Compile Data Set for Download or QSAR
maximum 50k data
Found 26 Enz. Inhib. hit(s) with all data for entry = 6088
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Shandong Institute of Pharmaceutical Industry

LigandPNGBDBM108055(4-((4-((2,3-dimethyl-2H-indazole-6-yl)(methyl) ami...)
Affinity DataIC50:  12nMT: 2°CAssay Description:To the assay kit, 2.5 µL of different concentrate of the test compounds, Pazopanib or water (control) were added and incubated for 1 h at room t...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Shandong Institute of Pharmaceutical Industry

LigandPNGBDBM108055(4-((4-((2,3-dimethyl-2H-indazole-6-yl)(methyl) ami...)
Affinity DataIC50:  22nMT: 2°CAssay Description:To the assay kit, 2.5 µL of different concentrate of the test compounds, Pazopanib or water (control) were added and incubated for 1 h at room t...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Shandong Institute of Pharmaceutical Industry

LigandPNGBDBM108053(4-((4-((2,3-dimethyl-2H-indazole-6-yl)(methyl) ami...)
Affinity DataIC50:  25nMT: 2°CAssay Description:To the assay kit, 2.5 µL of different concentrate of the test compounds, Pazopanib or water (control) were added and incubated for 1 h at room t...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Shandong Institute of Pharmaceutical Industry

LigandPNGBDBM108051(4-((4-((2,3-dimethyl-2H-indazole-6-yl)(methyl) ami...)
Affinity DataIC50:  29nMT: 2°CAssay Description:To the assay kit, 2.5 µL of different concentrate of the test compounds, Pazopanib or water (control) were added and incubated for 1 h at room t...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Shandong Institute of Pharmaceutical Industry

LigandPNGBDBM108050(4-((4-((2,3-dimethyl-2H-indazole-6-yl)amino) pyrim...)
Affinity DataIC50:  34nMT: 2°CAssay Description:To the assay kit, 2.5 µL of different concentrate of the test compounds, Pazopanib or water (control) were added and incubated for 1 h at room t...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Shandong Institute of Pharmaceutical Industry

LigandPNGBDBM26474(5-({4-[(2,3-dimethyl-2H-indazol-6-yl)(methyl)amino...)
Affinity DataIC50:  43nMT: 2°CAssay Description:To the assay kit, 2.5 µL of different concentrate of the test compounds, Pazopanib or water (control) were added and incubated for 1 h at room t...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Shandong Institute of Pharmaceutical Industry

LigandPNGBDBM108053(4-((4-((2,3-dimethyl-2H-indazole-6-yl)(methyl) ami...)
Affinity DataIC50:  62nMT: 2°CAssay Description:To the assay kit, 2.5 µL of different concentrate of the test compounds, Pazopanib or water (control) were added and incubated for 1 h at room t...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Shandong Institute of Pharmaceutical Industry

LigandPNGBDBM108054(4-((4-((2,3-dimethyl-2H-indazole-6-yl)amino) pyrim...)
Affinity DataIC50:  120nMT: 2°CAssay Description:To the assay kit, 2.5 µL of different concentrate of the test compounds, Pazopanib or water (control) were added and incubated for 1 h at room t...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Shandong Institute of Pharmaceutical Industry

LigandPNGBDBM108051(4-((4-((2,3-dimethyl-2H-indazole-6-yl)(methyl) ami...)
Affinity DataIC50:  120nMT: 2°CAssay Description:To the assay kit, 2.5 µL of different concentrate of the test compounds, Pazopanib or water (control) were added and incubated for 1 h at room t...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Shandong Institute of Pharmaceutical Industry

LigandPNGBDBM108052(4-((4-((2,3-dimethyl-2H-indazole-6-yl)amino) pyrim...)
Affinity DataIC50:  160nMT: 2°CAssay Description:To the assay kit, 2.5 µL of different concentrate of the test compounds, Pazopanib or water (control) were added and incubated for 1 h at room t...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Shandong Institute of Pharmaceutical Industry

LigandPNGBDBM108052(4-((4-((2,3-dimethyl-2H-indazole-6-yl)amino) pyrim...)
Affinity DataIC50:  280nMT: 2°CAssay Description:To the assay kit, 2.5 µL of different concentrate of the test compounds, Pazopanib or water (control) were added and incubated for 1 h at room t...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Shandong Institute of Pharmaceutical Industry

LigandPNGBDBM108057(4-((4-((2,3-dimethyl-2H-indazole-6-yl)(methyl) ami...)
Affinity DataIC50:  320nMT: 2°CAssay Description:To the assay kit, 2.5 µL of different concentrate of the test compounds, Pazopanib or water (control) were added and incubated for 1 h at room t...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Shandong Institute of Pharmaceutical Industry

LigandPNGBDBM108054(4-((4-((2,3-dimethyl-2H-indazole-6-yl)amino) pyrim...)
Affinity DataIC50:  360nMT: 2°CAssay Description:To the assay kit, 2.5 µL of different concentrate of the test compounds, Pazopanib or water (control) were added and incubated for 1 h at room t...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Shandong Institute of Pharmaceutical Industry

LigandPNGBDBM108059(N-carbamimidoyl-4-((4-((2,3-dimethyl-2H-indazole- ...)
Affinity DataIC50:  360nMT: 2°CAssay Description:To the assay kit, 2.5 µL of different concentrate of the test compounds, Pazopanib or water (control) were added and incubated for 1 h at room t...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Shandong Institute of Pharmaceutical Industry

LigandPNGBDBM108050(4-((4-((2,3-dimethyl-2H-indazole-6-yl)amino) pyrim...)
Affinity DataIC50:  460nMT: 2°CAssay Description:To the assay kit, 2.5 µL of different concentrate of the test compounds, Pazopanib or water (control) were added and incubated for 1 h at room t...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Shandong Institute of Pharmaceutical Industry

LigandPNGBDBM26474(5-({4-[(2,3-dimethyl-2H-indazol-6-yl)(methyl)amino...)
Affinity DataIC50:  620nMT: 2°CAssay Description:To the assay kit, 2.5 µL of different concentrate of the test compounds, Pazopanib or water (control) were added and incubated for 1 h at room t...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Shandong Institute of Pharmaceutical Industry

LigandPNGBDBM108057(4-((4-((2,3-dimethyl-2H-indazole-6-yl)(methyl) ami...)
Affinity DataIC50:  650nMT: 2°CAssay Description:To the assay kit, 2.5 µL of different concentrate of the test compounds, Pazopanib or water (control) were added and incubated for 1 h at room t...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Shandong Institute of Pharmaceutical Industry

LigandPNGBDBM108059(N-carbamimidoyl-4-((4-((2,3-dimethyl-2H-indazole- ...)
Affinity DataIC50:  720nMT: 2°CAssay Description:To the assay kit, 2.5 µL of different concentrate of the test compounds, Pazopanib or water (control) were added and incubated for 1 h at room t...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Shandong Institute of Pharmaceutical Industry

LigandPNGBDBM108049(4-((4-((2,3-dimethyl-2H-indazole-6-yl)(methyl) ami...)
Affinity DataIC50:  870nMT: 2°CAssay Description:To the assay kit, 2.5 µL of different concentrate of the test compounds, Pazopanib or water (control) were added and incubated for 1 h at room t...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Shandong Institute of Pharmaceutical Industry

LigandPNGBDBM108058(N-carbamimidoyl-4-((4-((2,3-dimethyl-2H-indazole- ...)
Affinity DataIC50:  930nMT: 2°CAssay Description:To the assay kit, 2.5 µL of different concentrate of the test compounds, Pazopanib or water (control) were added and incubated for 1 h at room t...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Shandong Institute of Pharmaceutical Industry

LigandPNGBDBM108058(N-carbamimidoyl-4-((4-((2,3-dimethyl-2H-indazole- ...)
Affinity DataIC50:  1.34E+3nMT: 2°CAssay Description:To the assay kit, 2.5 µL of different concentrate of the test compounds, Pazopanib or water (control) were added and incubated for 1 h at room t...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Shandong Institute of Pharmaceutical Industry

LigandPNGBDBM108049(4-((4-((2,3-dimethyl-2H-indazole-6-yl)(methyl) ami...)
Affinity DataIC50:  1.35E+3nMT: 2°CAssay Description:To the assay kit, 2.5 µL of different concentrate of the test compounds, Pazopanib or water (control) were added and incubated for 1 h at room t...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor protein-tyrosine kinase(Homo sapiens (Human))
Shandong Institute of Pharmaceutical Industry

LigandPNGBDBM108059(N-carbamimidoyl-4-((4-((2,3-dimethyl-2H-indazole- ...)
Affinity DataIC50:  1.37E+3nMT: 2°CAssay Description:To the assay kit, 2.5 µL of different concentrate of the test compounds, Pazopanib or water (control) were added and incubated for 1 h at room t...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Shandong Institute of Pharmaceutical Industry

LigandPNGBDBM108056(4-((4-((2,3-dimethyl-2H-indazole-6-yl)amino) pyrim...)
Affinity DataIC50:  1.63E+3nMT: 2°CAssay Description:To the assay kit, 2.5 µL of different concentrate of the test compounds, Pazopanib or water (control) were added and incubated for 1 h at room t...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Shandong Institute of Pharmaceutical Industry

LigandPNGBDBM108056(4-((4-((2,3-dimethyl-2H-indazole-6-yl)amino) pyrim...)
Affinity DataIC50:  2.18E+3nMT: 2°CAssay Description:To the assay kit, 2.5 µL of different concentrate of the test compounds, Pazopanib or water (control) were added and incubated for 1 h at room t...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor protein-tyrosine kinase(Homo sapiens (Human))
Shandong Institute of Pharmaceutical Industry

LigandPNGBDBM26474(5-({4-[(2,3-dimethyl-2H-indazol-6-yl)(methyl)amino...)
Affinity DataIC50:  5.95E+3nMT: 2°CAssay Description:To the assay kit, 2.5 µL of different concentrate of the test compounds, Pazopanib or water (control) were added and incubated for 1 h at room t...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed