Compile Data Set for Download or QSAR
maximum 50k data
Found 28 Enz. Inhib. hit(s) with all data for entry = 2993
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Abbott Laboratories

LigandPNGBDBM26732(Benzothiazole-based analogue, 1 | N-[4-(4-methoxy-...)
Affinity DataIC50:  1.70nMpH: 8.0 T: 2°CAssay Description:[3H]anandamide was incubated with membranes to produce radiolabeled ethanolamine and unlabeled arachidonic acid. Charcoal selectively binds anandamid...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Abbott Laboratories

LigandPNGBDBM26712(1-(benzenesulfonyl)-N-[4-(6-methyl-1,3-benzothiazo...)
Affinity DataIC50:  13nMpH: 8.0 T: 2°CAssay Description:[3H]anandamide was incubated with membranes to produce radiolabeled ethanolamine and unlabeled arachidonic acid. Charcoal selectively binds anandamid...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Abbott Laboratories

LigandPNGBDBM26729(N-[4-(6-chloro-1,3-benzothiazol-2-yl)phenyl]-1-(th...)
Affinity DataIC50:  14nMpH: 8.0 T: 2°CAssay Description:[3H]anandamide was incubated with membranes to produce radiolabeled ethanolamine and unlabeled arachidonic acid. Charcoal selectively binds anandamid...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Abbott Laboratories

LigandPNGBDBM26731(N-[4-(4-methyl-1,3-benzothiazol-2-yl)phenyl]-1-(th...)
Affinity DataIC50:  14nMpH: 8.0 T: 2°CAssay Description:[3H]anandamide was incubated with membranes to produce radiolabeled ethanolamine and unlabeled arachidonic acid. Charcoal selectively binds anandamid...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Abbott Laboratories

LigandPNGBDBM26728(N-[4-(1,3-benzothiazol-2-yl)phenyl]-1-(thiophene-2...)
Affinity DataIC50:  15nMpH: 8.0 T: 2°CAssay Description:[3H]anandamide was incubated with membranes to produce radiolabeled ethanolamine and unlabeled arachidonic acid. Charcoal selectively binds anandamid...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Abbott Laboratories

LigandPNGBDBM26722(4-(6-methyl-1,3-benzothiazol-2-yl)-N-{[1-(thiophen...)
Affinity DataIC50:  16nMpH: 8.0 T: 2°CAssay Description:[3H]anandamide was incubated with membranes to produce radiolabeled ethanolamine and unlabeled arachidonic acid. Charcoal selectively binds anandamid...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Abbott Laboratories

LigandPNGBDBM26708(N-[4-(6-methyl-1,3-benzothiazol-2-yl)phenyl]-1-(th...)
Affinity DataIC50:  18nMpH: 8.0 T: 2°CAssay Description:[3H]anandamide was incubated with membranes to produce radiolabeled ethanolamine and unlabeled arachidonic acid. Charcoal selectively binds anandamid...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Abbott Laboratories

LigandPNGBDBM26733(N-{4-[4-(3-methoxyphenyl)-1,3-thiazol-2-yl]phenyl}...)
Affinity DataIC50:  19nMpH: 8.0 T: 2°CAssay Description:[3H]anandamide was incubated with membranes to produce radiolabeled ethanolamine and unlabeled arachidonic acid. Charcoal selectively binds anandamid...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Abbott Laboratories

LigandPNGBDBM26724(N-[4-(quinolin-2-yl)phenyl]-1-(thiophene-2-sulfony...)
Affinity DataIC50:  21nMpH: 8.0 T: 2°CAssay Description:[3H]anandamide was incubated with membranes to produce radiolabeled ethanolamine and unlabeled arachidonic acid. Charcoal selectively binds anandamid...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Abbott Laboratories

LigandPNGBDBM26734(N-{4-[4-(4-methoxyphenyl)-1,3-thiazol-2-yl]phenyl}...)
Affinity DataIC50:  25nMpH: 8.0 T: 2°CAssay Description:[3H]anandamide was incubated with membranes to produce radiolabeled ethanolamine and unlabeled arachidonic acid. Charcoal selectively binds anandamid...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Abbott Laboratories

LigandPNGBDBM26713(1-[(2-fluorobenzene)sulfonyl]-N-[4-(6-methyl-1,3-b...)
Affinity DataIC50:  29nMpH: 8.0 T: 2°CAssay Description:[3H]anandamide was incubated with membranes to produce radiolabeled ethanolamine and unlabeled arachidonic acid. Charcoal selectively binds anandamid...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Abbott Laboratories

LigandPNGBDBM26735(N-{4-[4-(4-chlorophenyl)-1,3-thiazol-2-yl]phenyl}-...)
Affinity DataIC50:  44nMpH: 8.0 T: 2°CAssay Description:[3H]anandamide was incubated with membranes to produce radiolabeled ethanolamine and unlabeled arachidonic acid. Charcoal selectively binds anandamid...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Abbott Laboratories

LigandPNGBDBM26711(1-(dimethylsulfamoyl)-N-[4-(6-methyl-1,3-benzothia...)
Affinity DataIC50:  48nMpH: 8.0 T: 2°CAssay Description:[3H]anandamide was incubated with membranes to produce radiolabeled ethanolamine and unlabeled arachidonic acid. Charcoal selectively binds anandamid...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Abbott Laboratories

LigandPNGBDBM26710(N-[4-(6-methyl-1,3-benzothiazol-2-yl)phenyl]-1-(pr...)
Affinity DataIC50:  63nMpH: 8.0 T: 2°CAssay Description:[3H]anandamide was incubated with membranes to produce radiolabeled ethanolamine and unlabeled arachidonic acid. Charcoal selectively binds anandamid...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Abbott Laboratories

LigandPNGBDBM26720(N-[4-(6-methyl-1,3-benzothiazol-2-yl)phenyl]-1-(th...)
Affinity DataIC50:  65nMpH: 8.0 T: 2°CAssay Description:[3H]anandamide was incubated with membranes to produce radiolabeled ethanolamine and unlabeled arachidonic acid. Charcoal selectively binds anandamid...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Abbott Laboratories

LigandPNGBDBM26730(N-[4-(6-methoxy-1,3-benzothiazol-2-yl)phenyl]-1-(t...)
Affinity DataIC50:  71nMpH: 8.0 T: 2°CAssay Description:[3H]anandamide was incubated with membranes to produce radiolabeled ethanolamine and unlabeled arachidonic acid. Charcoal selectively binds anandamid...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Abbott Laboratories

LigandPNGBDBM26725(N-[4-(quinoxalin-2-yl)phenyl]-1-(thiophene-2-sulfo...)
Affinity DataIC50:  91nMpH: 8.0 T: 2°CAssay Description:[3H]anandamide was incubated with membranes to produce radiolabeled ethanolamine and unlabeled arachidonic acid. Charcoal selectively binds anandamid...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Abbott Laboratories

LigandPNGBDBM26709(1-(ethanesulfonyl)-N-[4-(6-methyl-1,3-benzothiazol...)
Affinity DataIC50:  109nMpH: 8.0 T: 2°CAssay Description:[3H]anandamide was incubated with membranes to produce radiolabeled ethanolamine and unlabeled arachidonic acid. Charcoal selectively binds anandamid...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Abbott Laboratories

LigandPNGBDBM26719(N-[4-(6-methyl-1,3-benzothiazol-2-yl)phenyl]-1-(th...)
Affinity DataIC50:  201nMpH: 8.0 T: 2°CAssay Description:[3H]anandamide was incubated with membranes to produce radiolabeled ethanolamine and unlabeled arachidonic acid. Charcoal selectively binds anandamid...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Abbott Laboratories

LigandPNGBDBM26726(N-[4-(6-methyl-1,3-benzoxazol-2-yl)phenyl]-1-(thio...)
Affinity DataIC50:  235nMpH: 8.0 T: 2°CAssay Description:[3H]anandamide was incubated with membranes to produce radiolabeled ethanolamine and unlabeled arachidonic acid. Charcoal selectively binds anandamid...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Abbott Laboratories

LigandPNGBDBM26714(1-[(2-chlorobenzene)sulfonyl]-N-[4-(6-methyl-1,3-b...)
Affinity DataIC50:  263nMpH: 8.0 T: 2°CAssay Description:[3H]anandamide was incubated with membranes to produce radiolabeled ethanolamine and unlabeled arachidonic acid. Charcoal selectively binds anandamid...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Abbott Laboratories

LigandPNGBDBM26723(N-[4-(1,3-thiazol-2-yl)phenyl]-1-(thiophene-2-sulf...)
Affinity DataIC50:  270nMpH: 8.0 T: 2°CAssay Description:[3H]anandamide was incubated with membranes to produce radiolabeled ethanolamine and unlabeled arachidonic acid. Charcoal selectively binds anandamid...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Abbott Laboratories

LigandPNGBDBM26715(1-[(3-chlorobenzene)sulfonyl]-N-[4-(6-methyl-1,3-b...)
Affinity DataIC50:  1.78E+3nMpH: 8.0 T: 2°CAssay Description:[3H]anandamide was incubated with membranes to produce radiolabeled ethanolamine and unlabeled arachidonic acid. Charcoal selectively binds anandamid...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Abbott Laboratories

LigandPNGBDBM26717(N-[4-(6-methyl-1,3-benzothiazol-2-yl)phenyl]-1-(th...)
Affinity DataIC50:  2.37E+3nMpH: 8.0 T: 2°CAssay Description:[3H]anandamide was incubated with membranes to produce radiolabeled ethanolamine and unlabeled arachidonic acid. Charcoal selectively binds anandamid...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Abbott Laboratories

LigandPNGBDBM26727(N-[4-(6-methyl-1H-1,3-benzodiazol-2-yl)phenyl]-1-(...)
Affinity DataIC50: >1.00E+4nMpH: 8.0 T: 2°CAssay Description:[3H]anandamide was incubated with membranes to produce radiolabeled ethanolamine and unlabeled arachidonic acid. Charcoal selectively binds anandamid...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Abbott Laboratories

LigandPNGBDBM26718(N-[4-(6-methyl-1,3-benzothiazol-2-yl)phenyl]-1-(th...)
Affinity DataIC50: >1.00E+4nMpH: 8.0 T: 2°CAssay Description:[3H]anandamide was incubated with membranes to produce radiolabeled ethanolamine and unlabeled arachidonic acid. Charcoal selectively binds anandamid...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Abbott Laboratories

LigandPNGBDBM26721(N-[4-(6-methyl-1,3-benzothiazol-2-yl)phenyl]-2-[1-...)
Affinity DataIC50: >1.00E+4nMpH: 8.0 T: 2°CAssay Description:[3H]anandamide was incubated with membranes to produce radiolabeled ethanolamine and unlabeled arachidonic acid. Charcoal selectively binds anandamid...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Abbott Laboratories

LigandPNGBDBM26716(1-[(4-chlorobenzene)sulfonyl]-N-[4-(6-methyl-1,3-b...)
Affinity DataIC50: >1.00E+4nMpH: 8.0 T: 2°CAssay Description:[3H]anandamide was incubated with membranes to produce radiolabeled ethanolamine and unlabeled arachidonic acid. Charcoal selectively binds anandamid...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed