Compile Data Set for Download or QSAR
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Found 2 of ic50 for monomerid = 7602
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D1(Homo sapiens (Human))
Astrazeneca

LigandPNGBDBM7602(4,6-bis anilino pyrimidine deriv. 15 | 4-N-(2,5-di...)
Affinity DataIC50:  800nMpH: 7.0 T: 2°CAssay Description:The kinase activity was assayed using an in vitro scintillation proximity assay (SPA) for measuring incorporation of [gamma-33P] ATP into GST-Rb.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Astrazeneca

LigandPNGBDBM7602(4,6-bis anilino pyrimidine deriv. 15 | 4-N-(2,5-di...)
Affinity DataIC50:  1.90E+4nMAssay Description:The kinase activity was assayed using an in vitro scintillation proximity assay (SPA) for measuring incorporation of [gamma-33P] ATP into GST-Rb.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed