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Found 13 Enz. Inhib. hit(s) with all data for entry = 7015
TargetDipeptidyl peptidase 4 [K6R,T557I](Homo sapiens (Human))
China Pharmaceutical University

LigandPNGBDBM50228403((R)-8-(3-aminopiperidin-1-yl)-7-(but-2-ynyl)-3-met...)
Affinity DataIC50:  1nMAssay Description:The DPP-4 Drug Discovery Kit (Enzo Life Sciences International, Inc.) was used for the assay of inhibition of DPP-4 activity. The assay is based on t...More data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4 [K6R,T557I](Homo sapiens (Human))
China Pharmaceutical University

LigandPNGBDBM16285(2-({6-[(3R)-3-aminopiperidin-1-yl]-3-methyl-2,4-di...)
Affinity DataIC50:  7nMAssay Description:The DPP-4 Drug Discovery Kit (Enzo Life Sciences International, Inc.) was used for the assay of inhibition of DPP-4 activity. The assay is based on t...More data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4 [K6R,T557I](Homo sapiens (Human))
China Pharmaceutical University

LigandPNGBDBM166622((2-(2,4-Dichlorophenyl)imidazo[1,2-a]pyridin-3-yl)...)
Affinity DataIC50:  130nMAssay Description:The DPP-4 Drug Discovery Kit (Enzo Life Sciences International, Inc.) was used for the assay of inhibition of DPP-4 activity. The assay is based on t...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4 [K6R,T557I](Homo sapiens (Human))
China Pharmaceutical University

LigandPNGBDBM166624((2-(o-Tolyl)imidazo[1,2-a]pyridin-3-yl)methanamine...)
Affinity DataIC50:  290nMAssay Description:The DPP-4 Drug Discovery Kit (Enzo Life Sciences International, Inc.) was used for the assay of inhibition of DPP-4 activity. The assay is based on t...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4 [K6R,T557I](Homo sapiens (Human))
China Pharmaceutical University

LigandPNGBDBM166623((2-(2,5-Dichlorophenyl)imidazo[1,2-a]pyridin-3-yl)...)
Affinity DataIC50:  650nMAssay Description:The DPP-4 Drug Discovery Kit (Enzo Life Sciences International, Inc.) was used for the assay of inhibition of DPP-4 activity. The assay is based on t...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4 [K6R,T557I](Homo sapiens (Human))
China Pharmaceutical University

LigandPNGBDBM166627((7-Methyl-2-(p-tolyl)imidazo[1,2-a]pyridin-3-yl)me...)
Affinity DataIC50:  840nMAssay Description:The DPP-4 Drug Discovery Kit (Enzo Life Sciences International, Inc.) was used for the assay of inhibition of DPP-4 activity. The assay is based on t...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4 [K6R,T557I](Homo sapiens (Human))
China Pharmaceutical University

LigandPNGBDBM166625((2-(4-Bromophenyl)imidazo[1,2-a]pyridin-3-yl)metha...)
Affinity DataIC50:  940nMAssay Description:The DPP-4 Drug Discovery Kit (Enzo Life Sciences International, Inc.) was used for the assay of inhibition of DPP-4 activity. The assay is based on t...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4 [K6R,T557I](Homo sapiens (Human))
China Pharmaceutical University

LigandPNGBDBM166621((2-(4-Chlorophenyl)imidazo[1,2-a]pyridin-3-yl)meth...)
Affinity DataIC50:  6.46E+3nMAssay Description:The DPP-4 Drug Discovery Kit (Enzo Life Sciences International, Inc.) was used for the assay of inhibition of DPP-4 activity. The assay is based on t...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4 [K6R,T557I](Homo sapiens (Human))
China Pharmaceutical University

LigandPNGBDBM166626((6-Methyl-2-(p-tolyl)imidazo[1,2-a]pyridin-3-yl)me...)
Affinity DataIC50:  7.46E+3nMAssay Description:The DPP-4 Drug Discovery Kit (Enzo Life Sciences International, Inc.) was used for the assay of inhibition of DPP-4 activity. The assay is based on t...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4 [K6R,T557I](Homo sapiens (Human))
China Pharmaceutical University

LigandPNGBDBM166619((2-Phenylimidazo[1,2-a]pyridin-3-yl)methanamine hy...)
Affinity DataIC50:  1.37E+4nMAssay Description:The DPP-4 Drug Discovery Kit (Enzo Life Sciences International, Inc.) was used for the assay of inhibition of DPP-4 activity. The assay is based on t...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4 [K6R,T557I](Homo sapiens (Human))
China Pharmaceutical University

LigandPNGBDBM166620((2-(3-Chlorophenyl)imidazo[1,2-a]pyridin-3-yl)meth...)
Affinity DataIC50: >5.00E+4nMAssay Description:The DPP-4 Drug Discovery Kit (Enzo Life Sciences International, Inc.) was used for the assay of inhibition of DPP-4 activity. The assay is based on t...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4 [K6R,T557I](Homo sapiens (Human))
China Pharmaceutical University

LigandPNGBDBM166628((8-Methyl-2-(p-tolyl)imidazo[1,2-a]pyridin-3-yl)me...)
Affinity DataIC50: >5.00E+4nMAssay Description:The DPP-4 Drug Discovery Kit (Enzo Life Sciences International, Inc.) was used for the assay of inhibition of DPP-4 activity. The assay is based on t...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4 [K6R,T557I](Homo sapiens (Human))
China Pharmaceutical University

LigandPNGBDBM166629(Methyl 3-(aminomethyl)-2-(p-tolyl)imidazo[1,2-a]py...)
Affinity DataIC50: >5.00E+4nMAssay Description:The DPP-4 Drug Discovery Kit (Enzo Life Sciences International, Inc.) was used for the assay of inhibition of DPP-4 activity. The assay is based on t...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed