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Found 5 of ec50 for monomerid = 21785
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Bayer Healthcare Pharmaceuticals

LigandPNGBDBM21785(2-[(1S)-5-(3-{4-[5-(trifluoromethyl)pyridin-2-yl]p...)
Affinity DataEC50:  0.950nMT: 2°CAssay Description:Activity was assessed by measuring the human PPAR ligand binding domain with the co-activator protein. Europium labeled anti-GST antibody, streptavid...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Bayer Healthcare Pharmaceuticals

LigandPNGBDBM21785(2-[(1S)-5-(3-{4-[5-(trifluoromethyl)pyridin-2-yl]p...)
Affinity DataEC50:  1.80E+3nMT: 2°CAssay Description:PPAR gamma activity was assessed by using the IRBA in mouse 3T3-L1 cells. This assay measures the ability of test compound to cause an increase in th...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Bayer Healthcare Pharmaceuticals

LigandPNGBDBM21785(2-[(1S)-5-(3-{4-[5-(trifluoromethyl)pyridin-2-yl]p...)
Affinity DataEC50:  2.90E+3nMT: 2°CAssay Description:Activity was assessed by measuring the human PPAR ligand binding domain with the co-activator protein. Europium labeled anti-GST antibody, streptavid...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Bayer Healthcare Pharmaceuticals

LigandPNGBDBM21785(2-[(1S)-5-(3-{4-[5-(trifluoromethyl)pyridin-2-yl]p...)
Affinity DataEC50:  3.45E+5nMAssay Description:Agonist activity at GST-tagged Homo sapiens (human) PPARalpha ligand binding domain after 2 hr by FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Bayer Healthcare Pharmaceuticals

LigandPNGBDBM21785(2-[(1S)-5-(3-{4-[5-(trifluoromethyl)pyridin-2-yl]p...)
Affinity DataEC50:  5.62E+5nMAssay Description:Agonist activity at Homo sapiens (human) PPARgamma expressed in mouse 3T3-L1 cells incubated for 2 days followed by compound wash out measured after ...More data for this Ligand-Target Pair
In DepthDetails Article