Compile Data Set for Download or QSAR
maximum 50k data
Found 2 of ki for monomerid = 25375
TargetDimer of Gag-Pol polyprotein [501-599,Q508K,L534I,L564I,C568A,C596A](Human immunodeficiency virus type 1)
Purdue University

LigandPNGBDBM25375((R)-(hydroxyethylamino)sulfonamide isostere, 3l | ...)
Affinity DataKi:  1.90nM ΔG°:  -49.8kJ/mole IC50: >1.00E+3nMpH: 6.4 T: 2°CAssay Description:The Ki values were determined by substrate cleavage assay using fluorogenic substrate, 2-(aminobenzoyl)-Thr-Ile-Nle-Phe(p-NO2)-Gln-Arg-NH2. A standar...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein(Human immunodeficiency virus type 1 group M subtyp...)
Purdue Research Foundation

US Patent
LigandPNGBDBM25375((R)-(hydroxyethylamino)sulfonamide isostere, 3l | ...)
Affinity DataKi:  1.90nMAssay Description:Enzyme inhibitory assay utilizes a protocol described by Toth and Marshall (Toth, M. V.; Marshall G.R. A simple, continuous fluormetric assay for HIV...More data for this Ligand-Target Pair
In DepthDetails US Patent