Affinity DataEC50: 0.0800nMAssay Description:Transcriptional activation in CV-1 cells expressing retinoid X receptor RXR gammaMore data for this Ligand-Target Pair
TargetRetinoic acid receptor RXR-alpha/RXR-beta/RXR-gamma(Homo sapiens (Human))
Tohoku Pharmaceutical University
Curated by ChEMBL
Tohoku Pharmaceutical University
Curated by ChEMBL
Affinity DataEC50: 0.130nMAssay Description:Agonist activity at RXR (unknown origin) in presence of RAR agonist Am80More data for this Ligand-Target Pair
TargetRetinoic acid receptor RXR-alpha/RXR-beta/RXR-gamma(Homo sapiens (Human))
Tohoku Pharmaceutical University
Curated by ChEMBL
Tohoku Pharmaceutical University
Curated by ChEMBL
Affinity DataEC50: 0.140nMAssay Description:Agonist activity at RXR (unknown origin) in presence of RAR agonist Am80More data for this Ligand-Target Pair
Affinity DataEC50: 1nMAssay Description:Compound was tested for functional activity in CV-1 cells transfected with an expression vector for retinoid X receptor gamma using transactivation a...More data for this Ligand-Target Pair
Affinity DataEC50: 2nMAssay Description:Effective concentrations against Retinoic acid receptor RXR-gammaMore data for this Ligand-Target Pair
Affinity DataEC50: 2nMAssay Description:Effective concentrations against Retinoic acid receptor RXR-gammaMore data for this Ligand-Target Pair
Affinity DataEC50: 4nMAssay Description:Agonist activity for retinoic acid receptor RXR gamma in transcriptional activation assayMore data for this Ligand-Target Pair
Affinity DataEC50: 4nMAssay Description:Transcriptional activity was evaluated in CV-1 cells transfected with expression vector for Retinoic acid receptor RXR-gammaMore data for this Ligand-Target Pair
Affinity DataEC50: 4nMAssay Description:Transcriptional activation of Retinoid X receptor RXR gammaMore data for this Ligand-Target Pair
Affinity DataEC50: 4.30nMAssay Description:Effective concentrations against Retinoic acid receptor RXR-gammaMore data for this Ligand-Target Pair
Affinity DataEC50: 4.5nMAssay Description:Transcriptional activation in CV-1 cells expressing retinoid X receptor RXR gammaMore data for this Ligand-Target Pair
Affinity DataEC50: 6nMAssay Description:Transcriptional activation in CV-1 cells expressing retinoid X receptor RXR gammaMore data for this Ligand-Target Pair
Affinity DataEC50: 7nMAssay Description:Transcriptional activity was evaluated in CV-1 cells transfected with expression vector for Retinoic acid receptor RXR-gammaMore data for this Ligand-Target Pair
Affinity DataEC50: 7nMAssay Description:Transcriptional activity was evaluated in CV-1 cells transfected with expression vector for Retinoic acid receptor RXR-gammaMore data for this Ligand-Target Pair
Affinity DataEC50: 7nMAssay Description:Transcriptional activation of Retinoid X receptor RXR gammaMore data for this Ligand-Target Pair
Affinity DataEC50: 7nMAssay Description:Transcriptional activation in CV-1 cells expressing retinoid X receptor RXR gammaMore data for this Ligand-Target Pair
TargetRetinoic acid receptor RXR-alpha/RXR-beta/RXR-gamma(Homo sapiens (Human))
Tohoku Pharmaceutical University
Curated by ChEMBL
Tohoku Pharmaceutical University
Curated by ChEMBL
Affinity DataEC50: 7.90nMAssay Description:Agonist activity at human RXR binding domain and activation domain expressed in human HCT116 cells assessed as rexinoid activity incubated for 24 hrs...More data for this Ligand-Target Pair
Affinity DataEC50: 9nMAssay Description:Transcriptional activation of Retinoid X receptor RXR gammaMore data for this Ligand-Target Pair
Affinity DataEC50: 9nMAssay Description:Transcriptional activity was evaluated in CV-1 cells transfected with expression vector for Retinoic acid receptor RXR-gammaMore data for this Ligand-Target Pair
Affinity DataEC50: 11nMAssay Description:Transcriptional activity was evaluated in CV-1 cells transfected with expression vector for Retinoic acid receptor RXR-gammaMore data for this Ligand-Target Pair
TargetRetinoic acid receptor RXR-alpha/RXR-beta/RXR-gamma(Homo sapiens (Human))
Tohoku Pharmaceutical University
Curated by ChEMBL
Tohoku Pharmaceutical University
Curated by ChEMBL
Affinity DataEC50: 14nMAssay Description:Agonist activity at human RXR binding domain and activation domain expressed in human HCT116 cells assessed as rexinoid activity incubated for 24 hrs...More data for this Ligand-Target Pair
TargetRetinoic acid receptor RXR-alpha/RXR-beta/RXR-gamma(Homo sapiens (Human))
Tohoku Pharmaceutical University
Curated by ChEMBL
Tohoku Pharmaceutical University
Curated by ChEMBL
Affinity DataEC50: 14nMAssay Description:Agonist activity at human RXR binding domain and activation domain expressed in human HCT116 cells assessed as rexinoid activity incubated for 24 hrs...More data for this Ligand-Target Pair
TargetRetinoic acid receptor RXR-alpha/RXR-beta/RXR-gamma(Homo sapiens (Human))
Tohoku Pharmaceutical University
Curated by ChEMBL
Tohoku Pharmaceutical University
Curated by ChEMBL
Affinity DataEC50: 18nMAssay Description:Agonist activity at human RXR binding domain and activation domain expressed in human HCT116 cells assessed as rexinoid activity incubated for 24 hrs...More data for this Ligand-Target Pair
Affinity DataEC50: 19nMAssay Description:Transactivation of RXRgamma in CV1 cells by cotransfection assayMore data for this Ligand-Target Pair
Affinity DataEC50: 20nMAssay Description:Transcriptional activity was evaluated in CV-1 cells transfected with expression vector for Retinoic acid receptor RXR-gammaMore data for this Ligand-Target Pair
Affinity DataEC50: 24nMAssay Description:Inhibition of [3H]-9-cis-RA binding to RXR alpha receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 25nMAssay Description:Transcriptional activation in CV-1 cells expressing retinoic acid receptor RAR gammaMore data for this Ligand-Target Pair
Affinity DataEC50: 25nMAssay Description:Agonist activity RXRgamma (unknown origin)More data for this Ligand-Target Pair
Affinity DataEC50: 25nMAssay Description:Agonist activity RXRgamma (unknown origin)More data for this Ligand-Target Pair
Affinity DataEC50: 25nMAssay Description:Agonist activity at RXRgamma (unknown origin)More data for this Ligand-Target Pair
Affinity DataEC50: 26nMAssay Description:Transcriptional activity was evaluated in CV-1 cells transfected with expression vector for Retinoic acid receptor RXR-gammaMore data for this Ligand-Target Pair
Affinity DataEC50: 28nMAssay Description:Transcriptional activity was evaluated in CV-1 cells transfected with expression vector for Retinoic acid receptor RXR-gammaMore data for this Ligand-Target Pair
Affinity DataEC50: 33nMAssay Description:Agonist activity for retinoic acid receptor RXR gamma in transcriptional activation assayMore data for this Ligand-Target Pair
Affinity DataEC50: 34nMAssay Description:Transcriptional activity was evaluated in CV-1 cells transfected with expression vector for Retinoic acid receptor RXR-gammaMore data for this Ligand-Target Pair
TargetRetinoic acid receptor RXR-alpha/RXR-beta/RXR-gamma(Homo sapiens (Human))
Tohoku Pharmaceutical University
Curated by ChEMBL
Tohoku Pharmaceutical University
Curated by ChEMBL
Affinity DataEC50: 34nMAssay Description:Agonist activity at human RXR binding domain and activation domain expressed in human HCT116 cells assessed as rexinoid activity incubated for 24 hrs...More data for this Ligand-Target Pair
Affinity DataEC50: 35nMAssay Description:Transactivation of RXRgamma in CV1 cells by cotransfection assayMore data for this Ligand-Target Pair
TargetRetinoic acid receptor RXR-alpha/RXR-beta/RXR-gamma(Homo sapiens (Human))
Tohoku Pharmaceutical University
Curated by ChEMBL
Tohoku Pharmaceutical University
Curated by ChEMBL
Affinity DataEC50: 41nMAssay Description:Agonist activity at human RXR binding domain and activation domain expressed in human HCT116 cells assessed as rexinoid activity incubated for 24 hrs...More data for this Ligand-Target Pair
Affinity DataEC50: 42nMAssay Description:Transcriptional activation of Retinoid X receptor RXR gammaMore data for this Ligand-Target Pair
Affinity DataEC50: 50nMAssay Description:Agonist activity at human RXRgamma transfected in human HEK293T cells co-expressing pFR/pRL-Luc incubated for 14 to 16 hrs by hybrid reporter gene as...More data for this Ligand-Target Pair
Affinity DataEC50: 50nMAssay Description:Transactivation of RXRgamma in CV1 cells by cotransfection assayMore data for this Ligand-Target Pair
TargetRetinoic acid receptor RXR-alpha/RXR-beta/RXR-gamma(Homo sapiens (Human))
Tohoku Pharmaceutical University
Curated by ChEMBL
Tohoku Pharmaceutical University
Curated by ChEMBL
Affinity DataEC50: 52nMAssay Description:Agonist activity at human RXR binding domain and activation domain expressed in human HCT116 cells assessed as rexinoid activity incubated for 24 hrs...More data for this Ligand-Target Pair
Affinity DataEC50: 63nMAssay Description:Transactivation of RXRgamma in CV1 cells by cotransfection assayMore data for this Ligand-Target Pair
Affinity DataEC50: 71nMAssay Description:Compound was tested for functional activity in CV-1 cells transfected with an expression vector for retinoid X receptor gamma using transactivation a...More data for this Ligand-Target Pair
Affinity DataEC50: 77nMAssay Description:Transcriptional activation in CV-1 cells expressing Retinoid X receptor RXR gammaMore data for this Ligand-Target Pair
Affinity DataEC50: 86nMAssay Description:Agonist activity for retinoic acid receptor RXR gamma in transcriptional activation assayMore data for this Ligand-Target Pair
Affinity DataEC50: 99nMAssay Description:Transcriptional activity was evaluated in CV-1 cells transfected with expression vector for Retinoic acid receptor RXR-gammaMore data for this Ligand-Target Pair
Affinity DataEC50: 100nMAssay Description:Transactivation of RXRgamma in CV1 cells by cotransfection assayMore data for this Ligand-Target Pair
Affinity DataEC50: 105nMAssay Description:Agonist activity for retinoic acid receptor RXR gamma in transcriptional activation assayMore data for this Ligand-Target Pair
Affinity DataEC50: 122nMAssay Description:Effective concentrations against Retinoic acid receptor RXR-gammaMore data for this Ligand-Target Pair
Affinity DataEC50: 124nMAssay Description:Transcriptional activity was evaluated in CV-1 cells transfected with expression vector for Retinoic acid receptor RXR-gammaMore data for this Ligand-Target Pair