Filter my 1564 hits
Targets 30▿
Alpha-1A adrenergic receptor 270
Alpha-1D adrenergic receptor 250
Alpha-1B adrenergic receptor 248
Type-2 angiotensin II receptor 225
Type-1 angiotensin II receptor 222
B1 bradykinin receptor 91
Botulinum neurotoxin type A 30
Calmodulin-sensitive adenylate cyclase 24
Alpha-2C adrenergic receptor 19
Alpha-2B adrenergic receptor 19
Amyloid-beta precursor protein 19
Alpha-2A adrenergic receptor 19
Fatty-acid amide hydrolase 1 [30-579] 18
Fatty-acid amide hydrolase 1 18
Type-1 angiotensin II receptor A/B 13
Mu-type opioid receptor 13
Endothelin-1 receptor 12
Endothelin receptor type B 12
Histamine H1 receptor 10
B2 bradykinin receptor 8
Potassium voltage-gated channel subfamily H member 2 8
Lethal factor 5
Voltage-dependent L-type calcium channel subunit alpha-1C 3
5-hydroxytryptamine receptor 1A 2
Alpha-1A/Alpha-1B/Alpha-1D adrenergic receptor 1
5-hydroxytryptamine receptor 1B 1
5-hydroxytryptamine receptor 2A 1
Voltage-dependent L-type calcium channel subunit alpha-1C/alpha-1D/alpha-1S 1
5-hydroxytryptamine receptor 1D 1
Histamine H2 receptor 1
...
Publications 25▿
J Med Chem 38: 3741 -58 (1995) 258 J Med Chem 42: 4778 -93 (1999) 113 Bioorg Med Chem Lett 9: 2843 -8 (1999) 103 J Med Chem 43: 2703 -18 (2000) 102 J Med Chem 42: 4794 -803 (1999) 91 J Med Chem 42: 4764 -77 (1999) 88 J Med Chem 37: 4464 -78 (1995) 86 J Med Chem 42: 4804 -13 (1999) 81 Bioorg Med Chem Lett 10: 1625 -8 (2000) 81 Bioorg Med Chem Lett 8: 2467 -72 (1999) 67 Bioorg Med Chem Lett 5: 1359 -1364 (1995) 60 Bioorg Med Chem Lett 4: 2787 -2792 (1994) 56 Bioorg Med Chem Lett 10: 1917 -20 (2001) 48 Bioorg Med Chem Lett 9: 291 -4 (1999) 44 J Med Chem 51: 3946 -52 (2008) 38 ACS Med Chem Lett 4: 509 -13 (2013) 36 Bioorg Med Chem Lett 23: 2505 -11 (2013) 30 J Med Chem 46: 1803 -6 (2003) 29 Bioorg Med Chem Lett 28: 134 -139 (2018) 29 Bioorg Med Chem Lett 5: 1155 -1158 (1995) 24 Bioorg Med Chem Lett 14: 6045 -8 (2004) 22 Bioorg Med Chem Lett 8: 2495 -500 (1999) 22 ACS Med Chem Lett 2: 498 -502 (2011) 19 J Med Chem 43: 2775 -8 (2000) 19 Bioorg Med Chem Lett 17: 3006 -9 (2007) 18
Institutions 6▿
Merck Research Laboratories 638 Synaptic Pharmaceutical 495 Merck 232 TBA 140 Panthera Biopharma 30 Hawaii Biotech 29
Affinity: 0.010 to 9.5E+5 nM▿
Xtal structures: 0 Docked structures: 0 Catalog Cmpds: 16