Compile Data Set for Download or QSAR
maximum 50k data
Found 4 of ec50 for monomerid = 21762
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Bayer Healthcare Pharmaceuticals

LigandPNGBDBM21762(2-[(1S)-5-[3-(3,4-dimethylphenoxy)propoxy]-2,3-dih...)
Affinity DataEC50:  67nMT: 2°CAssay Description:Activity was assessed by measuring the human PPAR ligand binding domain with the co-activator protein. Europium labeled anti-GST antibody, streptavid...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Bayer Healthcare Pharmaceuticals

LigandPNGBDBM21762(2-[(1S)-5-[3-(3,4-dimethylphenoxy)propoxy]-2,3-dih...)
Affinity DataEC50: >1.00E+4nMT: 2°CAssay Description:PPAR gamma activity was assessed by using the IRBA in mouse 3T3-L1 cells. This assay measures the ability of test compound to cause an increase in th...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Bayer Healthcare Pharmaceuticals

LigandPNGBDBM21762(2-[(1S)-5-[3-(3,4-dimethylphenoxy)propoxy]-2,3-dih...)
Affinity DataEC50: >1.00E+4nMpH: 7.4 T: 2°CAssay Description:Activity was assessed by measuring the human PPAR ligand binding domain with the co-activator protein. Europium labeled anti-GST antibody, streptavid...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Bayer Healthcare Pharmaceuticals

LigandPNGBDBM21762(2-[(1S)-5-[3-(3,4-dimethylphenoxy)propoxy]-2,3-dih...)
Affinity DataEC50:  1.49E+7nMAssay Description:Agonist activity at GST-tagged Homo sapiens (human) PPARdelta ligand binding domain after 2 hr by FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article