Compile Data Set for Download or QSAR
maximum 50k data
Found 4 of ic50 for monomerid = 236660
TargetDual specificity protein kinase TTK(Homo sapiens (Human))
Bayer

Curated by ChEMBL
LigandPNGBDBM236660(US9388140, 1)
Affinity DataIC50:  24nMAssay Description:Inhibition of GST-tagged recombinant human MPS1 expressed in baculovirus expression system using biotin-Ahx-PWDPDDADITEILG as substrate preincubated ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDual specificity protein kinase TTK(Homo sapiens (Human))
Bayer

Curated by ChEMBL
LigandPNGBDBM236660(US9388140, 1)
Affinity DataIC50:  24.4nMpH: 7.7 T: 2°CAssay Description:For the assay 50 nL of a 100-fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384 well microtiter plate (...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDual specificity protein kinase TTK(Homo sapiens (Human))
Bayer

Curated by ChEMBL
LigandPNGBDBM236660(US9388140, 1)
Affinity DataIC50:  1.16E+3nMAssay Description:Inhibition of GST-tagged recombinant human MPS1 expressed in baculovirus expression system using biotin-Ahx-PWDPDDADITEILG as substrate preincubated ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDual specificity protein kinase TTK(Homo sapiens (Human))
Bayer

Curated by ChEMBL
LigandPNGBDBM236660(US9388140, 1)
Affinity DataIC50:  3.44E+3nMAssay Description:Inhibition of MPS1 in human HeLa cells assessed as reduction in spindle assembly checkpoint incubated for 4 hrs by p-histone H3/Hoechst 33342 stainin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed