Compile Data Set for Download or QSAR
maximum 50k data
Found 507 Enz. Inhib. hit(s) with all data for entry = 9100
TargetAlpha-1A adrenergic receptor(CALF)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50328480(1-Methyl-4-(8-(1-methyl-1H-pyrazol-5-yl)-10,11-dih...)
Affinity DataKi:  0.410nMAssay Description:Displacement of [3H]prozosin from bovine cloned alpha1a receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(CALF)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50328503((R)-N-((11-(4-methylpiperazin-1-yl)-10,11-dihydrod...)
Affinity DataKi:  0.420nMAssay Description:Displacement of [3H]prozosin from bovine cloned alpha1a receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(C.H.O.)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50007567(1-(8-Chloro-10,11-dihydro-dibenzo[b,f]thiepin-10-y...)
Affinity DataKi:  0.420nMAssay Description:Displacement of [3H]prozosin from hamster cloned alpha1b receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(C.H.O.)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50328504((S)-N-((11-(4-methylpiperazin-1-yl)-10,11-dihydrod...)
Affinity DataKi:  0.420nMAssay Description:Displacement of [3H]prozosin from hamster cloned alpha1b receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(CALF)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50328505((R)-N-((11-(4-methylpiperazin-1-yl)-10,11-dihydrod...)
Affinity DataKi:  0.430nMAssay Description:Displacement of [3H]prozosin from bovine cloned alpha1a receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50328478(1-Methyl-4-(8-(2-methyl-2H-tetrazol-5-yl)-10,11-di...)
Affinity DataKi:  0.440nMAssay Description:Displacement of [3H]spiperone from human cloned dopamine D2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50001786(1-(2-{4-[5-chloro-1-(4-fluorophenyl)-1H-indol-3-yl...)
Affinity DataKi:  0.450nMAssay Description:Displacement of [3H]prozosin from human cloned dopamine D2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetAlpha-1A adrenergic receptor(CALF)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50328489(1-Methyl-4-(8-phenyl-10,11-dihydrodibenzo[b,f]thie...)
Affinity DataKi:  0.5nMAssay Description:Displacement of [3H]prozosin from bovine cloned alpha1a receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Homo sapiens (Human))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50001786(1-(2-{4-[5-chloro-1-(4-fluorophenyl)-1H-indol-3-yl...)
Affinity DataKi:  0.510nMAssay Description:Displacement of [3H]prozosin from human cloned histamine H1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(CALF)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50328484(1-Methyl-4-(8-(5-methylthiophen-2-yl)-10,11-dihydr...)
Affinity DataKi:  0.520nMAssay Description:Displacement of [3H]prozosin from bovine cloned alpha1a receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(C.H.O.)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50328502(CHEMBL1259158 | N-((11-(4-Methylpiperazin-1-yl)-10...)
Affinity DataKi:  0.520nMAssay Description:Displacement of [3H]prozosin from hamster cloned alpha1b receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(CALF)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50328477(1-(8-chloro-10,11-dihydrodibenzo[b,f]thiepin-10-yl...)
Affinity DataKi:  0.520nMAssay Description:Displacement of [3H]prozosin from bovine cloned alpha1a receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(C.H.O.)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50328476(1-(2-(4-(1-(4-fluorophenyl)-5-((2-methyl-2H-tetraz...)
Affinity DataKi:  0.560nMAssay Description:Displacement of [3H]prozosin from hamster cloned alpha1b receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(C.H.O.)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM22872(1-(3-chloro-5,6-dihydrobenzo[b][1]benzothiepin-5-y...)
Affinity DataKi:  0.560nMAssay Description:Displacement of [3H]prozosin from hamster cloned alpha1b receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM22872(1-(3-chloro-5,6-dihydrobenzo[b][1]benzothiepin-5-y...)
Affinity DataKi:  0.570nMAssay Description:Displacement of [3H]prozosin from human cloned 5HT2C receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Rattus norvegicus (Rat))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50328485(1-Methyl-4-(8-(pyridin-2-yl)-10,11-dihydrodibenzo[...)
Affinity DataKi:  0.610nMAssay Description:Displacement of [3H]prozosin from rat cloned alpha1d receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50328486(1-Methyl-4-(8-(pyridin-3-yl)-10,11-dihydrodibenzo[...)
Affinity DataKi:  0.620nMAssay Description:Displacement of [3H]prozosin from human cloned dopamine D2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Rattus norvegicus (Rat))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50328505((R)-N-((11-(4-methylpiperazin-1-yl)-10,11-dihydrod...)
Affinity DataKi:  0.640nMAssay Description:Displacement of [3H]prozosin from rat cloned alpha1d receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Rattus norvegicus (Rat))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50328487(1-Methyl-4-(8-(pyridin-4-yl)-10,11-dihydrodibenzo[...)
Affinity DataKi:  0.660nMAssay Description:Displacement of [3H]prozosin from rat cloned alpha1d receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(CALF)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM22872(1-(3-chloro-5,6-dihydrobenzo[b][1]benzothiepin-5-y...)
Affinity DataKi:  0.660nMAssay Description:Displacement of [3H]prozosin from bovine cloned alpha1a receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(CALF)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50328476(1-(2-(4-(1-(4-fluorophenyl)-5-((2-methyl-2H-tetraz...)
Affinity DataKi:  0.660nMAssay Description:Displacement of [3H]prozosin from bovine cloned alpha1a receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Rattus norvegicus (Rat))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50001786(1-(2-{4-[5-chloro-1-(4-fluorophenyl)-1H-indol-3-yl...)
Affinity DataKi:  0.660nMAssay Description:Displacement of [3H]prozosin from rat cloned alpha1d receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM22872(1-(3-chloro-5,6-dihydrobenzo[b][1]benzothiepin-5-y...)
Affinity DataKi:  0.670nMAssay Description:Displacement of [3H]prozosin from human cloned dopamine D2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(CALF)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50328475(CHEMBL1259187 | N-((1-(4-fluorophenyl)-3-(1-(2-(2-...)
Affinity DataKi:  0.680nMAssay Description:Displacement of [3H]prozosin from bovine cloned alpha1a receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Rattus norvegicus (Rat))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50328474(1-(2-(4-(5-(aminomethyl)-1-(4-fluorophenyl)-1H-ind...)
Affinity DataKi:  0.690nMAssay Description:Displacement of [3H]prozosin from rat cloned alpha1d receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(CALF)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50007567(1-(8-Chloro-10,11-dihydro-dibenzo[b,f]thiepin-10-y...)
Affinity DataKi:  0.700nMAssay Description:Displacement of [3H]prozosin from bovine cloned alpha1a receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(C.H.O.)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50328484(1-Methyl-4-(8-(5-methylthiophen-2-yl)-10,11-dihydr...)
Affinity DataKi:  0.720nMAssay Description:Displacement of [3H]prozosin from hamster cloned alpha1b receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50328488(5-(11-(4-Methylpiperazin-1-yl)-10,11-dihydrodibenz...)
Affinity DataKi:  0.730nMAssay Description:Displacement of [3H]prozosin from human cloned dopamine D2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Rattus norvegicus (Rat))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM22872(1-(3-chloro-5,6-dihydrobenzo[b][1]benzothiepin-5-y...)
Affinity DataKi:  0.770nMAssay Description:Displacement of [3H]prozosin from rat cloned alpha1d receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Rattus norvegicus (Rat))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50328476(1-(2-(4-(1-(4-fluorophenyl)-5-((2-methyl-2H-tetraz...)
Affinity DataKi:  0.770nMAssay Description:Displacement of [3H]prozosin from rat cloned alpha1d receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(C.H.O.)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50328492(1-Methyl-4-(8-p-tolyl-10,11-dihydrodibenzo[b,f]thi...)
Affinity DataKi:  0.820nMAssay Description:Displacement of [3H]prozosin from hamster cloned alpha1b receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50328480(1-Methyl-4-(8-(1-methyl-1H-pyrazol-5-yl)-10,11-dih...)
Affinity DataKi:  0.860nMAssay Description:Displacement of [3H]prozosin from human cloned dopamine D2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(CALF)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50328490(1-Methyl-4-(8-o-tolyl-10,11-dihydrodibenzo[b,f]thi...)
Affinity DataKi:  0.870nMAssay Description:Displacement of [3H]prozosin from bovine cloned alpha1a receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(C.H.O.)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50328503((R)-N-((11-(4-methylpiperazin-1-yl)-10,11-dihydrod...)
Affinity DataKi:  0.900nMAssay Description:Displacement of [3H]prozosin from hamster cloned alpha1b receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(C.H.O.)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50328491(1-Methyl-4-(8-m-tolyl-10,11-dihydrodibenzo[b,f]thi...)
Affinity DataKi:  0.950nMAssay Description:Displacement of [3H]prozosin from hamster cloned alpha1b receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(CALF)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50328491(1-Methyl-4-(8-m-tolyl-10,11-dihydrodibenzo[b,f]thi...)
Affinity DataKi:  0.950nMAssay Description:Displacement of [3H]prozosin from bovine cloned alpha1a receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Rattus norvegicus (Rat))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50328480(1-Methyl-4-(8-(1-methyl-1H-pyrazol-5-yl)-10,11-dih...)
Affinity DataKi:  0.970nMAssay Description:Displacement of [3H]prozosin from rat cloned alpha1d receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Rattus norvegicus (Rat))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50328504((S)-N-((11-(4-methylpiperazin-1-yl)-10,11-dihydrod...)
Affinity DataKi:  0.980nMAssay Description:Displacement of [3H]prozosin from rat cloned alpha1d receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Rattus norvegicus (Rat))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50328486(1-Methyl-4-(8-(pyridin-3-yl)-10,11-dihydrodibenzo[...)
Affinity DataKi:  1nMAssay Description:Displacement of [3H]prozosin from rat cloned alpha1d receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Rattus norvegicus (Rat))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50328478(1-Methyl-4-(8-(2-methyl-2H-tetrazol-5-yl)-10,11-di...)
Affinity DataKi:  1nMAssay Description:Displacement of [3H]prozosin from rat cloned alpha1d receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(CALF)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50328494(1-(8-(2,5-Dimethylphenyl)-10,11-dihydrodibenzo[b,f...)
Affinity DataKi:  1nMAssay Description:Displacement of [3H]prozosin from bovine cloned alpha1a receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50007568(1-((S)-8-Chloro-10,11-dihydro-dibenzo[b,f]thiepin-...)
Affinity DataKi:  1.10nMAssay Description:Displacement of [3H]prozosin from human cloned dopamine D2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50328487(1-Methyl-4-(8-(pyridin-4-yl)-10,11-dihydrodibenzo[...)
Affinity DataKi:  1.10nMAssay Description:Displacement of [3H]prozosin from human cloned dopamine D2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(C.H.O.)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50328474(1-(2-(4-(5-(aminomethyl)-1-(4-fluorophenyl)-1H-ind...)
Affinity DataKi:  1.10nMAssay Description:Displacement of [3H]prozosin from hamster cloned alpha1b receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(C.H.O.)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50122815(1-(2-{4-[1-(4-Fluoro-phenyl)-5-(2-methyl-2H-tetraz...)
Affinity DataKi:  1.10nMAssay Description:Displacement of [3H]prozosin from hamster cloned alpha1b receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(CALF)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50328492(1-Methyl-4-(8-p-tolyl-10,11-dihydrodibenzo[b,f]thi...)
Affinity DataKi:  1.10nMAssay Description:Displacement of [3H]prozosin from bovine cloned alpha1a receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(C.H.O.)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50328493(1-(8-(2,3-Dimethylphenyl)-10,11-dihydrodibenzo[b,f...)
Affinity DataKi:  1.20nMAssay Description:Displacement of [3H]prozosin from hamster cloned alpha1b receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(C.H.O.)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50328483(1-Methyl-4-(8-(1-methyl-1H-1,2,4-triazol-3-yl)-10,...)
Affinity DataKi:  1.20nMAssay Description:Displacement of [3H]prozosin from hamster cloned alpha1b receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(CALF)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50328502(CHEMBL1259158 | N-((11-(4-Methylpiperazin-1-yl)-10...)
Affinity DataKi:  1.30nMAssay Description:Displacement of [3H]prozosin from bovine cloned alpha1a receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Rattus norvegicus (Rat))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50328482(1-Methyl-4-(8-(1-methyl-1H-pyrazol-4-yl)-10,11-dih...)
Affinity DataKi:  1.40nMAssay Description:Displacement of [3H]prozosin from rat cloned alpha1d receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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