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Found 3 Enz. Inhib. hit(s) with Target = 'UDP-N-acetylglucosamine--peptide N-acetylglucosaminyltransferase 110 kDa subunit' and Ligand = 'BDBM50200111'
TargetUDP-N-acetylglucosamine--peptide N-acetylglucosaminyltransferase 110 kDa subunit(Homo sapiens (Human))
University Of Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50200111(CHEMBL3981566)
Affinity DataKi:  9.20E+4nMAssay Description:Noncompetitive inhibition of OGT (unknown origin) using variable UDP-GlcNAc levels and fixed CKII peptide level by UDP-Glo glycosyltransferase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUDP-N-acetylglucosamine--peptide N-acetylglucosaminyltransferase 110 kDa subunit(Homo sapiens (Human))
University Of Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50200111(CHEMBL3981566)
Affinity DataKi:  3.10E+5nMAssay Description:Noncompetitive inhibition of OGT (unknown origin) using fixed UDP-GlcNAc levels and variable CKII peptide level by UDP-Glo glycosyltransferase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUDP-N-acetylglucosamine--peptide N-acetylglucosaminyltransferase 110 kDa subunit(Homo sapiens (Human))
University Of Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50200111(CHEMBL3981566)
Affinity DataIC50:  1.39E+5nMAssay Description:Inhibition of OGT (unknown origin) assessed as reduction in GlcNAc transfer to CKII peptide incubated for 60 mins by HPLC methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed