Compile Data Set for Download or QSAR
maximum 50k data
Found 2 Enz. Inhib. hit(s) with Target = 'Tyrosine-protein kinase JAK2' and Ligand = 'BDBM50361204'
TargetTyrosine-protein kinase JAK2(Homo sapiens (Human))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50361204(CHEMBL1934353)
Affinity DataIC50:  2.5nMAssay Description:Inhibition of human recombinant JAK2 expressed in baculovirus expression system after 20 mins by time resolved fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK2(Homo sapiens (Human))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50361204(CHEMBL1934353)
Affinity DataIC50:  12nMAssay Description:Inhibition of JAK2 in GM-CSF-stimulated human TF1 cells preincubated for 1 hr prior to challengeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed