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Found 3 of ec50 for monomerid = 293987
TargetMelanocortin receptor 4(Rattus norvegicus)TBA
LigandPNGBDBM293987(5-((2S)-2-(4-((2-Methyl-3-(2- methylphenyl)benzo[b...)
Affinity DataEC50:  10nMAssay Description:Agonist activity at rat GPR40 assessed as increase in intracellular calcium flux by cell based FLIPR assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))TBA
LigandPNGBDBM293987(5-((2S)-2-(4-((2-Methyl-3-(2- methylphenyl)benzo[b...)
Affinity DataEC50:  20nMAssay Description:Agonist activity at human GPR40 assessed as increase in intracellular calcium flux by cell based FLIPR assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))TBA
LigandPNGBDBM293987(5-((2S)-2-(4-((2-Methyl-3-(2- methylphenyl)benzo[b...)
Affinity DataEC50:  28nMT: 2°CAssay Description:Compounds were tested in a calcium flux assay using transfected HEK293 cells stably expressing either human GPR40 or rat GPR40. Human GPR40 expressin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent