Compile Data Set for Download or QSAR
maximum 50k data
Found 3 of ki for monomerid = 50437949
TargetCalpain-1 catalytic subunit(Sus scrofa (pig))
The Trustees of Columbia University In The City of New York

US Patent
LigandPNGBDBM50437949(CHEMBL2408918 | US9403843, 34)
Affinity DataKi:  3.50E+3nM ΔG°:  -31.7kJ/molepH: 7.6 T: 2°CAssay Description:Full length porcine calpain (156 nM), or papain (236 pM) was added to a solution of 100 mM NaCl, 50 mM HEPES, pH 7.6, 1 mM TCEP, 30 μM Suc-LLVY-AM...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCalpain-1 catalytic subunit(Sus scrofa (pig))
The Trustees of Columbia University In The City of New York

US Patent
LigandPNGBDBM50437949(CHEMBL2408918 | US9403843, 34)
Affinity DataKi:  3.53E+3nMAssay Description:Inhibition of pig full length Cal1 after using SucLLVYAMC as substrate by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPapain(Carica papaya)
University Of Illinois College Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50437949(CHEMBL2408918 | US9403843, 34)
Affinity DataKi:  9.70E+3nMAssay Description:Inhibition of papain after using SucLLVYAMC as substrate by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed