Compile Data Set for Download or QSAR
maximum 50k data
Found 2 of ic50 for monomerid = 50224352
TargetAdenosine receptor A3(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM50224352(4-methoxy-N-(1-oxo-2-p-tolyl-1H-3,3,5,9b-tetraaza-...)
Affinity DataIC50:  0.580nMAssay Description:Antagonist activity at human adenosine A3 receptor expressed in CHO cells assessed as inhibition of forskolin-stimulated cAMP accumulationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM50224352(4-methoxy-N-(1-oxo-2-p-tolyl-1H-3,3,5,9b-tetraaza-...)
Affinity DataIC50:  1.53E+3nMAssay Description:Antagonist activity at human adenosine A2B receptor expressed in CHO cells assessed as inhibition of NECA-stimulated cAMP accumulationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed