TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Centro Nacional de Investigaciones Oncologicas (CNIO)
US Patent
Centro Nacional de Investigaciones Oncologicas (CNIO)
US Patent
Affinity DataIC50: 676nMpH: 7.5 T: 2°CAssay Description:The kinase activity was measured by using the commercial ADP Hunter Plus assay available from DiscoveRx (#33-016), which is a homogeneous assay to me...More data for this Ligand-Target Pair