Compile Data Set for Download or QSAR
maximum 50k data
Found 5 of ic50 for monomerid = 50006638
TargetNeuronal acetylcholine receptor subunit beta-2(Mus musculus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50006638(CHEMBL2140445)
Affinity DataIC50:  2.60E+3nMAssay Description:Antagonist activity at mouse alpha4/beta2 nAChR expressed in HEK293 cells assessed as inhibition of (S)-nicotine-induced activity by FLIPR membrane p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit beta-2/beta-4(Mus musculus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50006638(CHEMBL2140445)
Affinity DataIC50:  2.60E+3nMAssay Description:Antagonist activity at mouse alpha4beta2 nAChR expressed in HEK293 cells assessed as inhibition of (S)-nicotine-induced current response measured up ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Homo sapiens (Human))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50006638(CHEMBL2140445)
Affinity DataIC50: >1.00E+5nMAssay Description:Antagonist activity at human alpha7 nAChR expressed in HEK293 cells co-expressing Ric-3/NACHO assessed as inhibition of ACh-induced calcium mobilizat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Rattus norvegicus (Rat))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50006638(CHEMBL2140445)
Affinity DataIC50:  3.00E+5nMAssay Description:Antagonist activity at rat alpha3beta4 nAChR expressed in HEK293 cells assessed as inhibition of (S)-nicotine-induced current response measured up to...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Rattus norvegicus (Rat))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50006638(CHEMBL2140445)
Affinity DataIC50:  3.00E+5nMAssay Description:Antagonist activity at rat alpha3/beta4 nAChR expressed in HEK293 cells assessed as inhibition of (S)-nicotine-induced activity by FLIPR membrane pot...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed