Compile Data Set for Download or QSAR
maximum 50k data
Found 3 of ic50 for monomerid = 50319837
TargetProstaglandin E2 receptor EP4 subtype(Homo sapiens (Human))
Merck Frosst Canada

Curated by ChEMBL
LigandPNGBDBM50319837(4-(1-(1-(4-(trifluoromethyl)benzyl)-1H-indole-7-ca...)
Affinity DataIC50:  1.30nMAssay Description:Antagonist activity at human prostanoid EP4 receptor expressed in HEK293 cells assessed as inhibition of PGE2-induced cAMP accumulation by scintillat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP4 subtype(Homo sapiens (Human))
Merck Frosst Canada

Curated by ChEMBL
LigandPNGBDBM50319837(4-(1-(1-(4-(trifluoromethyl)benzyl)-1H-indole-7-ca...)
Affinity DataIC50:  1.80nMAssay Description:Antagonist activity at human prostanoid EP4 receptor expressed in HEK293 cells assessed as inhibition of PGE2-induced cAMP accumulation by scintillat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP4 subtype(Homo sapiens (Human))
Merck Frosst Canada

Curated by ChEMBL
LigandPNGBDBM50319837(4-(1-(1-(4-(trifluoromethyl)benzyl)-1H-indole-7-ca...)
Affinity DataIC50:  9.5nMAssay Description:Antagonist activity at prostanoid EP4 receptor in human whole blood assessed as inhibition of TNFalpha-induced IP-10 release in presence EP4 agonist ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed