Compile Data Set for Download or QSAR
maximum 50k data
Found 3 of ki for monomerid = 50389025
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Institut F£R Pharmazeutische Und Medizinische Chemie Der Westf£Lischen Wilhelms-Universit£T M£Nster

Curated by ChEMBL
LigandPNGBDBM50389025(CHEMBL2064198)
Affinity DataKi:  0.310nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma 1 receptor in guinea pig brain cortex membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Institut F£R Pharmazeutische Und Medizinische Chemie Der Westf£Lischen Wilhelms-Universit£T M£Nster

Curated by ChEMBL
LigandPNGBDBM50389025(CHEMBL2064198)
Affinity DataKi:  0.310nMAssay Description:Displacement of [3H]-(+)pentazocine from guinea pig brain sigma 1-type opioid receptor after 120 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Institut F£R Pharmazeutische Und Medizinische Chemie Der Universit£T M£Nster

Curated by ChEMBL
LigandPNGBDBM50389025(CHEMBL2064198)
Affinity DataKi:  2.10nMAssay Description:Binding affinity to human sigma 1-type opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed