Compile Data Set for Download or QSAR
maximum 50k data
Found 9 Enz. Inhib. hit(s) with all data for assayid = 1 entry = 50012880
TargetProtein phosphatase 3 catalytic subunit alpha(Homo sapiens (Human))
Enanta Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50022815((3S,6S,9S,12R,15S,18S,21S,24S,30S,33S)-30-ethyl-33...)
Affinity DataIC50:  183nMAssay Description:Compound was evaluated for its inhibitory activity in a calcineurin inhibition assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein phosphatase 3 catalytic subunit alpha(Homo sapiens (Human))
Enanta Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50123747(6-(5-Ethyl-11,17,26,29-tetraisobutyl-14,32-diisopr...)
Affinity DataIC50:  363nMAssay Description:Compound was evaluated for its inhibitory activity in a calcineurin inhibition assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein phosphatase 3 catalytic subunit alpha(Homo sapiens (Human))
Enanta Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50123748(6-(5-Ethyl-11,17,26,29-tetraisobutyl-14,32-diisopr...)
Affinity DataIC50:  581nMAssay Description:Compound was evaluated for its inhibitory activity in a calcineurin inhibition assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein phosphatase 3 catalytic subunit alpha(Homo sapiens (Human))
Enanta Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50123744(6-(5-Ethyl-11,17,26,29-tetraisobutyl-14,32-diisopr...)
Affinity DataIC50:  636nMAssay Description:Compound was evaluated for its inhibitory activity in a calcineurin inhibition assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein phosphatase 3 catalytic subunit alpha(Homo sapiens (Human))
Enanta Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50123741(6-(5-Ethyl-11,17,26,29-tetraisobutyl-14,32-diisopr...)
Affinity DataIC50:  840nMAssay Description:Compound was evaluated for its inhibitory activity in a calcineurin inhibition assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein phosphatase 3 catalytic subunit alpha(Homo sapiens (Human))
Enanta Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50123743(6-(5-Ethyl-11,17,26,29-tetraisobutyl-14,32-diisopr...)
Affinity DataIC50:  890nMAssay Description:Compound was evaluated for its inhibitory activity in a calcineurin inhibition assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein phosphatase 3 catalytic subunit alpha(Homo sapiens (Human))
Enanta Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50123746(6-(5-Ethyl-11,17,26,29-tetraisobutyl-14,32-diisopr...)
Affinity DataIC50:  1.54E+3nMAssay Description:Compound was evaluated for its inhibitory activity in a calcineurin inhibition assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein phosphatase 3 catalytic subunit alpha(Homo sapiens (Human))
Enanta Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50123740(6-(5-Ethyl-11,17,26,29-tetraisobutyl-14,32-diisopr...)
Affinity DataIC50: >5.00E+3nMAssay Description:Compound was evaluated for its inhibitory activity in a calcineurin inhibition assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein phosphatase 3 catalytic subunit alpha(Homo sapiens (Human))
Enanta Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50123739(6-(5-Ethyl-11,17,26,29-tetraisobutyl-14,32-diisopr...)
Affinity DataIC50: >5.00E+3nMAssay Description:Compound was evaluated for its inhibitory activity in a calcineurin inhibition assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed