Compile Data Set for Download or QSAR
maximum 50k data
Found 45 Enz. Inhib. hit(s) with all data for entry = 50030025
TargetProgesterone receptor(Oryctolagus cuniculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50290345(7-(3,4-Difluoro-benzyl)-1-(4-fluoro-phenyl)-4,5,6,...)
Affinity DataIC50:  2nMAssay Description:Binding affinity determined by ability to displace [3H]-R5020 radioligand using uterine progesterone receptor obtained from estrogen-primed rabbitMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProgesterone receptor(Oryctolagus cuniculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50290353(CHEMBL422241 | [1-[1-(4-Fluoro-phenyl)-7-naphthale...)
Affinity DataIC50:  2.30nMAssay Description:Binding affinity determined by ability to displace [3H]-R5020 radioligand using uterine progesterone receptor obtained from estrogen-primed rabbitMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProgesterone receptor(Oryctolagus cuniculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50290364(7-Benzyl-1-(4-fluoro-phenyl)-4,5,6,7-tetrahydro-1H...)
Affinity DataIC50:  3nMAssay Description:Binding affinity determined by ability to displace [3H]-R5020 radioligand using uterine progesterone receptor obtained from estrogen-primed rabbitMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProgesterone receptor(Oryctolagus cuniculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50290359(1-(4-Fluoro-phenyl)-7-naphthalen-1-ylmethyl-4,5,6,...)
Affinity DataIC50:  3.20nMAssay Description:Binding affinity determined by ability to displace [3H]-R5020 radioligand using uterine progesterone receptor obtained from estrogen-primed rabbitMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProgesterone receptor(Oryctolagus cuniculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50290336(Acetic acid acetoxy-[1-(4-fluoro-phenyl)-7-naphtha...)
Affinity DataIC50:  5.30nMAssay Description:Binding affinity determined by ability to displace [3H]-R5020 radioligand using uterine progesterone receptor obtained from estrogen-primed rabbitMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProgesterone receptor(Oryctolagus cuniculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50290361(7-Naphthalen-1-ylmethyl-1-phenyl-4,5,6,7-tetrahydr...)
Affinity DataIC50:  6nMAssay Description:Binding affinity determined by ability to displace [3H]-R5020 radioligand using uterine progesterone receptor obtained from estrogen-primed rabbitMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProgesterone receptor(Oryctolagus cuniculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50290333(7-(4-Fluoro-benzyl)-1-(4-fluoro-phenyl)-4,5,6,7-te...)
Affinity DataIC50:  6.5nMAssay Description:Binding affinity determined by ability to displace [3H]-R5020 radioligand using uterine progesterone receptor obtained from estrogen-primed rabbitMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProgesterone receptor(Oryctolagus cuniculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50290356(1-(4-Fluoro-phenyl)-7-(4-methyl-benzyl)-4,5,6,7-te...)
Affinity DataIC50:  7.70nMAssay Description:Binding affinity determined by ability to displace [3H]-R5020 radioligand using uterine progesterone receptor obtained from estrogen-primed rabbitMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProgesterone receptor(Oryctolagus cuniculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50290334(1-(4-Chloro-phenyl)-7-naphthalen-1-ylmethyl-4,5,6,...)
Affinity DataIC50:  9nMAssay Description:Binding affinity determined by ability to displace [3H]-R5020 radioligand using uterine progesterone receptor obtained from estrogen-primed rabbitMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProgesterone receptor(Oryctolagus cuniculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50290362(7-(2-Chloro-benzyl)-1-(4-fluoro-phenyl)-4,5,6,7-te...)
Affinity DataIC50:  11nMAssay Description:Binding affinity determined by ability to displace [3H]-R5020 radioligand using uterine progesterone receptor obtained from estrogen-primed rabbitMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProgesterone receptor(Oryctolagus cuniculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50290358(7-(4-Chloro-benzyl)-1-(4-fluoro-phenyl)-4,5,6,7-te...)
Affinity DataIC50:  12nMAssay Description:Binding affinity determined by ability to displace [3H]-R5020 radioligand using uterine progesterone receptor obtained from estrogen-primed rabbitMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProgesterone receptor(Oryctolagus cuniculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50290349(1-(4-Methoxy-phenyl)-7-naphthalen-1-ylmethyl-4,5,6...)
Affinity DataIC50:  13nMAssay Description:Binding affinity determined by ability to displace [3H]-R5020 radioligand using uterine progesterone receptor obtained from estrogen-primed rabbitMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProgesterone receptor(Oryctolagus cuniculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50290338(1-(4-Fluoro-phenyl)-7-(3-methoxy-benzyl)-octahydro...)
Affinity DataIC50:  17nMAssay Description:Binding affinity determined by ability to displace [3H]-R5020 radioligand using uterine progesterone receptor obtained from estrogen-primed rabbitMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProgesterone receptor(Oryctolagus cuniculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50290354(1-(4-Fluoro-phenyl)-7-naphthalen-1-ylmethyl-4,5,6,...)
Affinity DataIC50:  41nMAssay Description:Binding affinity determined by ability to displace [3H]-R5020 radioligand using uterine progesterone receptor obtained from estrogen-primed rabbitMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProgesterone receptor(Oryctolagus cuniculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50290375(CHEMBL314154 | N-[1-[1-(4-Fluoro-phenyl)-7-naphtha...)
Affinity DataIC50:  49nMAssay Description:Binding affinity determined by ability to displace [3H]-R5020 radioligand using uterine progesterone receptor obtained from estrogen-primed rabbitMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProgesterone receptor(Oryctolagus cuniculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50290360(CHEMBL315787 | [1-(4-Fluoro-phenyl)-7-naphthalen-1...)
Affinity DataIC50:  52nMAssay Description:Binding affinity determined by ability to displace [3H]-R5020 radioligand using uterine progesterone receptor obtained from estrogen-primed rabbitMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProgesterone receptor(Oryctolagus cuniculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50290372(1-(4-Fluoro-phenyl)-7-naphthalen-2-ylmethyl-octahy...)
Affinity DataIC50:  56nMAssay Description:Binding affinity determined by ability to displace [3H]-R5020 radioligand using uterine progesterone receptor obtained from estrogen-primed rabbitMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProgesterone receptor(Oryctolagus cuniculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50290368(1-(3-Chloro-phenyl)-7-naphthalen-1-ylmethyl-4,5,6,...)
Affinity DataIC50:  69nMAssay Description:Binding affinity determined by ability to displace [3H]-R5020 radioligand using uterine progesterone receptor obtained from estrogen-primed rabbitMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProgesterone receptor(Oryctolagus cuniculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50290352(Acetic acid 1-(4-fluoro-phenyl)-7-naphthalen-1-ylm...)
Affinity DataIC50:  73nMAssay Description:Binding affinity determined by ability to displace [3H]-R5020 radioligand using uterine progesterone receptor obtained from estrogen-primed rabbitMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProgesterone receptor(Oryctolagus cuniculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50290344(CHEMBL420978 | Carbonic acid ethyl ester 1-(4-fluo...)
Affinity DataIC50:  90nMAssay Description:Binding affinity determined by ability to displace [3H]-R5020 radioligand using uterine progesterone receptor obtained from estrogen-primed rabbitMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProgesterone receptor(Oryctolagus cuniculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50290363(3-[1,3]Dioxolan-2-yl-1-(4-fluoro-phenyl)-7-naphtha...)
Affinity DataIC50:  97nMAssay Description:Binding affinity determined by ability to displace [3H]-R5020 radioligand using uterine progesterone receptor obtained from estrogen-primed rabbitMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProgesterone receptor(Oryctolagus cuniculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50290351(1-(4-Fluoro-phenyl)-7-naphthalen-1-ylmethyl-3-viny...)
Affinity DataIC50:  147nMAssay Description:Binding affinity determined by ability to displace [3H]-R5020 radioligand using uterine progesterone receptor obtained from estrogen-primed rabbitMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProgesterone receptor(Oryctolagus cuniculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50290376(1-(4-Fluoro-phenyl)-7-(4-methoxy-benzyl)-4,5,6,7-t...)
Affinity DataIC50:  163nMAssay Description:Binding affinity determined by ability to displace [3H]-R5020 radioligand using uterine progesterone receptor obtained from estrogen-primed rabbitMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProgesterone receptor(Oryctolagus cuniculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50290374(Benzoic acid 1-(4-fluoro-phenyl)-7-naphthalen-1-yl...)
Affinity DataIC50:  182nMAssay Description:Binding affinity determined by ability to displace [3H]-R5020 radioligand using uterine progesterone receptor obtained from estrogen-primed rabbitMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProgesterone receptor(Oryctolagus cuniculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50290369(1-[1-(4-Fluoro-phenyl)-7-naphthalen-1-ylmethyl-4,5...)
Affinity DataIC50:  236nMAssay Description:Binding affinity determined by ability to displace [3H]-R5020 radioligand using uterine progesterone receptor obtained from estrogen-primed rabbitMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProgesterone receptor(Oryctolagus cuniculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50290355(CHEMBL82911 | N'-[1-[1-(4-Fluoro-phenyl)-7-naphtha...)
Affinity DataIC50:  547nMAssay Description:Binding affinity determined by ability to displace [3H]-R5020 radioligand using uterine progesterone receptor obtained from estrogen-primed rabbitMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProgesterone receptor(Oryctolagus cuniculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50290343(1-(4-Fluoro-phenyl)-7-naphthalen-1-ylmethyl-4,5,6,...)
Affinity DataIC50:  628nMAssay Description:Binding affinity determined by ability to displace [3H]-R5020 radioligand using uterine progesterone receptor obtained from estrogen-primed rabbitMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProgesterone receptor(Oryctolagus cuniculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50290371(1-[1-(4-Fluoro-phenyl)-7-naphthalen-1-ylmethyl-4,5...)
Affinity DataIC50:  690nMAssay Description:Binding affinity determined by ability to displace [3H]-R5020 radioligand using uterine progesterone receptor obtained from estrogen-primed rabbitMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProgesterone receptor(Oryctolagus cuniculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50290337(4-(3-Formyl-7-naphthalen-1-ylmethyl-4,5,6,7-tetrah...)
Affinity DataIC50:  851nMAssay Description:Binding affinity determined by ability to displace [3H]-R5020 radioligand using uterine progesterone receptor obtained from estrogen-primed rabbitMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProgesterone receptor(Oryctolagus cuniculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50290340(1-[1-(4-Fluoro-phenyl)-7-naphthalen-1-ylmethyl-4,5...)
Affinity DataIC50:  1.00E+3nMAssay Description:Binding affinity determined by ability to displace [3H]-R5020 radioligand using uterine progesterone receptor obtained from estrogen-primed rabbitMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProgesterone receptor(Oryctolagus cuniculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50290335(7-(4-tert-Butyl-benzyl)-1-(4-fluoro-phenyl)-4,5,6,...)
Affinity DataIC50:  1.00E+3nMAssay Description:Binding affinity determined by ability to displace [3H]-R5020 radioligand using uterine progesterone receptor obtained from estrogen-primed rabbitMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProgesterone receptor(Oryctolagus cuniculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50290350(CHEMBL315817 | Diethyl-[1-(4-fluoro-phenyl)-7-naph...)
Affinity DataIC50:  1.38E+3nMAssay Description:Binding affinity determined by ability to displace [3H]-R5020 radioligand using uterine progesterone receptor obtained from estrogen-primed rabbitMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProgesterone receptor(Oryctolagus cuniculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50290370(Benzyl-[1-(4-fluoro-phenyl)-7-naphthalen-1-ylmethy...)
Affinity DataIC50:  1.38E+3nMAssay Description:Binding affinity determined by ability to displace [3H]-R5020 radioligand using uterine progesterone receptor obtained from estrogen-primed rabbitMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProgesterone receptor(Oryctolagus cuniculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50290347(CHEMBL84715 | [1-(4-Fluoro-phenyl)-7-naphthalen-1-...)
Affinity DataIC50:  1.57E+3nMAssay Description:Binding affinity determined by ability to displace [3H]-R5020 radioligand using uterine progesterone receptor obtained from estrogen-primed rabbitMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProgesterone receptor(Oryctolagus cuniculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50290373(1-[1-(4-Fluoro-phenyl)-7-naphthalen-1-ylmethyl-4,5...)
Affinity DataIC50:  1.76E+3nMAssay Description:Binding affinity determined by ability to displace [3H]-R5020 radioligand using uterine progesterone receptor obtained from estrogen-primed rabbitMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProgesterone receptor(Oryctolagus cuniculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50290366(7-(3,4-Dimethoxy-benzyl)-1-(4-fluoro-phenyl)-4,5,6...)
Affinity DataIC50:  1.89E+3nMAssay Description:Binding affinity determined by ability to displace [3H]-R5020 radioligand using uterine progesterone receptor obtained from estrogen-primed rabbitMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProgesterone receptor(Oryctolagus cuniculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50290341(1-(4-Fluoro-phenyl)-7-(4-isopropyl-benzyl)-4,5,6,7...)
Affinity DataIC50:  2.20E+3nMAssay Description:Binding affinity determined by ability to displace [3H]-R5020 radioligand using uterine progesterone receptor obtained from estrogen-primed rabbitMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProgesterone receptor(Oryctolagus cuniculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50290342(1-(4-Fluoro-phenyl)-7-naphthalen-1-ylmethyl-4,5,6,...)
Affinity DataIC50:  3.00E+3nMAssay Description:Binding affinity determined by ability to displace [3H]-R5020 radioligand using uterine progesterone receptor obtained from estrogen-primed rabbitMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProgesterone receptor(Oryctolagus cuniculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50290346(CHEMBL85913 | Octanoic acid 1-(4-fluoro-phenyl)-7-...)
Affinity DataIC50:  4.01E+3nMAssay Description:Binding affinity determined by ability to displace [3H]-R5020 radioligand using uterine progesterone receptor obtained from estrogen-primed rabbitMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProgesterone receptor(Oryctolagus cuniculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50290367(Acetic acid [1-[1-(4-fluoro-phenyl)-7-naphthalen-1...)
Affinity DataIC50: >1.00E+4nMAssay Description:Binding affinity determined by ability to displace [3H]-R5020 radioligand using uterine progesterone receptor obtained from estrogen-primed rabbitMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProgesterone receptor(Oryctolagus cuniculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50290365(1-(4-Fluoro-phenyl)-3-(N'-[(E)-methylene]benzenesu...)
Affinity DataIC50: >1.00E+4nMAssay Description:Binding affinity determined by ability to displace [3H]-R5020 radioligand using uterine progesterone receptor obtained from estrogen-primed rabbitMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProgesterone receptor(Oryctolagus cuniculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50290348(1-(4-Fluoro-phenyl)-7-naphthalen-1-ylmethyl-4,5,6,...)
Affinity DataIC50: >1.00E+4nMAssay Description:Binding affinity determined by ability to displace [3H]-R5020 radioligand using uterine progesterone receptor obtained from estrogen-primed rabbitMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProgesterone receptor(Oryctolagus cuniculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50290332(4-(3-Formyl-7-naphthalen-1-ylmethyl-4,5,6,7-tetrah...)
Affinity DataIC50: >1.00E+4nMAssay Description:Binding affinity determined by ability to displace [3H]-R5020 radioligand using uterine progesterone receptor obtained from estrogen-primed rabbitMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProgesterone receptor(Oryctolagus cuniculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50290357(7-Biphenyl-4-ylmethyl-1-(4-fluoro-phenyl)-4,5,6,7-...)
Affinity DataIC50:  1.00E+4nMAssay Description:Binding affinity determined by ability to displace [3H]-R5020 radioligand using uterine progesterone receptor obtained from estrogen-primed rabbitMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProgesterone receptor(Oryctolagus cuniculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50290339(Benzoic acid [1-[1-(4-fluoro-phenyl)-7-naphthalen-...)
Affinity DataIC50: >1.00E+4nMAssay Description:Binding affinity determined by ability to displace [3H]-R5020 radioligand using uterine progesterone receptor obtained from estrogen-primed rabbitMore data for this Ligand-Target Pair
In DepthDetails Article