Compile Data Set for Download or QSAR
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Found 63 Enz. Inhib. hit(s) with all data for entry = 50044403
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
Critical Therapeutics

Curated by ChEMBL
LigandPNGBDBM50049750((S)-3-(azetidin-2-ylmethoxy)pyridine | 3-((S)-1-Az...)
Affinity DataKi:  0.0520nMAssay Description:Agonist activity at alpha4beta2 nAChR (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Homo sapiens (Human))
Critical Therapeutics

Curated by ChEMBL
LigandPNGBDBM50049750((S)-3-(azetidin-2-ylmethoxy)pyridine | 3-((S)-1-Az...)
Affinity DataKi:  148nMAssay Description:Agonist activity at alpha7 nAChR (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Critical Therapeutics

Curated by ChEMBL
LigandPNGBDBM50016200(CHEMBL3262146)
Affinity DataIC50:  4nMAssay Description:Inhibition of biotinylated alpha-bungarotoxin binding to alpha7 nAChR in rat PC12 cells by FACS analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Critical Therapeutics

Curated by ChEMBL
LigandPNGBDBM50016184(CHEMBL3262131)
Affinity DataIC50:  4nMAssay Description:Inhibition of biotinylated alpha-bungarotoxin binding to alpha7 nAChR in rat PC12 cells by FACS analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Critical Therapeutics

Curated by ChEMBL
LigandPNGBDBM50016185(CHEMBL3262132)
Affinity DataIC50:  5.5nMAssay Description:Inhibition of biotinylated alpha-bungarotoxin binding to alpha7 nAChR in rat PC12 cells by FACS analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Critical Therapeutics

Curated by ChEMBL
LigandPNGBDBM50016209(CHEMBL3262155)
Affinity DataIC50:  9.5nMAssay Description:Inhibition of biotinylated alpha-bungarotoxin binding to alpha7 nAChR in rat PC12 cells by FACS analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Critical Therapeutics

Curated by ChEMBL
LigandPNGBDBM50016210(CHEMBL3262156)
Affinity DataIC50:  11nMAssay Description:Inhibition of biotinylated alpha-bungarotoxin binding to alpha7 nAChR in rat PC12 cells by FACS analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Critical Therapeutics

Curated by ChEMBL
LigandPNGBDBM50016227(CHEMBL3262173)
Affinity DataIC50:  13nMAssay Description:Inhibition of biotinylated alpha-bungarotoxin binding to alpha7 nAChR in rat PC12 cells by FACS analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Critical Therapeutics

Curated by ChEMBL
LigandPNGBDBM50016225(CHEMBL3262171)
Affinity DataIC50:  14nMAssay Description:Inhibition of biotinylated alpha-bungarotoxin binding to alpha7 nAChR in rat PC12 cells by FACS analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Critical Therapeutics

Curated by ChEMBL
LigandPNGBDBM50016197(CHEMBL3262143)
Affinity DataIC50:  17nMAssay Description:Inhibition of biotinylated alpha-bungarotoxin binding to alpha7 nAChR in rat PC12 cells by FACS analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Critical Therapeutics

Curated by ChEMBL
LigandPNGBDBM50016217(CHEMBL3262163)
Affinity DataIC50:  19nMAssay Description:Inhibition of biotinylated alpha-bungarotoxin binding to alpha7 nAChR in rat PC12 cells by FACS analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Critical Therapeutics

Curated by ChEMBL
LigandPNGBDBM50016198(CHEMBL3262144)
Affinity DataIC50:  19nMAssay Description:Inhibition of biotinylated alpha-bungarotoxin binding to alpha7 nAChR in rat PC12 cells by FACS analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Critical Therapeutics

Curated by ChEMBL
LigandPNGBDBM50016179(CHEMBL3262126)
Affinity DataIC50:  22nMAssay Description:Inhibition of biotinylated alpha-bungarotoxin binding to alpha7 nAChR in rat PC12 cells by FACS analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Critical Therapeutics

Curated by ChEMBL
LigandPNGBDBM50016199(CHEMBL3262145)
Affinity DataIC50:  32nMAssay Description:Inhibition of biotinylated alpha-bungarotoxin binding to alpha7 nAChR in rat PC12 cells by FACS analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Critical Therapeutics

Curated by ChEMBL
LigandPNGBDBM50016208(CHEMBL3262154)
Affinity DataIC50:  37nMAssay Description:Inhibition of biotinylated alpha-bungarotoxin binding to alpha7 nAChR in rat PC12 cells by FACS analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Critical Therapeutics

Curated by ChEMBL
LigandPNGBDBM50016212(CHEMBL3262158)
Affinity DataIC50:  40nMAssay Description:Inhibition of biotinylated alpha-bungarotoxin binding to alpha7 nAChR in rat PC12 cells by FACS analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Critical Therapeutics

Curated by ChEMBL
LigandPNGBDBM50016228(CHEMBL3262174)
Affinity DataIC50:  41nMAssay Description:Inhibition of biotinylated alpha-bungarotoxin binding to alpha7 nAChR in rat PC12 cells by FACS analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Critical Therapeutics

Curated by ChEMBL
LigandPNGBDBM50016226(CHEMBL3262172)
Affinity DataIC50:  42nMAssay Description:Inhibition of biotinylated alpha-bungarotoxin binding to alpha7 nAChR in rat PC12 cells by FACS analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Critical Therapeutics

Curated by ChEMBL
LigandPNGBDBM50016222(CHEMBL3262168)
Affinity DataIC50:  45nMAssay Description:Inhibition of biotinylated alpha-bungarotoxin binding to alpha7 nAChR in rat PC12 cells by FACS analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Critical Therapeutics

Curated by ChEMBL
LigandPNGBDBM50016189(CHEMBL3262135)
Affinity DataIC50:  46nMAssay Description:Inhibition of biotinylated alpha-bungarotoxin binding to alpha7 nAChR in rat PC12 cells by FACS analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Critical Therapeutics

Curated by ChEMBL
LigandPNGBDBM50016224(CHEMBL3262170)
Affinity DataIC50:  50nMAssay Description:Inhibition of biotinylated alpha-bungarotoxin binding to alpha7 nAChR in rat PC12 cells by FACS analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
Critical Therapeutics

Curated by ChEMBL
LigandPNGBDBM50016185(CHEMBL3262132)
Affinity DataIC50:  58nMAssay Description:Inhibition of human alpha4beta2 nAChR expressed in Xenopus oocytes by voltage clamp methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Critical Therapeutics

Curated by ChEMBL
LigandPNGBDBM50016216(CHEMBL3262162)
Affinity DataIC50:  60nMAssay Description:Inhibition of biotinylated alpha-bungarotoxin binding to alpha7 nAChR in rat PC12 cells by FACS analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Critical Therapeutics

Curated by ChEMBL
LigandPNGBDBM50016182(CHEMBL3262129)
Affinity DataIC50:  67nMAssay Description:Inhibition of biotinylated alpha-bungarotoxin binding to alpha7 nAChR in rat PC12 cells by FACS analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Critical Therapeutics

Curated by ChEMBL
LigandPNGBDBM50016207(CHEMBL3262153)
Affinity DataIC50:  70nMAssay Description:Inhibition of biotinylated alpha-bungarotoxin binding to alpha7 nAChR in rat PC12 cells by FACS analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Critical Therapeutics

Curated by ChEMBL
LigandPNGBDBM50016180(CHEMBL3262127)
Affinity DataIC50:  71nMAssay Description:Inhibition of biotinylated alpha-bungarotoxin binding to alpha7 nAChR in rat PC12 cells by FACS analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Critical Therapeutics

Curated by ChEMBL
LigandPNGBDBM50016213(CHEMBL3262159)
Affinity DataIC50:  74nMAssay Description:Inhibition of biotinylated alpha-bungarotoxin binding to alpha7 nAChR in rat PC12 cells by FACS analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Critical Therapeutics

Curated by ChEMBL
LigandPNGBDBM50016181(CHEMBL3262128)
Affinity DataIC50:  75nMAssay Description:Inhibition of biotinylated alpha-bungarotoxin binding to alpha7 nAChR in rat PC12 cells by FACS analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Critical Therapeutics

Curated by ChEMBL
LigandPNGBDBM50016188(CHEMBL3259843)
Affinity DataIC50:  79nMAssay Description:Inhibition of biotinylated alpha-bungarotoxin binding to alpha7 nAChR in rat PC12 cells by FACS analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Critical Therapeutics

Curated by ChEMBL
LigandPNGBDBM50016221(CHEMBL3262167)
Affinity DataIC50:  80nMAssay Description:Inhibition of biotinylated alpha-bungarotoxin binding to alpha7 nAChR in rat PC12 cells by FACS analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Critical Therapeutics

Curated by ChEMBL
LigandPNGBDBM50016192(CHEMBL3262138)
Affinity DataIC50:  85nMAssay Description:Inhibition of biotinylated alpha-bungarotoxin binding to alpha7 nAChR in rat PC12 cells by FACS analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Critical Therapeutics

Curated by ChEMBL
LigandPNGBDBM50016178(CHEMBL3262125)
Affinity DataIC50:  106nMAssay Description:Inhibition of biotinylated alpha-bungarotoxin binding to alpha7 nAChR in rat PC12 cells by FACS analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Critical Therapeutics

Curated by ChEMBL
LigandPNGBDBM50016191(CHEMBL3262137)
Affinity DataIC50:  107nMAssay Description:Inhibition of biotinylated alpha-bungarotoxin binding to alpha7 nAChR in rat PC12 cells by FACS analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Critical Therapeutics

Curated by ChEMBL
LigandPNGBDBM50016204(CHEMBL3262150)
Affinity DataIC50:  110nMAssay Description:Inhibition of biotinylated alpha-bungarotoxin binding to alpha7 nAChR in rat PC12 cells by FACS analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Critical Therapeutics

Curated by ChEMBL
LigandPNGBDBM50016196(CHEMBL3262142)
Affinity DataIC50:  132nMAssay Description:Inhibition of biotinylated alpha-bungarotoxin binding to alpha7 nAChR in rat PC12 cells by FACS analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Critical Therapeutics

Curated by ChEMBL
LigandPNGBDBM50016223(CHEMBL3262169)
Affinity DataIC50:  152nMAssay Description:Inhibition of biotinylated alpha-bungarotoxin binding to alpha7 nAChR in rat PC12 cells by FACS analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Critical Therapeutics

Curated by ChEMBL
LigandPNGBDBM50016193(CHEMBL3262139)
Affinity DataIC50:  153nMAssay Description:Inhibition of biotinylated alpha-bungarotoxin binding to alpha7 nAChR in rat PC12 cells by FACS analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Critical Therapeutics

Curated by ChEMBL
LigandPNGBDBM50016211(CHEMBL3262157)
Affinity DataIC50:  210nMAssay Description:Inhibition of biotinylated alpha-bungarotoxin binding to alpha7 nAChR in rat PC12 cells by FACS analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Critical Therapeutics

Curated by ChEMBL
LigandPNGBDBM50016214(CHEMBL3262160)
Affinity DataIC50:  220nMAssay Description:Inhibition of biotinylated alpha-bungarotoxin binding to alpha7 nAChR in rat PC12 cells by FACS analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Critical Therapeutics

Curated by ChEMBL
LigandPNGBDBM50016194(CHEMBL3262140)
Affinity DataIC50:  270nMAssay Description:Inhibition of biotinylated alpha-bungarotoxin binding to alpha7 nAChR in rat PC12 cells by FACS analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Critical Therapeutics

Curated by ChEMBL
LigandPNGBDBM50016215(CHEMBL3262161)
Affinity DataIC50:  280nMAssay Description:Inhibition of biotinylated alpha-bungarotoxin binding to alpha7 nAChR in rat PC12 cells by FACS analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Critical Therapeutics

Curated by ChEMBL
LigandPNGBDBM50016195(CHEMBL3262141)
Affinity DataIC50:  338nMAssay Description:Inhibition of biotinylated alpha-bungarotoxin binding to alpha7 nAChR in rat PC12 cells by FACS analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Critical Therapeutics

Curated by ChEMBL
LigandPNGBDBM50016219(CHEMBL3262165)
Affinity DataIC50:  340nMAssay Description:Inhibition of biotinylated alpha-bungarotoxin binding to alpha7 nAChR in rat PC12 cells by FACS analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Critical Therapeutics

Curated by ChEMBL
LigandPNGBDBM50016187(CHEMBL3262134)
Affinity DataIC50:  490nMAssay Description:Inhibition of biotinylated alpha-bungarotoxin binding to alpha7 nAChR in rat PC12 cells by FACS analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Critical Therapeutics

Curated by ChEMBL
LigandPNGBDBM50016203(CHEMBL3262149)
Affinity DataIC50:  560nMAssay Description:Inhibition of biotinylated alpha-bungarotoxin binding to alpha7 nAChR in rat PC12 cells by FACS analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Critical Therapeutics

Curated by ChEMBL
LigandPNGBDBM50016229(CHEMBL3262175)
Affinity DataIC50:  630nMAssay Description:Inhibition of biotinylated alpha-bungarotoxin binding to alpha7 nAChR in rat PC12 cells by FACS analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Critical Therapeutics

Curated by ChEMBL
LigandPNGBDBM50016206(CHEMBL3262152)
Affinity DataIC50:  680nMAssay Description:Inhibition of biotinylated alpha-bungarotoxin binding to alpha7 nAChR in rat PC12 cells by FACS analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Critical Therapeutics

Curated by ChEMBL
LigandPNGBDBM50016220(CHEMBL3262166)
Affinity DataIC50:  850nMAssay Description:Inhibition of biotinylated alpha-bungarotoxin binding to alpha7 nAChR in rat PC12 cells by FACS analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Critical Therapeutics

Curated by ChEMBL
LigandPNGBDBM50016201(CHEMBL3262147)
Affinity DataIC50:  1.08E+3nMAssay Description:Inhibition of biotinylated alpha-bungarotoxin binding to alpha7 nAChR in rat PC12 cells by FACS analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Critical Therapeutics

Curated by ChEMBL
LigandPNGBDBM50016186(CHEMBL3262133)
Affinity DataIC50:  1.58E+3nMAssay Description:Inhibition of biotinylated alpha-bungarotoxin binding to alpha7 nAChR in rat PC12 cells by FACS analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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