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Targets 377▿
Tyrosine-protein kinase ABL1 15
Epidermal growth factor receptor 12
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform 10
Mast/stem cell growth factor receptor Kit 8
Receptor-type tyrosine-protein kinase FLT3 7
Proto-oncogene tyrosine-protein kinase receptor Ret 4
Hepatocyte growth factor receptor 3
Ephrin type-A receptor 6 2
Tyrosine-protein kinase JAK1 2
Ribosomal protein S6 kinase alpha-6 2
Cyclin-dependent kinase 4 2
Ribosomal protein S6 kinase alpha-4 2
Ribosomal protein S6 kinase alpha-5 2
Ribosomal protein S6 kinase alpha-2 2
Ribosomal protein S6 kinase alpha-1 2
Leucine-rich repeat serine/threonine-protein kinase 2 2
Non-receptor tyrosine-protein kinase TYK2 2
Mitogen-activated protein kinase 14 2
Serine/threonine-protein kinase B-raf 2
Fibroblast growth factor receptor 3 2
Tyrosine-protein kinase Tec 1
BMP-2-inducible protein kinase 1
Rhodopsin kinase GRK1 1
Cyclin-dependent kinase 11B 1
Cyclin-dependent kinase 11A 1
Uncharacterized serine/threonine-protein kinase SBK3 1
LIM domain kinase 1 1
LIM domain kinase 2 1
ALK tyrosine kinase receptor 1
NUAK family SNF1-like kinase 2 1
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform 1
Glycogen synthase kinase-3 beta 1
Calcium/calmodulin-dependent protein kinase type 1 1
Protein kinase C iota type 1
NUAK family SNF1-like kinase 1 1
Transient receptor potential cation channel subfamily M member 6 1
AP2-associated protein kinase 1 1
Calcium/calmodulin-dependent protein kinase type II subunit beta 1
Phosphorylase b kinase gamma catalytic chain, skeletal muscle/heart isoform 1
Serine/threonine-protein kinase PAK 1 1
Protein kinase C theta type 1
Serine/threonine-protein kinase PAK 2 1
Serine/threonine-protein kinase PAK 3 1
Dual specificity mitogen-activated protein kinase kinase 2 1
Serine/threonine-protein kinase PAK 4 1
Phosphatidylinositol 5-phosphate 4-kinase type-2 beta 1
Serine/threonine-protein kinase tousled-like 2 1
Dual specificity mitogen-activated protein kinase kinase 3 1
Serine/threonine-protein kinase PAK 5 1
Serine/threonine-protein kinase PAK 6 1
Serine/threonine-protein kinase tousled-like 1 1
Tyrosine-protein kinase JAK3 1
Tyrosine-protein kinase JAK2 1
Dual specificity mitogen-activated protein kinase kinase 1 1
Dual specificity mitogen-activated protein kinase kinase 6 1
Dual specificity mitogen-activated protein kinase kinase 7 1
Dual specificity mitogen-activated protein kinase kinase 4 1
Dual specificity mitogen-activated protein kinase kinase 5 1
Tyrosine-protein kinase ZAP-70 1
Casein kinase I isoform gamma-3 1
Casein kinase I isoform gamma-2 1
Serine/threonine-protein kinase Sgk3 1
Casein kinase I isoform epsilon 1
Casein kinase I isoform gamma-1 1
Myosin light chain kinase 3 1
Ephrin type-A receptor 1 1
Ephrin type-A receptor 3 1
Ephrin type-A receptor 2 1
Ephrin type-A receptor 5 1
Tyrosine-protein kinase BTK 1
Ephrin type-A receptor 4 1
Tyrosine-protein kinase receptor UFO 1
Insulin-like growth factor 1 receptor 1
Activin receptor type-1 1
Myosin light chain kinase 2, skeletal/cardiac muscle 1
Tyrosine-protein kinase Srms 1
Wee1-like protein kinase 1
Serine/threonine-protein kinase/endoribonuclease IRE1 1
Serine/threonine-protein kinase MAK 1
Phosphatidylinositol 3-kinase C2 domain-containing subunit gamma 1
Ankyrin repeat and protein kinase domain-containing protein 1 1
Tyrosine-protein kinase Lyn 1
Focal adhesion kinase 1 1
Phosphatidylinositol 4-phosphate 5-kinase type-1 gamma 1
Cyclin-dependent kinase 2 1
Tyrosine-protein kinase TXK 1
Rhodopsin kinase GRK7 1
Ephrin type-A receptor 8 1
Phosphatidylinositol 4-kinase beta 1
Death-associated protein kinase 2 1
Death-associated protein kinase 1 1
Serine/threonine-protein kinase D2 1
Serine/threonine-protein kinase D3 1
TGF-beta receptor type-2 1
Serine/threonine-protein kinase D1 1
Dual specificity tyrosine-phosphorylation-regulated kinase 1B 1
Dual serine/threonine and tyrosine protein kinase 1
Dual specificity tyrosine-phosphorylation-regulated kinase 1A 1
Death-associated protein kinase 3 1
Cyclin-dependent kinase 9 1
Serine/threonine-protein kinase pim-3 1
Cyclin-dependent kinase 8 1
Cyclin-dependent kinase 7 1
Serine/threonine-protein kinase pim-1 1
Cyclin-dependent kinase 5 1
Serine/threonine-protein kinase pim-2 1
Serine/threonine-protein kinase 38 1
Serine/threonine-protein kinase 35 1
Cyclin-dependent kinase 3 1
Serine/threonine-protein kinase 36 1
Cyclin-dependent kinase 16 1
Testis-specific serine/threonine-protein kinase 1 1
Protein kinase C epsilon type 1
Cyclin-dependent kinase 17 1
Bone morphogenetic protein receptor type-2 1
Cyclin-dependent kinase 19 1
Cyclin-dependent kinase 2 homolog 1
Protein-tyrosine kinase 6 1
Casein kinase II subunit alpha 1
Cyclin-dependent kinase 13 1
Cyclin-dependent kinase 14 1
Cyclin-dependent kinase 15 1
Leukocyte tyrosine kinase receptor 1
Cytoplasmic tyrosine-protein kinase BMX 1
Tyrosine-protein kinase ABL2 1
Atypical kinase COQ8B, mitochondrial 1
Microtubule-associated serine/threonine-protein kinase 1 1
Calcium/calmodulin-dependent protein kinase type II subunit alpha 1
cGMP-dependent protein kinase 2 1
Rho-associated protein kinase 2 1
cGMP-dependent protein kinase 1 1
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform 1
Rho-associated protein kinase 1 1
Serine/threonine-protein kinase ULK1 1
Serine/threonine-protein kinase SIK2 1
Tyrosine-protein kinase Fes/Fps 1
Serine/threonine-protein kinase SIK1 1
Serine/threonine-protein kinase ULK2 1
Serine/threonine-protein kinase ULK3 1
3-phosphoinositide-dependent protein kinase 1 1
Mitogen-activated protein kinase 1 1
Serine/threonine-protein kinase 3 1
Mitogen-activated protein kinase 3 1
Discoidin domain-containing receptor 2 1
Mitogen-activated protein kinase 4 1
Serine/threonine-protein kinase 4 1
SRSF protein kinase 3 1
Mitogen-activated protein kinase 9 1
SRSF protein kinase 2 1
Mitogen-activated protein kinase 6 1
Mitogen-activated protein kinase 7 1
Calcium/calmodulin-dependent protein kinase type IV 1
Mitogen-activated protein kinase 8 1
Tyrosine-protein kinase SYK 1
Serine/threonine-protein kinase TBK1 1
Serine/threonine-protein kinase RIO1 1
Serine/threonine-protein kinase LATS1 1
Serine/threonine-protein kinase RIO3 1
Serine/threonine-protein kinase 32B 1
Serine/threonine-protein kinase RIO2 1
Serine/threonine-protein kinase 32A 1
Serine/threonine-protein kinase 32C 1
Vascular endothelial growth factor receptor 2 1
Insulin receptor 1
Tyrosine-protein kinase HCK 1
Vascular endothelial growth factor receptor 3 1
Vascular endothelial growth factor receptor 1 1
Serine/threonine-protein kinase PLK1 1
Serine/threonine-protein kinase PLK2 1
Insulin receptor-related protein 1
Inhibitor of nuclear factor kappa-B kinase subunit beta 1
Serine/threonine-protein kinase NIM1 1
Serine/threonine-protein kinase PLK3 1
Serine/threonine-protein kinase PLK4 1
Tyrosine-protein kinase receptor TYRO3 1
Wee1-like protein kinase 2 1
Serine/threonine-protein kinase BRSK1 1
Serine/threonine-protein kinase LATS2 1
cAMP-dependent protein kinase catalytic subunit alpha 1
Citron Rho-interacting kinase 1
Platelet-derived growth factor receptor alpha 1
Serine/threonine-protein kinase BRSK2 1
Serine/threonine-protein kinase Chk2 1
Serine/threonine-protein kinase Chk1 1
cAMP-dependent protein kinase catalytic subunit PRKX 1
SRSF protein kinase 1 1
Tyrosine-protein kinase Yes 1
Serine/threonine-protein kinase MRCK beta 1
Serine/threonine-protein kinase MRCK gamma 1
Casein kinase II subunit alpha' 1
Dual specificity tyrosine-phosphorylation-regulated kinase 2 1
Serine/threonine-protein kinase STK11 1
Cyclin-G-associated kinase 1
Peripheral plasma membrane protein CASK 1
Receptor tyrosine-protein kinase erbB-4 1
Receptor tyrosine-protein kinase erbB-2 1
Tyrosine-protein kinase FRK 1
Receptor tyrosine-protein kinase erbB-3 1
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform 1
Serine/threonine-protein kinase Nek9 1
Serine/threonine-protein kinase Nek7 1
Glycogen synthase kinase-3 alpha 1
Serine/threonine-protein kinase Nek6 1
Serine/threonine-protein kinase Nek5 1
Serine/threonine-protein kinase Nek4 1
Serine/threonine-protein kinase Nek3 1
Serine/threonine-protein kinase Nek2 1
Serine/threonine-protein kinase receptor R3 1
Serine/threonine-protein kinase Nek1 1
Macrophage-stimulating protein receptor 1
Cyclin-dependent kinase-like 3 1
Serine/threonine-protein kinase SIK3 [59-1321] 1
Cyclin-dependent kinase-like 2 1
MAP/microtubule affinity-regulating kinase 3 1
Homeodomain-interacting protein kinase 4 1
Homeodomain-interacting protein kinase 3 1
MAP kinase-interacting serine/threonine-protein kinase 2 1
MAP kinase-interacting serine/threonine-protein kinase 1 1
Cyclin-dependent kinase-like 5 1
Membrane-associated tyrosine- and threonine-specific cdc2-inhibitory kinase 1
Serine/threonine-protein kinase 10 1
MAP/microtubule affinity-regulating kinase 4 1
Serine/threonine-protein kinase 38-like 1
Dual specificity protein kinase TTK 1
Myosin-IIIb 1
Serine/threonine-protein kinase Nek11 1
Myosin-IIIa 1
Eukaryotic translation initiation factor 2-alpha kinase 1 1
Serine/threonine-protein kinase mTOR 1
Tyrosine-protein kinase ITK/TSK 1
Myotonin-protein kinase 1
Protein kinase C eta type 1
Bone morphogenetic protein receptor type-1B 1
Bone morphogenetic protein receptor type-1A 1
Tyrosine-protein kinase Blk 1
Receptor-interacting serine/threonine-protein kinase 1 1
Serine/threonine-protein kinase 16 1
Receptor-interacting serine/threonine-protein kinase 2 1
SNF-related serine/threonine-protein kinase 1
Non-receptor tyrosine-protein kinase TNK1 1
Inhibitor of nuclear factor kappa-B kinase subunit epsilon 1
Serine/threonine-protein kinase NLK 1
Homeodomain-interacting protein kinase 2 1
Homeodomain-interacting protein kinase 1 1
Receptor-interacting serine/threonine-protein kinase 4 1
Ribosomal protein S6 kinase beta-1 1
Serine/threonine-protein kinase OSR1 1
Casein kinase I isoform delta 1
Cyclin-dependent kinase 18 [3-474] 1
RAF proto-oncogene serine/threonine-protein kinase 1
Serine/threonine-protein kinase 26 1
Serine/threonine-protein kinase 24 1
Serine/threonine-protein kinase 25 1
Dual specificity testis-specific protein kinase 1 1
Ephrin type-B receptor 3 1
Serine/threonine-protein kinase 33 1
Ephrin type-B receptor 4 1
Ephrin type-B receptor 1 1
Serine/threonine-protein kinase SBK1 1
Ephrin type-B receptor 2 1
Activated CDC42 kinase 1 1
MAP kinase-activated protein kinase 2 1
Ephrin type-B receptor 6 1
Platelet-derived growth factor receptor beta 1
Epithelial discoidin domain-containing receptor 1 1
MAP kinase-activated protein kinase 5 1
STE20/SPS1-related proline-alanine-rich protein kinase 1
Muscle, skeletal receptor tyrosine-protein kinase 1
Tyrosine-protein kinase Fer 1
Calcium-dependent protein kinase 1 1
Tyrosine-protein kinase receptor Tie-1 1
5'-AMP-activated protein kinase catalytic subunit alpha-2 1
Calcium/calmodulin-dependent protein kinase type II subunit delta 1
Proto-oncogene tyrosine-protein kinase ROS 1
Phosphatidylinositol 5-phosphate 4-kinase type-2 gamma 1
Serine/threonine-protein kinase TAO1 1
Serine/threonine-protein kinase DCLK1 1
Calcium/calmodulin-dependent protein kinase kinase 1 1
Serine/threonine-protein kinase PknB 1
Serine/threonine-protein kinase DCLK2 1
Serine/threonine-protein kinase TAO3 1
Serine/threonine-protein kinase PRP4 homolog 1
Calcium/calmodulin-dependent protein kinase kinase 2 1
Serine/threonine-protein kinase TAO2 1
Serine/threonine-protein kinase DCLK3 1
Serine/threonine-protein kinase TNNI3K 1
Interferon-induced, double-stranded RNA-activated protein kinase 1
Angiopoietin-1 receptor 1
Mitogen-activated protein kinase kinase kinase kinase 2 1
Cyclin-dependent kinase-like 1 [2-358] 1
Mitogen-activated protein kinase kinase kinase kinase 3 1
Mitogen-activated protein kinase kinase kinase kinase 1 1
Serine/threonine-protein kinase MRCK alpha 1
Casein kinase I isoform alpha-like 1
Mitogen-activated protein kinase kinase kinase kinase 4 1
Mitogen-activated protein kinase kinase kinase kinase 5 1
Mitogen-activated protein kinase 15 1
5'-AMP-activated protein kinase catalytic subunit alpha-1 1
Activin receptor type-1B 1
Interleukin-1 receptor-associated kinase 4 1
Myosin light chain kinase family member 4 1
Mitogen-activated protein kinase kinase kinase 9 1
Serine/threonine-protein kinase VRK2 1
Mitogen-activated protein kinase kinase kinase 6 1
RAC-gamma serine/threonine-protein kinase 1
Mitogen-activated protein kinase kinase kinase 5 1
Interleukin-1 receptor-associated kinase 1 1
Mitogen-activated protein kinase kinase kinase 7 1
Interleukin-1 receptor-associated kinase 3 1
Mitogen-activated protein kinase kinase kinase 2 1
Mitogen-activated protein kinase kinase kinase 1 1
Mitogen-activated protein kinase kinase kinase 4 1
Mitogen-activated protein kinase kinase kinase 3 1
Serine/threonine-protein kinase ICK 1
RAC-alpha serine/threonine-protein kinase 1
Megakaryocyte-associated tyrosine-protein kinase 1
Proto-oncogene tyrosine-protein kinase Src 1
Activin receptor type-2B 1
Myosin light chain kinase, smooth muscle 1
Activin receptor type-2A 1
BDNF/NT-3 growth factors receptor 1
Serine/threonine-protein kinase 17A 1
Tyrosine-protein kinase Lck 1
Serine/threonine-protein kinase 17B 1
Mitogen-activated protein kinase kinase kinase 19 1
Dual specificity protein kinase CLK1 1
Protein kinase C delta type 1
Mitogen-activated protein kinase kinase kinase 15 1
NT-3 growth factor receptor 1
G protein-coupled receptor kinase 4 1
Dual specificity protein kinase CLK4 1
Dual specificity protein kinase CLK3 1
Dual specificity protein kinase CLK2 1
High affinity nerve growth factor receptor 1
Protein-tyrosine kinase 2-beta 1
Tyrosine-protein kinase Mer 1
Serine/threonine-protein kinase N2 1
cAMP-dependent protein kinase catalytic subunit beta 1
Calcium/calmodulin-dependent protein kinase type II subunit gamma 1
Serine/threonine-protein kinase N1 1
Ribosomal protein S6 kinase alpha-3 1
Phosphorylase b kinase gamma catalytic chain, liver/testis isoform 1
Calcium/calmodulin-dependent protein kinase type 1D 1
STE20-like serine/threonine-protein kinase 1
Calcium/calmodulin-dependent protein kinase type 1G 1
Hormonally up-regulated neu tumor-associated kinase 1
Fibroblast growth factor receptor 4 1
Tyrosine-protein kinase Fgr 1
Aurora kinase B 1
Phosphatidylinositol 4-phosphate 3-kinase C2 domain-containing subunit beta 1
Aurora kinase A 1
Mitogen-activated protein kinase kinase kinase 20 1
Fibroblast growth factor receptor 1 1
Fibroblast growth factor receptor 2 1
Atypical kinase COQ8A, mitochondrial 1
Aurora kinase C 1
Mitogen-activated protein kinase 13 1
Inhibitor of nuclear factor kappa-B kinase subunit alpha 1
Mitogen-activated protein kinase 12 1
Mitogen-activated protein kinase 11 1
Phosphatidylinositol 4-phosphate 5-kinase type-1 alpha 1
RAC-beta serine/threonine-protein kinase 1
Mitogen-activated protein kinase 10 1
Casein kinase I isoform alpha 1
Misshapen-like kinase 1 1
Tyrosine-protein kinase Fyn 1
Tyrosine-protein kinase CSK 1
Macrophage colony-stimulating factor 1 receptor 1
eIF-2-alpha kinase GCN2 1
Maternal embryonic leucine zipper kinase 1
Serine/threonine-protein kinase MARK1 1
Serine/threonine-protein kinase MARK2 1
TRAF2 and NCK-interacting protein kinase 1
Mitogen-activated protein kinase kinase kinase 12 1
Mitogen-activated protein kinase kinase kinase 13 1
Mitogen-activated protein kinase kinase kinase 10 1
Mitogen-activated protein kinase kinase kinase 11 1
...
Publications 1▿
Nat Biotechnol 29: 1046 -51 (2011) 442
Institutions 1▿
Affinity: 0.093 to 1.0E+4 nM▿
Xtal structures: 0 Docked structures: 0 Catalog Cmpds: 0