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Found 40 Enz. Inhib. hit(s) with all data for entry = 7344
TargetPolyunsaturated fatty acid lipoxygenase ALOX15(Homo sapiens (Human))
Akaal Pharma

US Patent
LigandPNGBDBM60832(US9181182, 23)
Affinity DataEC50:  1.24E+3nMT: 2°CAssay Description:Selected Compounds of the Examples were evaluated at Millipore Corporation, USA, using S1P1 receptor; [35S]-GTPgamaS binding assay. A [35S]-GTPgamaS ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSphingosine 1-phosphate receptor 3(Homo sapiens (Human))
Akaal Pharma

US Patent
LigandPNGBDBM190520(US9181182, 47)
Affinity DataEC50:  96.5nMT: 2°CAssay Description:Selected Compounds of the Examples were evaluated at Millipore Corporation, USA, using S1P1 receptor; [35S]-GTPgamaS binding assay. A [35S]-GTPgamaS ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPolyunsaturated fatty acid lipoxygenase ALOX15(Homo sapiens (Human))
Akaal Pharma

US Patent
LigandPNGBDBM60834(US9181182, 30)
Affinity DataEC50: >5.54E+4nMT: 2°CAssay Description:Selected Compounds of the Examples were evaluated at Millipore Corporation, USA, using S1P1 receptor; [35S]-GTPgamaS binding assay. A [35S]-GTPgamaS ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPolyunsaturated fatty acid lipoxygenase ALOX15(Homo sapiens (Human))
Akaal Pharma

US Patent
LigandPNGBDBM60835(US9181182, 63)
Affinity DataEC50: >4.00E+4nMT: 2°CAssay Description:Selected Compounds of the Examples were evaluated at Millipore Corporation, USA, using S1P1 receptor; [35S]-GTPgamaS binding assay. A [35S]-GTPgamaS ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
Akaal Pharma

US Patent
LigandPNGBDBM190497(US9181182, 1)
Affinity DataEC50: >2.50E+4nMT: 2°CAssay Description:Selected Compounds of the Examples were evaluated at Millipore Corporation, USA, using S1P1 receptor; [35S]-GTPgamaS binding assay. A [35S]-GTPgamaS ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
Akaal Pharma

US Patent
LigandPNGBDBM190498(US9181182, 2)
Affinity DataEC50:  1.56E+3nMT: 2°CAssay Description:Selected Compounds of the Examples were evaluated at Millipore Corporation, USA, using S1P1 receptor; [35S]-GTPgamaS binding assay. A [35S]-GTPgamaS ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
Akaal Pharma

US Patent
LigandPNGBDBM190499(US9181182, 3)
Affinity DataEC50:  2.11E+3nMT: 2°CAssay Description:Selected Compounds of the Examples were evaluated at Millipore Corporation, USA, using S1P1 receptor; [35S]-GTPgamaS binding assay. A [35S]-GTPgamaS ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
Akaal Pharma

US Patent
LigandPNGBDBM190500(US9181182, 9)
Affinity DataEC50: >860nMT: 2°CAssay Description:Selected Compounds of the Examples were evaluated at Millipore Corporation, USA, using S1P1 receptor; [35S]-GTPgamaS binding assay. A [35S]-GTPgamaS ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
Akaal Pharma

US Patent
LigandPNGBDBM190501(US9181182, 8)
Affinity DataEC50:  131nMT: 2°CAssay Description:Selected Compounds of the Examples were evaluated at Millipore Corporation, USA, using S1P1 receptor; [35S]-GTPgamaS binding assay. A [35S]-GTPgamaS ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
Akaal Pharma

US Patent
LigandPNGBDBM190502(US9181182, 7)
Affinity DataEC50:  783nMT: 2°CAssay Description:Selected Compounds of the Examples were evaluated at Millipore Corporation, USA, using S1P1 receptor; [35S]-GTPgamaS binding assay. A [35S]-GTPgamaS ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
Akaal Pharma

US Patent
LigandPNGBDBM190503(US9181182, 34)
Affinity DataEC50:  6.80nMT: 2°CAssay Description:Selected Compounds of the Examples were evaluated at Millipore Corporation, USA, using S1P1 receptor; [35S]-GTPgamaS binding assay. A [35S]-GTPgamaS ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
Akaal Pharma

US Patent
LigandPNGBDBM190504(US9181182, 35)
Affinity DataEC50:  54nMT: 2°CAssay Description:Selected Compounds of the Examples were evaluated at Millipore Corporation, USA, using S1P1 receptor; [35S]-GTPgamaS binding assay. A [35S]-GTPgamaS ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
Akaal Pharma

US Patent
LigandPNGBDBM190505(US9181182, 36)
Affinity DataEC50:  501nMT: 2°CAssay Description:Selected Compounds of the Examples were evaluated at Millipore Corporation, USA, using S1P1 receptor; [35S]-GTPgamaS binding assay. A [35S]-GTPgamaS ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
Akaal Pharma

US Patent
LigandPNGBDBM190506(US9181182, 39)
Affinity DataEC50: >3.24E+3nMT: 2°CAssay Description:Selected Compounds of the Examples were evaluated at Millipore Corporation, USA, using S1P1 receptor; [35S]-GTPgamaS binding assay. A [35S]-GTPgamaS ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
Akaal Pharma

US Patent
LigandPNGBDBM190507(US9181182, 40)
Affinity DataEC50:  344nMT: 2°CAssay Description:Selected Compounds of the Examples were evaluated at Millipore Corporation, USA, using S1P1 receptor; [35S]-GTPgamaS binding assay. A [35S]-GTPgamaS ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
Akaal Pharma

US Patent
LigandPNGBDBM190508(US9181182, 41(a))
Affinity DataEC50: >1.36E+3nMT: 2°CAssay Description:Selected Compounds of the Examples were evaluated at Millipore Corporation, USA, using S1P1 receptor; [35S]-GTPgamaS binding assay. A [35S]-GTPgamaS ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
Akaal Pharma

US Patent
LigandPNGBDBM190509(US9181182, 41(b))
Affinity DataEC50: >2.90E+4nMT: 2°CAssay Description:Selected Compounds of the Examples were evaluated at Millipore Corporation, USA, using S1P1 receptor; [35S]-GTPgamaS binding assay. A [35S]-GTPgamaS ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
Akaal Pharma

US Patent
LigandPNGBDBM190510(US9181182, 42)
Affinity DataEC50:  1.42E+3nMT: 2°CAssay Description:Selected Compounds of the Examples were evaluated at Millipore Corporation, USA, using S1P1 receptor; [35S]-GTPgamaS binding assay. A [35S]-GTPgamaS ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
Akaal Pharma

US Patent
LigandPNGBDBM190511(US9181182, 12)
Affinity DataEC50:  1.82E+3nMT: 2°CAssay Description:Selected Compounds of the Examples were evaluated at Millipore Corporation, USA, using S1P1 receptor; [35S]-GTPgamaS binding assay. A [35S]-GTPgamaS ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
Akaal Pharma

US Patent
LigandPNGBDBM190512(US9181182, 10)
Affinity DataEC50: >510nMT: 2°CAssay Description:Selected Compounds of the Examples were evaluated at Millipore Corporation, USA, using S1P1 receptor; [35S]-GTPgamaS binding assay. A [35S]-GTPgamaS ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
Akaal Pharma

US Patent
LigandPNGBDBM190513(US9181182, 49)
Affinity DataEC50:  114nMT: 2°CAssay Description:Selected Compounds of the Examples were evaluated at Millipore Corporation, USA, using S1P1 receptor; [35S]-GTPgamaS binding assay. A [35S]-GTPgamaS ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
Akaal Pharma

US Patent
LigandPNGBDBM190514(US9181182, 50)
Affinity DataEC50:  17.9nMT: 2°CAssay Description:Selected Compounds of the Examples were evaluated at Millipore Corporation, USA, using S1P1 receptor; [35S]-GTPgamaS binding assay. A [35S]-GTPgamaS ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
Akaal Pharma

US Patent
LigandPNGBDBM190515(US9181182, 55)
Affinity DataEC50:  31.6nMT: 2°CAssay Description:Selected Compounds of the Examples were evaluated at Millipore Corporation, USA, using S1P1 receptor; [35S]-GTPgamaS binding assay. A [35S]-GTPgamaS ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
Akaal Pharma

US Patent
LigandPNGBDBM190516(US9181182, 58)
Affinity DataEC50: >2.06E+3nMT: 2°CAssay Description:Selected Compounds of the Examples were evaluated at Millipore Corporation, USA, using S1P1 receptor; [35S]-GTPgamaS binding assay. A [35S]-GTPgamaS ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
Akaal Pharma

US Patent
LigandPNGBDBM190517(US9181182, 59)
Affinity DataEC50: >2.13E+3nMT: 2°CAssay Description:Selected Compounds of the Examples were evaluated at Millipore Corporation, USA, using S1P1 receptor; [35S]-GTPgamaS binding assay. A [35S]-GTPgamaS ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
Akaal Pharma

US Patent
LigandPNGBDBM190518(US9181182, 65)
Affinity DataEC50:  7.40nMT: 2°CAssay Description:Selected Compounds of the Examples were evaluated at Millipore Corporation, USA, using S1P1 receptor; [35S]-GTPgamaS binding assay. A [35S]-GTPgamaS ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
Akaal Pharma

US Patent
LigandPNGBDBM190519(US9181182, 43)
Affinity DataEC50:  18nMT: 2°CAssay Description:Selected Compounds of the Examples were evaluated at Millipore Corporation, USA, using S1P1 receptor; [35S]-GTPgamaS binding assay. A [35S]-GTPgamaS ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
Akaal Pharma

US Patent
LigandPNGBDBM190520(US9181182, 47)
Affinity DataEC50:  2.40nMT: 2°CAssay Description:Selected Compounds of the Examples were evaluated at Millipore Corporation, USA, using S1P1 receptor; [35S]-GTPgamaS binding assay. A [35S]-GTPgamaS ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
Akaal Pharma

US Patent
LigandPNGBDBM190521(US9181182, 46)
Affinity DataEC50:  88nMT: 2°CAssay Description:Selected Compounds of the Examples were evaluated at Millipore Corporation, USA, using S1P1 receptor; [35S]-GTPgamaS binding assay. A [35S]-GTPgamaS ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
Akaal Pharma

US Patent
LigandPNGBDBM190522(US9181182, 44)
Affinity DataEC50:  48.1nMT: 2°CAssay Description:Selected Compounds of the Examples were evaluated at Millipore Corporation, USA, using S1P1 receptor; [35S]-GTPgamaS binding assay. A [35S]-GTPgamaS ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
Akaal Pharma

US Patent
LigandPNGBDBM190523(US9181182, 48)
Affinity DataEC50:  6.70nMT: 2°CAssay Description:Selected Compounds of the Examples were evaluated at Millipore Corporation, USA, using S1P1 receptor; [35S]-GTPgamaS binding assay. A [35S]-GTPgamaS ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
Akaal Pharma

US Patent
LigandPNGBDBM190524(US9181182, 52)
Affinity DataEC50:  34.5nMT: 2°CAssay Description:Selected Compounds of the Examples were evaluated at Millipore Corporation, USA, using S1P1 receptor; [35S]-GTPgamaS binding assay. A [35S]-GTPgamaS ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
Akaal Pharma

US Patent
LigandPNGBDBM190525(US9181182, 54)
Affinity DataEC50:  43.8nMT: 2°CAssay Description:Selected Compounds of the Examples were evaluated at Millipore Corporation, USA, using S1P1 receptor; [35S]-GTPgamaS binding assay. A [35S]-GTPgamaS ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
Akaal Pharma

US Patent
LigandPNGBDBM190526(US9181182, 56)
Affinity DataEC50:  2.90nMT: 2°CAssay Description:Selected Compounds of the Examples were evaluated at Millipore Corporation, USA, using S1P1 receptor; [35S]-GTPgamaS binding assay. A [35S]-GTPgamaS ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
Akaal Pharma

US Patent
LigandPNGBDBM190527(US9181182, 51)
Affinity DataEC50:  3.5nMT: 2°CAssay Description:Selected Compounds of the Examples were evaluated at Millipore Corporation, USA, using S1P1 receptor; [35S]-GTPgamaS binding assay. A [35S]-GTPgamaS ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSphingosine 1-phosphate receptor 3(Homo sapiens (Human))
Akaal Pharma

US Patent
LigandPNGBDBM190503(US9181182, 34)
Affinity DataEC50:  129nMT: 2°CAssay Description:Selected Compounds of the Examples were evaluated at Millipore Corporation, USA, using S1P1 receptor; [35S]-GTPgamaS binding assay. A [35S]-GTPgamaS ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSphingosine 1-phosphate receptor 3(Homo sapiens (Human))
Akaal Pharma

US Patent
LigandPNGBDBM190507(US9181182, 40)
Affinity DataEC50: >1.56E+3nMT: 2°CAssay Description:Selected Compounds of the Examples were evaluated at Millipore Corporation, USA, using S1P1 receptor; [35S]-GTPgamaS binding assay. A [35S]-GTPgamaS ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSphingosine 1-phosphate receptor 3(Homo sapiens (Human))
Akaal Pharma

US Patent
LigandPNGBDBM190518(US9181182, 65)
Affinity DataEC50:  39nMT: 2°CAssay Description:Selected Compounds of the Examples were evaluated at Millipore Corporation, USA, using S1P1 receptor; [35S]-GTPgamaS binding assay. A [35S]-GTPgamaS ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSphingosine 1-phosphate receptor 3(Homo sapiens (Human))
Akaal Pharma

US Patent
LigandPNGBDBM190519(US9181182, 43)
Affinity DataEC50:  310nMT: 2°CAssay Description:Selected Compounds of the Examples were evaluated at Millipore Corporation, USA, using S1P1 receptor; [35S]-GTPgamaS binding assay. A [35S]-GTPgamaS ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPolyunsaturated fatty acid lipoxygenase ALOX15(Homo sapiens (Human))
Akaal Pharma

US Patent
LigandPNGBDBM60833(US9181182, 33)
Affinity DataEC50: >2.40E+4nMT: 2°CAssay Description:Selected Compounds of the Examples were evaluated at Millipore Corporation, USA, using S1P1 receptor; [35S]-GTPgamaS binding assay. A [35S]-GTPgamaS ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent