Found 1 Enz. Inhib. hit(s) with Target = 'UDP-N-acetylglucosamine--peptide N-acetylglucosaminyltransferase 110 kDa subunit' and Ligand = 'BDBM50200118'
TargetUDP-N-acetylglucosamine--peptide N-acetylglucosaminyltransferase 110 kDa subunit(Homo sapiens (Human))
University Of Chinese Academy Of Sciences
Curated by ChEMBL
University Of Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibition of OGT (unknown origin) assessed as reduction in GlcNAc transfer to CKII peptide incubated for 60 mins by HPLC methodMore data for this Ligand-Target Pair