Compile Data Set for Download or QSAR
maximum 50k data
Found 24 Enz. Inhib. hit(s) with all data for entry = 50029596
TargetSubstance-K receptor(HAMSTER)
TBA

Curated by ChEMBL
LigandPNGBDBM50285956(4-(4-Chloro-phenylamino)-6-isopropyl-2-morpholin-4...)
Affinity DataKi:  15nMAssay Description:Inhibition constant for displacement of [3H]-NKA from Tachykinin receptor 2 found in hamster urinary bladder membrane (HUBM)More data for this Ligand-Target Pair
In DepthDetails Article
TargetSubstance-K receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50285956(4-(4-Chloro-phenylamino)-6-isopropyl-2-morpholin-4...)
Affinity DataKi:  15nMAssay Description:Inhibition constant for displacement of [3H]-NKA from Tachykinin receptor 2 found in hamster urinary bladder membrane (HUBM)More data for this Ligand-Target Pair
In DepthDetails Article
TargetSubstance-K receptor(HAMSTER)
TBA

Curated by ChEMBL
LigandPNGBDBM50285943((4-Chloro-phenyl)-(2-morpholin-4-yl-8-propyl-9H-pu...)
Affinity DataKi:  54nMAssay Description:Inhibition constant for displacement of [3H]-NKA from Tachykinin receptor 2 found in hamster urinary bladder membrane (HUBM)More data for this Ligand-Target Pair
In DepthDetails Article
TargetSubstance-K receptor(HAMSTER)
TBA

Curated by ChEMBL
LigandPNGBDBM50285955((4-Chloro-phenyl)-(8-isopropyl-2-morpholin-4-yl-9H...)
Affinity DataKi:  67nMAssay Description:Inhibition constant for displacement of [3H]-NKA from Tachykinin receptor 2 found in hamster urinary bladder membrane (HUBM)More data for this Ligand-Target Pair
In DepthDetails Article
TargetSubstance-K receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50285955((4-Chloro-phenyl)-(8-isopropyl-2-morpholin-4-yl-9H...)
Affinity DataKi:  67nMAssay Description:Inhibition constant for displacement of [3H]-NKA from Tachykinin receptor 2 found in hamster urinary bladder membrane (HUBM)More data for this Ligand-Target Pair
In DepthDetails Article
TargetSubstance-K receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50285944((4-Chloro-phenyl)-(8-ethyl-2-morpholin-4-yl-9H-pur...)
Affinity DataKi:  520nMAssay Description:Inhibition constant for displacement of [3H]-NKA from Tachykinin receptor 2 found in hamster urinary bladder membrane (HUBM)More data for this Ligand-Target Pair
In DepthDetails Article
TargetSubstance-K receptor(HAMSTER)
TBA

Curated by ChEMBL
LigandPNGBDBM50285944((4-Chloro-phenyl)-(8-ethyl-2-morpholin-4-yl-9H-pur...)
Affinity DataKi:  520nMAssay Description:Inhibition constant for displacement of [3H]-NKA from Tachykinin receptor 2 found in hamster urinary bladder membrane (HUBM)More data for this Ligand-Target Pair
In DepthDetails Article
TargetSubstance-K receptor(HAMSTER)
TBA

Curated by ChEMBL
LigandPNGBDBM50285950(4-(4-Chloro-phenylamino)-2-morpholin-4-yl-quinazol...)
Affinity DataKi:  820nMAssay Description:Inhibition constant for displacement of [3H]-NKA from Tachykinin receptor 2 found in hamster urinary bladder membrane (HUBM)More data for this Ligand-Target Pair
In DepthDetails Article
TargetSubstance-K receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50285957(1-[8-Isopropyl-6-(4-trifluoromethyl-phenylamino)-9...)
Affinity DataKi:  1.77E+3nMAssay Description:Displacement of [3H]-NKA from the cloned human Tachykinin receptor 2 which has been expressed in baculovirus infected insect sf21 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSubstance-K receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50285959(1-[6-(4-Chloro-phenylamino)-8-isopropyl-9H-purin-2...)
Affinity DataKi:  2.10E+3nMAssay Description:Displacement of [3H]-NKA from the cloned human Tachykinin receptor 2 which has been expressed in baculovirus infected insect sf21 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSubstance-K receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50285945(1-[6-(4-Chloro-phenylamino)-8-isopropyl-9H-purin-2...)
Affinity DataKi:  2.24E+3nMAssay Description:Displacement of [3H]-NKA from the cloned human Tachykinin receptor 2 which has been expressed in baculovirus infected insect sf21 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSubstance-K receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50285943((4-Chloro-phenyl)-(2-morpholin-4-yl-8-propyl-9H-pu...)
Affinity DataKi:  2.34E+3nMAssay Description:Inhibition constant for displacement of [3H]-NKA from the cloned human NK2 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSubstance-K receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50285952(CHEMBL321137 | N*2*-(3-Amino-propyl)-N*6*-(4-chlor...)
Affinity DataKi:  2.55E+3nMAssay Description:Displacement of [3H]-NKA from the cloned human Tachykinin receptor 2 which has been expressed in baculovirus infected insect sf21 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSubstance-K receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50285948((8-Isopropyl-2-morpholin-4-yl-9H-purin-6-yl)-(4-tr...)
Affinity DataKi:  2.85E+3nMAssay Description:Displacement of [3H]-NKA from the cloned human Tachykinin receptor 2 which has been expressed in baculovirus infected insect sf21 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSubstance-K receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50285946((4-Chloro-phenyl)-[2-(4,4-dimethoxy-piperidin-1-yl...)
Affinity DataKi:  3.44E+3nMAssay Description:Displacement of [3H]-NKA from the cloned human Tachykinin receptor 2 which has been expressed in baculovirus infected insect sf21 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSubstance-K receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50285949(CHEMBL97140 | N*6*-(4-Chloro-phenyl)-8-isopropyl-N...)
Affinity DataKi:  3.49E+3nMAssay Description:Displacement of [3H]-NKA from the cloned human Tachykinin receptor 2 which has been expressed in baculovirus infected insect sf21 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSubstance-K receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50285958((4-Chloro-phenyl)-[2-(1,4-dioxa-8-aza-spiro[4.5]de...)
Affinity DataKi:  4.36E+3nMAssay Description:Displacement of [3H]-NKA from the cloned human Tachykinin receptor 2 which has been expressed in baculovirus infected insect sf21 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSubstance-K receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50285961(CHEMBL318880 | N*2*-Benzyl-N*6*-(4-chloro-phenyl)-...)
Affinity DataKi:  5.58E+3nMAssay Description:Displacement of [3H]-NKA from the cloned human Tachykinin receptor 2 which has been expressed in baculovirus infected insect sf21 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSubstance-K receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50285951(1-[6-(4-Chloro-phenylamino)-8-isopropyl-9H-purin-2...)
Affinity DataKi:  5.89E+3nMAssay Description:Displacement of [3H]-NKA from the cloned human Tachykinin receptor 2 which has been expressed in baculovirus infected insect sf21 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSubstance-K receptor(HAMSTER)
TBA

Curated by ChEMBL
LigandPNGBDBM50285954((4-Chloro-phenyl)-(8-methyl-2-morpholin-4-yl-9H-pu...)
Affinity DataKi:  6.60E+3nMAssay Description:Inhibition constant for displacement of [3H]-NKA from Tachykinin receptor 2 found in hamster urinary bladder membrane (HUBM)More data for this Ligand-Target Pair
In DepthDetails Article
TargetSubstance-K receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50285954((4-Chloro-phenyl)-(8-methyl-2-morpholin-4-yl-9H-pu...)
Affinity DataKi:  6.60E+3nMAssay Description:Inhibition constant for displacement of [3H]-NKA from Tachykinin receptor 2 found in hamster urinary bladder membrane (HUBM)More data for this Ligand-Target Pair
In DepthDetails Article
TargetSubstance-K receptor(HAMSTER)
TBA

Curated by ChEMBL
LigandPNGBDBM50285947(4-(4-Chloro-phenylamino)-2-morpholin-4-yl-quinazol...)
Affinity DataKi:  2.03E+4nMAssay Description:Inhibition constant for displacement of [3H]-NKA from Tachykinin receptor 2 found in hamster urinary bladder membrane (HUBM)More data for this Ligand-Target Pair
In DepthDetails Article
TargetSubstance-K receptor(HAMSTER)
TBA

Curated by ChEMBL
LigandPNGBDBM50285953((4-Chloro-phenyl)-(2-morpholin-4-yl-quinazolin-4-y...)
Affinity DataKi:  2.95E+4nMAssay Description:Inhibition constant for displacement of [3H]-NKA from Tachykinin receptor 2 found in hamster urinary bladder membrane (HUBM)More data for this Ligand-Target Pair
In DepthDetails Article
TargetSubstance-K receptor(HAMSTER)
TBA

Curated by ChEMBL
LigandPNGBDBM50285960(4-(4-Chloro-phenylamino)-2-morpholin-4-yl-quinazol...)
Affinity DataKi:  5.87E+4nMAssay Description:Inhibition constant for displacement of [3H]-NKA from Tachykinin receptor 2 found in hamster urinary bladder membrane (HUBM)More data for this Ligand-Target Pair
In DepthDetails Article