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Found 39 Enz. Inhib. hit(s) with all data for entry = 8429
TargetHistamine receptor H3(Macaca mulatta (Rhesus macaque))
Sanofi

US Patent
LigandPNGBDBM247467(US9453023, 26)
Affinity DataKi:  6.01nMAssay Description:Rhesus H3 radioligand binding assay was performed using rhesus H3 receptor membranes (prepared as described above), [3H]-Methylhistamine (Perkin Elme...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetHistamine receptor H3(Macaca mulatta (Rhesus macaque))
Sanofi

US Patent
LigandPNGBDBM247449(US9453023, 8)
Affinity DataKi:  6.07nMAssay Description:Rhesus H3 radioligand binding assay was performed using rhesus H3 receptor membranes (prepared as described above), [3H]-Methylhistamine (Perkin Elme...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetHistamine receptor H3(Macaca mulatta (Rhesus macaque))
Sanofi

US Patent
LigandPNGBDBM247453(US9453023, 12)
Affinity DataKi:  6.10nMAssay Description:Rhesus H3 radioligand binding assay was performed using rhesus H3 receptor membranes (prepared as described above), [3H]-Methylhistamine (Perkin Elme...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetHistamine receptor H3(Macaca mulatta (Rhesus macaque))
Sanofi

US Patent
LigandPNGBDBM247455(US9453023, 14)
Affinity DataKi:  6.61nMAssay Description:Rhesus H3 radioligand binding assay was performed using rhesus H3 receptor membranes (prepared as described above), [3H]-Methylhistamine (Perkin Elme...More data for this Ligand-Target Pair
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TargetHistamine receptor H3(Macaca mulatta (Rhesus macaque))
Sanofi

US Patent
LigandPNGBDBM247462(US9453023, 21)
Affinity DataKi:  6.88nMAssay Description:Rhesus H3 radioligand binding assay was performed using rhesus H3 receptor membranes (prepared as described above), [3H]-Methylhistamine (Perkin Elme...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetHistamine receptor H3(Macaca mulatta (Rhesus macaque))
Sanofi

US Patent
LigandPNGBDBM247459(US9453023, 18)
Affinity DataKi:  11.3nMAssay Description:Rhesus H3 radioligand binding assay was performed using rhesus H3 receptor membranes (prepared as described above), [3H]-Methylhistamine (Perkin Elme...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetHistamine receptor H3(Macaca mulatta (Rhesus macaque))
Sanofi

US Patent
LigandPNGBDBM247442(US9453023, 1)
Affinity DataKi:  11.9nMAssay Description:Rhesus H3 radioligand binding assay was performed using rhesus H3 receptor membranes (prepared as described above), [3H]-Methylhistamine (Perkin Elme...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetHistamine receptor H3(Macaca mulatta (Rhesus macaque))
Sanofi

US Patent
LigandPNGBDBM247465(US9453023, 24)
Affinity DataKi:  12.4nMAssay Description:Rhesus H3 radioligand binding assay was performed using rhesus H3 receptor membranes (prepared as described above), [3H]-Methylhistamine (Perkin Elme...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetHistamine receptor H3(Macaca mulatta (Rhesus macaque))
Sanofi

US Patent
LigandPNGBDBM247443(US9453023, 2)
Affinity DataKi:  12.8nMAssay Description:Rhesus H3 radioligand binding assay was performed using rhesus H3 receptor membranes (prepared as described above), [3H]-Methylhistamine (Perkin Elme...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetHistamine receptor H3(Macaca mulatta (Rhesus macaque))
Sanofi

US Patent
LigandPNGBDBM247444(US9453023, 3)
Affinity DataKi:  17.9nMAssay Description:Rhesus H3 radioligand binding assay was performed using rhesus H3 receptor membranes (prepared as described above), [3H]-Methylhistamine (Perkin Elme...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetHistamine receptor H3(Macaca mulatta (Rhesus macaque))
Sanofi

US Patent
LigandPNGBDBM247447(US9453023, 6)
Affinity DataKi:  26.8nMAssay Description:Rhesus H3 radioligand binding assay was performed using rhesus H3 receptor membranes (prepared as described above), [3H]-Methylhistamine (Perkin Elme...More data for this Ligand-Target Pair
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TargetHistamine receptor H3(Macaca mulatta (Rhesus macaque))
Sanofi

US Patent
LigandPNGBDBM247471(US9453023, 30)
Affinity DataKi:  27.4nMAssay Description:Rhesus H3 radioligand binding assay was performed using rhesus H3 receptor membranes (prepared as described above), [3H]-Methylhistamine (Perkin Elme...More data for this Ligand-Target Pair
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TargetHistamine receptor H3(Macaca mulatta (Rhesus macaque))
Sanofi

US Patent
LigandPNGBDBM247448(US9453023, 7)
Affinity DataKi:  27.5nMAssay Description:Rhesus H3 radioligand binding assay was performed using rhesus H3 receptor membranes (prepared as described above), [3H]-Methylhistamine (Perkin Elme...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHistamine receptor H3(Macaca mulatta (Rhesus macaque))
Sanofi

US Patent
LigandPNGBDBM247474(US9453023, 33)
Affinity DataKi:  32.6nMAssay Description:Rhesus H3 radioligand binding assay was performed using rhesus H3 receptor membranes (prepared as described above), [3H]-Methylhistamine (Perkin Elme...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHistamine receptor H3(Macaca mulatta (Rhesus macaque))
Sanofi

US Patent
LigandPNGBDBM247469(US9453023, 28)
Affinity DataKi:  33.7nMAssay Description:Rhesus H3 radioligand binding assay was performed using rhesus H3 receptor membranes (prepared as described above), [3H]-Methylhistamine (Perkin Elme...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHistamine receptor H3(Macaca mulatta (Rhesus macaque))
Sanofi

US Patent
LigandPNGBDBM247468(US9453023, 27)
Affinity DataKi:  34nMAssay Description:Rhesus H3 radioligand binding assay was performed using rhesus H3 receptor membranes (prepared as described above), [3H]-Methylhistamine (Perkin Elme...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHistamine receptor H3(Macaca mulatta (Rhesus macaque))
Sanofi

US Patent
LigandPNGBDBM247472(US9453023, 31)
Affinity DataKi:  34.9nMAssay Description:Rhesus H3 radioligand binding assay was performed using rhesus H3 receptor membranes (prepared as described above), [3H]-Methylhistamine (Perkin Elme...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHistamine receptor H3(Macaca mulatta (Rhesus macaque))
Sanofi

US Patent
LigandPNGBDBM247451(US9453023, 10)
Affinity DataKi:  35.3nMAssay Description:Rhesus H3 radioligand binding assay was performed using rhesus H3 receptor membranes (prepared as described above), [3H]-Methylhistamine (Perkin Elme...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHistamine receptor H3(Macaca mulatta (Rhesus macaque))
Sanofi

US Patent
LigandPNGBDBM247441(US9453023, Intermediate (13))
Affinity DataKi:  37.4nMAssay Description:Rhesus H3 radioligand binding assay was performed using rhesus H3 receptor membranes (prepared as described above), [3H]-Methylhistamine (Perkin Elme...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHistamine receptor H3(Macaca mulatta (Rhesus macaque))
Sanofi

US Patent
LigandPNGBDBM247452(US9453023, 11)
Affinity DataKi:  39.4nMAssay Description:Rhesus H3 radioligand binding assay was performed using rhesus H3 receptor membranes (prepared as described above), [3H]-Methylhistamine (Perkin Elme...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHistamine receptor H3(Macaca mulatta (Rhesus macaque))
Sanofi

US Patent
LigandPNGBDBM247446(US9453023, 5)
Affinity DataKi:  44.1nMAssay Description:Rhesus H3 radioligand binding assay was performed using rhesus H3 receptor membranes (prepared as described above), [3H]-Methylhistamine (Perkin Elme...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHistamine receptor H3(Macaca mulatta (Rhesus macaque))
Sanofi

US Patent
LigandPNGBDBM247457(US9453023, 16)
Affinity DataKi:  44.2nMAssay Description:Rhesus H3 radioligand binding assay was performed using rhesus H3 receptor membranes (prepared as described above), [3H]-Methylhistamine (Perkin Elme...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHistamine receptor H3(Macaca mulatta (Rhesus macaque))
Sanofi

US Patent
LigandPNGBDBM247466(US9453023, 25)
Affinity DataKi:  45.7nMAssay Description:Rhesus H3 radioligand binding assay was performed using rhesus H3 receptor membranes (prepared as described above), [3H]-Methylhistamine (Perkin Elme...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHistamine receptor H3(Macaca mulatta (Rhesus macaque))
Sanofi

US Patent
LigandPNGBDBM247464(US9453023, 23)
Affinity DataKi:  46.5nMAssay Description:Rhesus H3 radioligand binding assay was performed using rhesus H3 receptor membranes (prepared as described above), [3H]-Methylhistamine (Perkin Elme...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHistamine receptor H3(Macaca mulatta (Rhesus macaque))
Sanofi

US Patent
LigandPNGBDBM247477(US9453023, 36)
Affinity DataKi:  48.5nMAssay Description:Rhesus H3 radioligand binding assay was performed using rhesus H3 receptor membranes (prepared as described above), [3H]-Methylhistamine (Perkin Elme...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHistamine receptor H3(Macaca mulatta (Rhesus macaque))
Sanofi

US Patent
LigandPNGBDBM247440(US9453023, Intermediate (10))
Affinity DataKi:  65.4nMAssay Description:Rhesus H3 radioligand binding assay was performed using rhesus H3 receptor membranes (prepared as described above), [3H]-Methylhistamine (Perkin Elme...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHistamine receptor H3(Macaca mulatta (Rhesus macaque))
Sanofi

US Patent
LigandPNGBDBM247473(US9453023, 32)
Affinity DataKi:  65.5nMAssay Description:Rhesus H3 radioligand binding assay was performed using rhesus H3 receptor membranes (prepared as described above), [3H]-Methylhistamine (Perkin Elme...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHistamine receptor H3(Macaca mulatta (Rhesus macaque))
Sanofi

US Patent
LigandPNGBDBM247478(US9453023, 37)
Affinity DataKi:  71.4nMAssay Description:Rhesus H3 radioligand binding assay was performed using rhesus H3 receptor membranes (prepared as described above), [3H]-Methylhistamine (Perkin Elme...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHistamine receptor H3(Macaca mulatta (Rhesus macaque))
Sanofi

US Patent
LigandPNGBDBM247445(US9453023, 4)
Affinity DataKi:  75.2nMAssay Description:Rhesus H3 radioligand binding assay was performed using rhesus H3 receptor membranes (prepared as described above), [3H]-Methylhistamine (Perkin Elme...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHistamine receptor H3(Macaca mulatta (Rhesus macaque))
Sanofi

US Patent
LigandPNGBDBM247470(US9453023, 29)
Affinity DataKi:  75.3nMAssay Description:Rhesus H3 radioligand binding assay was performed using rhesus H3 receptor membranes (prepared as described above), [3H]-Methylhistamine (Perkin Elme...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHistamine receptor H3(Macaca mulatta (Rhesus macaque))
Sanofi

US Patent
LigandPNGBDBM247460(US9453023, 19)
Affinity DataKi:  82.2nMAssay Description:Rhesus H3 radioligand binding assay was performed using rhesus H3 receptor membranes (prepared as described above), [3H]-Methylhistamine (Perkin Elme...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHistamine receptor H3(Macaca mulatta (Rhesus macaque))
Sanofi

US Patent
LigandPNGBDBM247458(US9453023, 17)
Affinity DataKi:  84.3nMAssay Description:Rhesus H3 radioligand binding assay was performed using rhesus H3 receptor membranes (prepared as described above), [3H]-Methylhistamine (Perkin Elme...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHistamine receptor H3(Macaca mulatta (Rhesus macaque))
Sanofi

US Patent
LigandPNGBDBM247475(US9453023, 34)
Affinity DataKi:  98.7nMAssay Description:Rhesus H3 radioligand binding assay was performed using rhesus H3 receptor membranes (prepared as described above), [3H]-Methylhistamine (Perkin Elme...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHistamine receptor H3(Macaca mulatta (Rhesus macaque))
Sanofi

US Patent
LigandPNGBDBM247450(US9453023, 9)
Affinity DataKi:  112nMAssay Description:Rhesus H3 radioligand binding assay was performed using rhesus H3 receptor membranes (prepared as described above), [3H]-Methylhistamine (Perkin Elme...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHistamine receptor H3(Macaca mulatta (Rhesus macaque))
Sanofi

US Patent
LigandPNGBDBM247463(US9453023, 22)
Affinity DataKi:  118nMAssay Description:Rhesus H3 radioligand binding assay was performed using rhesus H3 receptor membranes (prepared as described above), [3H]-Methylhistamine (Perkin Elme...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHistamine receptor H3(Macaca mulatta (Rhesus macaque))
Sanofi

US Patent
LigandPNGBDBM247476(US9453023, 35)
Affinity DataKi:  136nMAssay Description:Rhesus H3 radioligand binding assay was performed using rhesus H3 receptor membranes (prepared as described above), [3H]-Methylhistamine (Perkin Elme...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHistamine receptor H3(Macaca mulatta (Rhesus macaque))
Sanofi

US Patent
LigandPNGBDBM247461(US9453023, 20)
Affinity DataKi:  137nMAssay Description:Rhesus H3 radioligand binding assay was performed using rhesus H3 receptor membranes (prepared as described above), [3H]-Methylhistamine (Perkin Elme...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHistamine receptor H3(Macaca mulatta (Rhesus macaque))
Sanofi

US Patent
LigandPNGBDBM247456(US9453023, 15)
Affinity DataKi:  220nMAssay Description:Rhesus H3 radioligand binding assay was performed using rhesus H3 receptor membranes (prepared as described above), [3H]-Methylhistamine (Perkin Elme...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHistamine receptor H3(Macaca mulatta (Rhesus macaque))
Sanofi

US Patent
LigandPNGBDBM247454(US9453023, 13)
Affinity DataKi:  379nMAssay Description:Rhesus H3 radioligand binding assay was performed using rhesus H3 receptor membranes (prepared as described above), [3H]-Methylhistamine (Perkin Elme...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent