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Found 4 of ic50 for monomerid = 50234942
TargetHistone acetyltransferase KAT2B(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50234942(CHEMBL4093233)
Affinity DataIC50:  2.00E+4nMAssay Description:Displacement of GSK3103956A from FLAG-6 His-Halo tagged human PCAF bromodomain (715 to 831 residues) incubated for 30 mins in dark by TR-FRET assayMore data for this Ligand-Target Pair
TargetHistone acetyltransferase KAT2B(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50234942(CHEMBL4093233)
Affinity DataIC50:  2.00E+4nMAssay Description:Binding affinity to PCAF (unknown origin) N-terminal bromodomain by TR-FRET assayMore data for this Ligand-Target Pair
TargetBromodomain-containing protein 9(Homo sapiens (Human))
Glaxosmithkline R&D

Curated by ChEMBL
LigandPNGBDBM50234942(CHEMBL4093233)
Affinity DataIC50:  2.51E+4nMAssay Description:Binding affinity to BRD9 (unknown origin) N-terminal bromodomain by TR-FRET assayMore data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Glaxosmithkline R&D

Curated by ChEMBL
LigandPNGBDBM50234942(CHEMBL4093233)
Affinity DataIC50:  1.26E+5nMAssay Description:Binding affinity to BRD4 (1) (unknown origin) N-terminal bromodomain by TR-FRET assayMore data for this Ligand-Target Pair