Compile Data Set for Download or QSAR
maximum 50k data
Found 3 of ki for monomerid = 936
TargetDimer of Gag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Sandoz Forschungsinstitut Ges.M.B.H.

LigandPNGBDBM936(5PhBuCOOH deriv. | Statine deriv. 16 | Tle-Val-Sta...)
Affinity DataKi:  7.40nM ΔG°:  -48.3kJ/molepH: 6.25 T: 2°CAssay Description:Enzymatic activity was measured by following cleavage of the substrate H-Lys-Ala-Arg-Val-Leu-pNph-Glu-Ala-Nle-NH2. Products of the cleavage reaction ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Sandoz Forschungsinstitut Ges.M.B.H.

Curated by ChEMBL
LigandPNGBDBM936(5PhBuCOOH deriv. | Statine deriv. 16 | Tle-Val-Sta...)
Affinity DataKi:  7.41nMAssay Description:Inhibitory activity was determined against HIV type 1 proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDimer of Gag-Pol polyprotein [514-612](Human immunodeficiency virus type 2)
Sandoz Forschungsinstitut Ges.M.B.H.

LigandPNGBDBM936(5PhBuCOOH deriv. | Statine deriv. 16 | Tle-Val-Sta...)
Affinity DataKi:  39nM ΔG°:  -44.0kJ/molepH: 4.7 T: 2°CAssay Description:Enzymatic activity was measured by following cleavage of the substrate H-Lys-Ala-Arg-Val-Leu-pNph-Glu-Ala-Nle-NH2. Products of the cleavage reaction ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed