Compile Data Set for Download or QSAR
maximum 50k data
Found 6 of ic50 for monomerid = 28669
LigandPNGBDBM28669(2-{[3-(1,2,3,4-tetrahydroisoquinoline-2-sulfonyl)b...)
Affinity DataIC50:  5nM EC50:  158nMpH: 7.0 T: 2°CAssay Description:Competition-binding curves for test compounds were determined with expressed human PPAR LBD. Plots of inhibitor concentration versus cpm of radioliga...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM28669(2-{[3-(1,2,3,4-tetrahydroisoquinoline-2-sulfonyl)b...)
Affinity DataIC50:  5nMAssay Description:Agonist activity at PPARdeltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Universidad Nacional Aut£Noma De M£Xico

Curated by ChEMBL
LigandPNGBDBM28669(2-{[3-(1,2,3,4-tetrahydroisoquinoline-2-sulfonyl)b...)
Affinity DataIC50:  1.58E+3nMAssay Description:Agonist activity at PPARalphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Universidad Nacional Aut£Noma De M£Xico

Curated by ChEMBL
LigandPNGBDBM28669(2-{[3-(1,2,3,4-tetrahydroisoquinoline-2-sulfonyl)b...)
Affinity DataIC50:  1.59E+3nMpH: 7.0 T: 2°CAssay Description:Competition-binding curves for test compounds were determined with expressed human PPAR LBD. Plots of inhibitor concentration versus cpm of radioliga...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM28669(2-{[3-(1,2,3,4-tetrahydroisoquinoline-2-sulfonyl)b...)
Affinity DataIC50:  3.16E+3nMAssay Description:Competition-binding curves for test compounds were determined with expressed human PPAR LBD. Plots of inhibitor concentration versus cpm of radioliga...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM28669(2-{[3-(1,2,3,4-tetrahydroisoquinoline-2-sulfonyl)b...)
Affinity DataIC50:  3.16E+3nMAssay Description:Agonist activity at PPARgammaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed