Affinity DataKi: 0.0800nMAssay Description:Binding affinity against Dopamine receptor D1 of rat striatal receptor using [3H]SCH-23390More data for this Ligand-Target Pair
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Friedrich-Schiller-Universit£T Jena
Curated by ChEMBL
Friedrich-Schiller-Universit£T Jena
Curated by ChEMBL
Affinity DataKi: 1.86nMAssay Description:Displacement of [3H]SCH23390 from human cloned dopamine D1 receptorMore data for this Ligand-Target Pair
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Friedrich-Schiller-Universit£T Jena
Curated by ChEMBL
Friedrich-Schiller-Universit£T Jena
Curated by ChEMBL
Affinity DataKi: 1.90nMAssay Description:Displacement of [3H]SCH 23390 from human cloned dopamine D1 receptor expressed in HEK 293 cellsMore data for this Ligand-Target Pair
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Friedrich-Schiller-Universit£T Jena
Curated by ChEMBL
Friedrich-Schiller-Universit£T Jena
Curated by ChEMBL
Affinity DataKi: 1.90nMAssay Description:Displacement of [3H]SCH 23390 from D1 dopamine receptorMore data for this Ligand-Target Pair
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Friedrich-Schiller-Universit£T Jena
Curated by ChEMBL
Friedrich-Schiller-Universit£T Jena
Curated by ChEMBL
Affinity DataKi: 1.90nMAssay Description:Displacement of [3H]SCH 23390 from human D1 dopamine receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Friedrich-Schiller-Universit£T Jena
Curated by ChEMBL
Friedrich-Schiller-Universit£T Jena
Curated by ChEMBL
Affinity DataKi: 2.90nMAssay Description:Displacement of [3H]-SCH23390 from D1 receptor (unknown origin) expressed in HEK293T cell membranes measured after 2 hrs by microbeta scintillation c...More data for this Ligand-Target Pair
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Friedrich-Schiller-Universit£T Jena
Curated by ChEMBL
Friedrich-Schiller-Universit£T Jena
Curated by ChEMBL
Affinity DataKi: 3nMAssay Description:Displacement of [3H]-SCH23390 from D1 receptor (unknown origin) expressed in HEK293T cell membranes measured after 2 hrs by microbeta scintillation c...More data for this Ligand-Target Pair
Affinity DataKi: 6nMAssay Description:Binding affinity against Dopamine receptor D2 of rat striatal mambranes using [3H]spiperoneMore data for this Ligand-Target Pair
TargetD(1B) dopamine receptor(Homo sapiens (Human))
Friedrich-Schiller-UniversitäT Jena
Curated by ChEMBL
Friedrich-Schiller-UniversitäT Jena
Curated by ChEMBL
Affinity DataKi: 7.5nMAssay Description:Displacement of [3H]SCH 23390 from human D5 dopamine receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetD(1B) dopamine receptor(Homo sapiens (Human))
Friedrich-Schiller-UniversitäT Jena
Curated by ChEMBL
Friedrich-Schiller-UniversitäT Jena
Curated by ChEMBL
Affinity DataKi: 7.5nMAssay Description:Binding affinity to human cloned dopamine D5 receptor expressed in HEK 293 cellsMore data for this Ligand-Target Pair
TargetD(1B) dopamine receptor(Homo sapiens (Human))
Friedrich-Schiller-UniversitäT Jena
Curated by ChEMBL
Friedrich-Schiller-UniversitäT Jena
Curated by ChEMBL
Affinity DataKi: 7.5nMAssay Description:Binding affinity to D5 dopamine receptor by radioligand binding assayMore data for this Ligand-Target Pair
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Friedrich-Schiller-Universit£T Jena
Curated by ChEMBL
Friedrich-Schiller-Universit£T Jena
Curated by ChEMBL
Affinity DataKi: <10nMAssay Description:Antagonist activity at dopamine D1 receptor (unknown origin)More data for this Ligand-Target Pair
TargetD(1B) dopamine receptor(Homo sapiens (Human))
Friedrich-Schiller-UniversitäT Jena
Curated by ChEMBL
Friedrich-Schiller-UniversitäT Jena
Curated by ChEMBL
Affinity DataKi: <10nMAssay Description:Antagonist activity at dopamine D5 receptor (unknown origin)More data for this Ligand-Target Pair
TargetD(1B) dopamine receptor(Homo sapiens (Human))
Friedrich-Schiller-UniversitäT Jena
Curated by ChEMBL
Friedrich-Schiller-UniversitäT Jena
Curated by ChEMBL
Affinity DataKi: 12.7nMAssay Description:Inhibition of D5 dopamine receptor in HEK 293 cells by intracellular calcium assayMore data for this Ligand-Target Pair
TargetD(1B) dopamine receptor(Homo sapiens (Human))
Friedrich-Schiller-UniversitäT Jena
Curated by ChEMBL
Friedrich-Schiller-UniversitäT Jena
Curated by ChEMBL
Affinity DataKi: 12.7nMAssay Description:Activity at human D5 dopamine receptor expressed in HEK293 cells by calcium fluorescence assayMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Schiller-UniversitäT Jena
Curated by ChEMBL
Friedrich-Schiller-UniversitäT Jena
Curated by ChEMBL
Affinity DataKi: 19nMAssay Description:Activity at human D2L dopamine receptor expressed in HEK293 cells by calcium fluorescence assayMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Schiller-UniversitäT Jena
Curated by ChEMBL
Friedrich-Schiller-UniversitäT Jena
Curated by ChEMBL
Affinity DataKi: 19nMAssay Description:Inhibition of D2L dopamine receptor in HEK 293 cells by intracellular calcium assayMore data for this Ligand-Target Pair
TargetD(3) dopamine receptor(Homo sapiens (Human))
Friedrich-Schiller-UniversitäT Jena
Curated by ChEMBL
Friedrich-Schiller-UniversitäT Jena
Curated by ChEMBL
Affinity DataKi: 25.9nMAssay Description:Displacement of [3H]spiperone from human D3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetD(3) dopamine receptor(Homo sapiens (Human))
Friedrich-Schiller-UniversitäT Jena
Curated by ChEMBL
Friedrich-Schiller-UniversitäT Jena
Curated by ChEMBL
Affinity DataKi: 40.3nMAssay Description:Binding affinity to human cloned dopamine D3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Schiller-UniversitäT Jena
Curated by ChEMBL
Friedrich-Schiller-UniversitäT Jena
Curated by ChEMBL
Affinity DataKi: 41.7nMAssay Description:Displacement of [3H]SCH23390 from human cloned dopamine D2L receptorMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Schiller-UniversitäT Jena
Curated by ChEMBL
Friedrich-Schiller-UniversitäT Jena
Curated by ChEMBL
Affinity DataKi: 44.5nMAssay Description:Displacement of [3H]spiperone from human cloned dopamine D2L receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Schiller-UniversitäT Jena
Curated by ChEMBL
Friedrich-Schiller-UniversitäT Jena
Curated by ChEMBL
Affinity DataKi: 44.5nMAssay Description:Displacement of [3H]spiperone from human D2L dopamine receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Schiller-UniversitäT Jena
Curated by ChEMBL
Friedrich-Schiller-UniversitäT Jena
Curated by ChEMBL
Affinity DataKi: 44.7nMAssay Description:Displacement of [3H]spiperone from D2L dopamine receptorMore data for this Ligand-Target Pair
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Friedrich-Schiller-Universit£T Jena
Curated by ChEMBL
Friedrich-Schiller-Universit£T Jena
Curated by ChEMBL
Affinity DataKi: 60.4nMAssay Description:Activity at human D1 dopamine receptor expressed in HEK293 cells by calcium fluorescence assayMore data for this Ligand-Target Pair
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Friedrich-Schiller-Universit£T Jena
Curated by ChEMBL
Friedrich-Schiller-Universit£T Jena
Curated by ChEMBL
Affinity DataKi: 60.4nMAssay Description:Inhibition of D1 dopamine receptor in HEK 293 cells by intracellular calcium assayMore data for this Ligand-Target Pair
TargetD(4) dopamine receptor(Homo sapiens (Human))
Friedrich-Schiller-UniversitäT Jena
Curated by ChEMBL
Friedrich-Schiller-UniversitäT Jena
Curated by ChEMBL
Affinity DataKi: 108nMAssay Description:Displacement of [3H]spiperone from human D4 dopamine receptor expressed in CHO cellsMore data for this Ligand-Target Pair