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Found 62 Enz. Inhib. hit(s) with all data for entry = 50048372
LigandPNGBDBM50213551(CHEMBL90618)
Affinity DataIC50:  0.0300nMAssay Description:In vitro displacement of [125I]angiotensin II from rat liver (Angiotensin 1 receptor) membrane preparationMore data for this Ligand-Target Pair
In DepthDetails
LigandPNGBDBM50213505(CHEMBL314975)
Affinity DataIC50:  0.0700nMAssay Description:In vitro displacement of [125I]angiotensin II from rat liver (Angiotensin 1 receptor) membrane preparationMore data for this Ligand-Target Pair
In DepthDetails
LigandPNGBDBM50213561(CHEMBL312937)
Affinity DataIC50:  0.0700nMAssay Description:In vitro displacement of [125I]angiotensin II from rat liver (Angiotensin 1 receptor) membrane preparationMore data for this Ligand-Target Pair
In DepthDetails
LigandPNGBDBM50213458(CHEMBL90672)
Affinity DataIC50:  0.100nMAssay Description:In vitro displacement of [125I]angiotensin II from rat liver (Angiotensin 1 receptor) membrane preparationMore data for this Ligand-Target Pair
In DepthDetails
LigandPNGBDBM50213500(CHEMBL86337)
Affinity DataIC50:  0.100nMAssay Description:In vitro displacement of [125I]angiotensin II from rat liver (Angiotensin 1 receptor) membrane preparationMore data for this Ligand-Target Pair
In DepthDetails
LigandPNGBDBM50213456(CHEMBL315000)
Affinity DataIC50:  0.100nMAssay Description:In vitro displacement of [125I]angiotensin II from rat liver (Angiotensin 1 receptor) membrane preparationMore data for this Ligand-Target Pair
In DepthDetails
LigandPNGBDBM50213457(CHEMBL84686)
Affinity DataIC50:  0.100nMAssay Description:In vitro displacement of [125I]angiotensin II from rat liver (Angiotensin 1 receptor) membrane preparationMore data for this Ligand-Target Pair
In DepthDetails
LigandPNGBDBM50213504(CHEMBL89369)
Affinity DataIC50:  0.100nMAssay Description:In vitro displacement of [125I]angiotensin II from rat liver (Angiotensin 1 receptor) membrane preparationMore data for this Ligand-Target Pair
In DepthDetails
LigandPNGBDBM50213460(CHEMBL85081)
Affinity DataIC50:  0.100nMAssay Description:In vitro displacement of [125I]angiotensin II from rat liver (Angiotensin 1 receptor) membrane preparationMore data for this Ligand-Target Pair
In DepthDetails
LigandPNGBDBM50213567(CHEMBL315983)
Affinity DataIC50:  0.100nMAssay Description:In vitro displacement of [125I]angiotensin II from rat liver (Angiotensin 1 receptor) membrane preparationMore data for this Ligand-Target Pair
In DepthDetails
LigandPNGBDBM50213552(CHEMBL328302)
Affinity DataIC50:  0.100nMAssay Description:In vitro displacement of [125I]angiotensin II from rat liver (Angiotensin 1 receptor) membrane preparationMore data for this Ligand-Target Pair
In DepthDetails
LigandPNGBDBM50213591(CHEMBL84795)
Affinity DataIC50:  0.100nMAssay Description:In vitro displacement of [125I]angiotensin II from rat liver (Angiotensin 1 receptor) membrane preparationMore data for this Ligand-Target Pair
In DepthDetails
LigandPNGBDBM50213499(CHEMBL88653)
Affinity DataIC50:  0.150nMAssay Description:In vitro displacement of [125I]angiotensin II from rat liver (Angiotensin 1 receptor) membrane preparationMore data for this Ligand-Target Pair
In DepthDetails
LigandPNGBDBM50213569(CHEMBL78866)
Affinity DataIC50:  0.200nMAssay Description:In vitro displacement of [125I]angiotensin II from rat liver (Angiotensin 1 receptor) membrane preparationMore data for this Ligand-Target Pair
In DepthDetails
LigandPNGBDBM50213550(CHEMBL87847)
Affinity DataIC50:  0.200nMAssay Description:In vitro displacement of [125I]angiotensin II from rat liver (Angiotensin 1 receptor) membrane preparationMore data for this Ligand-Target Pair
In DepthDetails
LigandPNGBDBM50213557(CHEMBL309602)
Affinity DataIC50:  0.200nMAssay Description:In vitro displacement of [125I]angiotensin II from rat liver (Angiotensin 1 receptor) membrane preparationMore data for this Ligand-Target Pair
In DepthDetails
LigandPNGBDBM50213564(CHEMBL316234)
Affinity DataIC50:  0.200nMAssay Description:In vitro displacement of [125I]angiotensin II from rat liver (Angiotensin 1 receptor) membrane preparationMore data for this Ligand-Target Pair
In DepthDetails
LigandPNGBDBM50213554(CHEMBL314527)
Affinity DataIC50:  0.200nMAssay Description:In vitro displacement of [125I]angiotensin II from rat liver (Angiotensin 1 receptor) membrane preparationMore data for this Ligand-Target Pair
In DepthDetails
LigandPNGBDBM50213461(CHEMBL407824)
Affinity DataIC50:  0.300nMAssay Description:In vitro displacement of [125I]angiotensin II from rat liver (Angiotensin 1 receptor) membrane preparationMore data for this Ligand-Target Pair
In DepthDetails
LigandPNGBDBM50213568(CHEMBL87108)
Affinity DataIC50:  0.300nMAssay Description:In vitro displacement of [125I]angiotensin II from rat liver (Angiotensin 1 receptor) membrane preparationMore data for this Ligand-Target Pair
In DepthDetails
LigandPNGBDBM50213562(CHEMBL327455)
Affinity DataIC50:  0.300nMAssay Description:In vitro displacement of [125I]angiotensin II from rat liver (Angiotensin 1 receptor) membrane preparationMore data for this Ligand-Target Pair
In DepthDetails
LigandPNGBDBM50213555(CHEMBL87030)
Affinity DataIC50:  0.400nMAssay Description:In vitro displacement of [125I]angiotensin II from rat liver (Angiotensin 1 receptor) membrane preparationMore data for this Ligand-Target Pair
In DepthDetails
LigandPNGBDBM50213583(CHEMBL421357)
Affinity DataIC50:  0.5nMAssay Description:In vitro displacement of [125I]angiotensin II from rat liver (Angiotensin 1 receptor) membrane preparationMore data for this Ligand-Target Pair
In DepthDetails
LigandPNGBDBM50031537(2-Butyl-3-(N'-propylureidylsulfonyl-biphenyl-4-ylm...)
Affinity DataIC50:  0.5nMAssay Description:In vitro displacement of [125I]angiotensin II from rat liver (Angiotensin 1 receptor) membrane preparationMore data for this Ligand-Target Pair
In DepthDetails
LigandPNGBDBM50213565(CHEMBL88349)
Affinity DataIC50:  0.5nMAssay Description:In vitro displacement of [125I]angiotensin II from rat liver (Angiotensin 1 receptor) membrane preparationMore data for this Ligand-Target Pair
In DepthDetails
LigandPNGBDBM50213489(CHEMBL316344)
Affinity DataIC50:  0.700nMAssay Description:In vitro displacement of [125I]angiotensin II from rat liver (Angiotensin 1 receptor) membrane preparationMore data for this Ligand-Target Pair
In DepthDetails
LigandPNGBDBM50213459(CHEMBL313032)
Affinity DataIC50:  1nMAssay Description:In vitro displacement of [125I]angiotensin II from rat liver (Angiotensin 1 receptor) membrane preparationMore data for this Ligand-Target Pair
In DepthDetails
LigandPNGBDBM50213560(CHEMBL87029)
Affinity DataIC50:  1.20nMAssay Description:In vitro displacement of [125I]angiotensin II from rat liver (Angiotensin 1 receptor) membrane preparationMore data for this Ligand-Target Pair
In DepthDetails
LigandPNGBDBM50213488(CHEMBL431466)
Affinity DataIC50:  1.30nMAssay Description:In vitro displacement of [125I]angiotensin II from rat liver (Angiotensin 1 receptor) membrane preparationMore data for this Ligand-Target Pair
In DepthDetails
TargetType-1/Type-2 angiotensin II receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50213488(CHEMBL431466)
Affinity DataIC50:  1.30nMAssay Description:In vitro displacement of [125I]angiotensin II from angiotensin 2 receptor on rabbit uterus membrane preparationMore data for this Ligand-Target Pair
In DepthDetails
TargetType-1/Type-2 angiotensin II receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50213505(CHEMBL314975)
Affinity DataIC50:  1.70nMAssay Description:In vitro displacement of [125I]angiotensin II from angiotensin 2 receptor on rabbit uterus membrane preparationMore data for this Ligand-Target Pair
In DepthDetails
LigandPNGBDBM50213556(CHEMBL310610)
Affinity DataIC50:  1.90nMAssay Description:In vitro displacement of [125I]angiotensin II from rat liver (Angiotensin 1 receptor) membrane preparationMore data for this Ligand-Target Pair
In DepthDetails
LigandPNGBDBM50213455(CHEMBL86603)
Affinity DataIC50:  2.30nMAssay Description:In vitro displacement of [125I]angiotensin II from rat liver (Angiotensin 1 receptor) membrane preparationMore data for this Ligand-Target Pair
In DepthDetails
TargetType-1/Type-2 angiotensin II receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50213550(CHEMBL87847)
Affinity DataIC50:  2.5nMAssay Description:In vitro displacement of [125I]angiotensin II from angiotensin 2 receptor on rabbit uterus membrane preparationMore data for this Ligand-Target Pair
In DepthDetails
TargetType-1/Type-2 angiotensin II receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50213458(CHEMBL90672)
Affinity DataIC50:  3.40nMAssay Description:In vitro displacement of [125I]angiotensin II from angiotensin 2 receptor on rabbit uterus membrane preparationMore data for this Ligand-Target Pair
In DepthDetails
TargetType-1/Type-2 angiotensin II receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50213567(CHEMBL315983)
Affinity DataIC50:  5.40nMAssay Description:In vitro displacement of [125I]angiotensin II from angiotensin 2 receptor on rabbit uterus membrane preparationMore data for this Ligand-Target Pair
In DepthDetails
TargetType-1/Type-2 angiotensin II receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50213564(CHEMBL316234)
Affinity DataIC50:  5.80nMAssay Description:In vitro displacement of [125I]angiotensin II from angiotensin 2 receptor on rabbit uterus membrane preparationMore data for this Ligand-Target Pair
In DepthDetails
TargetType-1/Type-2 angiotensin II receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50213504(CHEMBL89369)
Affinity DataIC50:  6.80nMAssay Description:In vitro displacement of [125I]angiotensin II from angiotensin 2 receptor on rabbit uterus membrane preparationMore data for this Ligand-Target Pair
In DepthDetails
TargetType-1/Type-2 angiotensin II receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50213456(CHEMBL315000)
Affinity DataIC50:  7nMAssay Description:In vitro displacement of [125I]angiotensin II from angiotensin 2 receptor on rabbit uterus membrane preparationMore data for this Ligand-Target Pair
In DepthDetails
TargetType-1/Type-2 angiotensin II receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50213561(CHEMBL312937)
Affinity DataIC50:  7.80nMAssay Description:In vitro displacement of [125I]angiotensin II from angiotensin 2 receptor on rabbit uterus membrane preparationMore data for this Ligand-Target Pair
In DepthDetails
TargetType-1/Type-2 angiotensin II receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50213499(CHEMBL88653)
Affinity DataIC50:  9nMAssay Description:In vitro displacement of [125I]angiotensin II from angiotensin 2 receptor on rabbit uterus membrane preparationMore data for this Ligand-Target Pair
In DepthDetails
TargetType-1/Type-2 angiotensin II receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50213554(CHEMBL314527)
Affinity DataIC50:  9.5nMAssay Description:In vitro displacement of [125I]angiotensin II from angiotensin 2 receptor on rabbit uterus membrane preparationMore data for this Ligand-Target Pair
In DepthDetails
TargetType-1/Type-2 angiotensin II receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50213562(CHEMBL327455)
Affinity DataIC50:  11nMAssay Description:In vitro displacement of [125I]angiotensin II from angiotensin 2 receptor on rabbit uterus membrane preparationMore data for this Ligand-Target Pair
In DepthDetails
TargetType-1/Type-2 angiotensin II receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50213500(CHEMBL86337)
Affinity DataIC50:  14nMAssay Description:In vitro displacement of [125I]angiotensin II from angiotensin 2 receptor on rabbit uterus membrane preparationMore data for this Ligand-Target Pair
In DepthDetails
TargetType-1/Type-2 angiotensin II receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50213591(CHEMBL84795)
Affinity DataIC50:  17nMAssay Description:In vitro displacement of [125I]angiotensin II from angiotensin 2 receptor on rabbit uterus membrane preparationMore data for this Ligand-Target Pair
In DepthDetails
TargetType-1/Type-2 angiotensin II receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50213457(CHEMBL84686)
Affinity DataIC50:  17nMAssay Description:In vitro displacement of [125I]angiotensin II from angiotensin 2 receptor on rabbit uterus membrane preparationMore data for this Ligand-Target Pair
In DepthDetails
TargetType-1/Type-2 angiotensin II receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50213551(CHEMBL90618)
Affinity DataIC50:  20nMAssay Description:In vitro displacement of [125I]angiotensin II from angiotensin 2 receptor on rabbit uterus membrane preparationMore data for this Ligand-Target Pair
In DepthDetails
TargetType-1/Type-2 angiotensin II receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50213461(CHEMBL407824)
Affinity DataIC50:  23nMAssay Description:In vitro displacement of [125I]angiotensin II from angiotensin 2 receptor on rabbit uterus membrane preparationMore data for this Ligand-Target Pair
In DepthDetails
TargetType-1/Type-2 angiotensin II receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50213552(CHEMBL328302)
Affinity DataIC50:  28nMAssay Description:In vitro displacement of [125I]angiotensin II from angiotensin 2 receptor on rabbit uterus membrane preparationMore data for this Ligand-Target Pair
In DepthDetails
TargetType-1/Type-2 angiotensin II receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50213568(CHEMBL87108)
Affinity DataIC50:  42nMAssay Description:In vitro displacement of [125I]angiotensin II from angiotensin 2 receptor on rabbit uterus membrane preparationMore data for this Ligand-Target Pair
In DepthDetails
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