Compile Data Set for Download or QSAR
maximum 50k data
Found 4 of ic50 for monomerid = 8393
TargetGlycogen synthase kinase-3 alpha(Homo sapiens (Human))
Glaxosmithkline

LigandPNGBDBM8393(CHEMBL261690 | N-[5-bromo-6-(1,3-thiazol-2-yl)-1H-...)
Affinity DataIC50:  99nMAssay Description:The biochemical activity of compounds was determined by incubation with specific enzyme and substrate in the presence 10 uM ATP/ [gamma-33P] ATP. Aft...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
University Of Jordan

Curated by ChEMBL
LigandPNGBDBM8393(CHEMBL261690 | N-[5-bromo-6-(1,3-thiazol-2-yl)-1H-...)
Affinity DataIC50:  99nMAssay Description:Inhibition of recombinant GSK3-betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
National Institute Of Pharmaceutical Education And Research

Curated by ChEMBL
LigandPNGBDBM8393(CHEMBL261690 | N-[5-bromo-6-(1,3-thiazol-2-yl)-1H-...)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of CDK2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
Glaxosmithkline

LigandPNGBDBM8393(CHEMBL261690 | N-[5-bromo-6-(1,3-thiazol-2-yl)-1H-...)
Affinity DataIC50: >1.00E+3nMAssay Description:In vitro kinase assay using purified CDK2/Cyclin A was incubated at room temperature with substrate, and test compounds in the presence of 100 uM ATP...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed