Compile Data Set for Download or QSAR
maximum 50k data
Found 4 of ki for monomerid = 32387
TargetPepsin A(Porcine)
Philipps University Marburg

LigandPNGBDBM32387(phenyl-substituted sulfonamides, 6d)
Affinity DataKi:  3.90E+3nM ΔG°:  -30.9kJ/moleT: 2°CAssay Description:Enzyme assay was performed at room temperature on a microplate reader (Safire2TM) using black 96-well microtiter plates purchased from Nunc. Inhibito...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin II(Plasmodium falciparum)
Philipps University Marburg

LigandPNGBDBM32387(phenyl-substituted sulfonamides, 6d)
Affinity DataKi:  4.20E+3nM ΔG°:  -30.5kJ/molepH: 4.5 T: 2°CAssay Description:Enzyme assay was performed at room temperature on a microplate reader (Safire2TM) using black 96-well microtiter plates purchased from Nunc. Inhibito...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasmepsin IV(Plasmodium falciparum)
Philipps University Marburg

LigandPNGBDBM32387(phenyl-substituted sulfonamides, 6d)
Affinity DataKi:  7.50E+3nM ΔG°:  -29.1kJ/molepH: 4.5 T: 2°CAssay Description:Enzyme assay was performed at room temperature on a microplate reader (Safire2TM) using black 96-well microtiter plates purchased from Nunc. Inhibito...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDimer of Gag-Pol polyprotein [501-599](Human immunodeficiency virus type 1)
Philipps University Marburg

LigandPNGBDBM32387(phenyl-substituted sulfonamides, 6d)
Affinity DataKi:  9.60E+3nM ΔG°:  -28.4kJ/molepH: 5.5 T: 2°CAssay Description:Enzyme assay was performed at room temperature on a microplate reader (Safire2TM) using black 96-well microtiter plates purchased from Nunc. Inhibito...More data for this Ligand-Target Pair