTaste receptor type 2 member 8(Homo sapiens (Human))
Senomyx

US Patent
LigandPNGBDBM210973(US9247759, 4-7 | US9247759, compound B)
Affinity DataIC50:  390nMAssay Description:In another embodiment, Fluorescence Polarization ("FP") based assays may be used to detect and monitor ligand binding. Fluorescence polarization is a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTaste receptor type 2 member 8(Homo sapiens (Human))
Senomyx

US Patent
LigandPNGBDBM210973(US9247759, 4-7 | US9247759, compound B)
Affinity DataIC50:  400nMAssay Description:In another embodiment, Fluorescence Polarization ("FP") based assays may be used to detect and monitor ligand binding. Fluorescence polarization is a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTaste receptor type 2 member 8(Homo sapiens (Human))
Senomyx

US Patent
LigandPNGBDBM210973(US9247759, 4-7 | US9247759, compound B)
Affinity DataIC50:  700nMAssay Description:Antagonist activity at recombinant human TAS2R8 stably expressed in cells co-expressing Galpha16gust44 assessed as inhibition of andrographolide-indu...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed