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Found 2 of ec50 for monomerid = 50172376
TargetApelin receptor(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM50172376(CHEMBL3810012)
Affinity DataEC50:  14nMAssay Description:Agonist activity at human APJ receptor expressed in HEK-293 cells assessed as dissociation of G-alpha-i1 protein after 5 mins by BRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetApelin receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50172376(CHEMBL3810012)
Affinity DataEC50:  316nMAssay Description:Agonist activity at human APJ receptor expressed in HEK-293 cells assessed as beta-arrestin2 recruitment after 30 mins by BRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed