Compile Data Set for Download or QSAR
maximum 50k data
Found 23 Enz. Inhib. hit(s) with all data for entry = 50031472
TargetTGF-beta receptor type-1(Homo sapiens (Human))
Northeastern Ohio Universities Colleges Of Medicine And Pharmacy

Curated by ChEMBL
LigandPNGBDBM50214864(3-((5-(6-methylpyridin-2-yl)-4-(quinoxalin-6-yl)-1...)
Affinity DataIC50:  10nMAssay Description:Antagonistic activity at TGFBR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTGF-beta receptor type-1(Homo sapiens (Human))
Northeastern Ohio Universities Colleges Of Medicine And Pharmacy

Curated by ChEMBL
LigandPNGBDBM50214857(3-((5-(6-methylpyridin-2-yl)-4-(quinoxalin-6-yl)-1...)
Affinity DataIC50:  12nMAssay Description:Antagonistic activity at TGFBR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTGF-beta receptor type-1(Homo sapiens (Human))
Northeastern Ohio Universities Colleges Of Medicine And Pharmacy

Curated by ChEMBL
LigandPNGBDBM50214853(3-((5-(6-ethylpyridin-2-yl)-4-(quinoxalin-6-yl)-1H...)
Affinity DataIC50:  15nMAssay Description:Antagonistic activity at TGFBR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTGF-beta receptor type-1(Homo sapiens (Human))
Northeastern Ohio Universities Colleges Of Medicine And Pharmacy

Curated by ChEMBL
LigandPNGBDBM50214868(3-((4-(benzo[d][1,3]dioxol-5-yl)-5-(6-methylpyridi...)
Affinity DataIC50:  21nMAssay Description:Antagonistic activity at TGFBR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTGF-beta receptor type-1(Homo sapiens (Human))
Northeastern Ohio Universities Colleges Of Medicine And Pharmacy

Curated by ChEMBL
LigandPNGBDBM50214866(3-((4-(benzo[d][1,3]dioxol-5-yl)-5-(6-methylpyridi...)
Affinity DataIC50:  24nMAssay Description:Antagonistic activity at TGFBR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTGF-beta receptor type-1(Homo sapiens (Human))
Northeastern Ohio Universities Colleges Of Medicine And Pharmacy

Curated by ChEMBL
LigandPNGBDBM50214859(4-((5-(6-methylpyridin-2-yl)-4-(quinoxalin-6-yl)-1...)
Affinity DataIC50:  42nMAssay Description:Antagonistic activity at TGFBR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTGF-beta receptor type-1(Homo sapiens (Human))
Northeastern Ohio Universities Colleges Of Medicine And Pharmacy

Curated by ChEMBL
LigandPNGBDBM50214862(3-((4-(benzo[d][1,3]dioxol-5-yl)-5-(6-ethylpyridin...)
Affinity DataIC50:  46nMAssay Description:Antagonistic activity at TGFBR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTGF-beta receptor type-1(Homo sapiens (Human))
Northeastern Ohio Universities Colleges Of Medicine And Pharmacy

Curated by ChEMBL
LigandPNGBDBM50214861(3-((4-(benzo[d][1,3]dioxol-5-yl)-5-(6-methylpyridi...)
Affinity DataIC50:  46nMAssay Description:Antagonistic activity at TGFBR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTGF-beta receptor type-1(Homo sapiens (Human))
Northeastern Ohio Universities Colleges Of Medicine And Pharmacy

Curated by ChEMBL
LigandPNGBDBM50214856(4-((5-(6-ethylpyridin-2-yl)-4-(quinoxalin-6-yl)-1H...)
Affinity DataIC50:  47nMAssay Description:Antagonistic activity at TGFBR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTGF-beta receptor type-1(Homo sapiens (Human))
Northeastern Ohio Universities Colleges Of Medicine And Pharmacy

Curated by ChEMBL
LigandPNGBDBM50214863(3-((4-(benzo[d][1,3]dioxol-5-yl)-5-(6-ethylpyridin...)
Affinity DataIC50:  73nMAssay Description:Antagonistic activity at TGFBR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTGF-beta receptor type-1(Homo sapiens (Human))
Northeastern Ohio Universities Colleges Of Medicine And Pharmacy

Curated by ChEMBL
LigandPNGBDBM50214865(4-((5-(6-methylpyridin-2-yl)-4-(quinoxalin-6-yl)-1...)
Affinity DataIC50:  75nMAssay Description:Antagonistic activity at TGFBR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTGF-beta receptor type-1(Homo sapiens (Human))
Northeastern Ohio Universities Colleges Of Medicine And Pharmacy

Curated by ChEMBL
LigandPNGBDBM50214867(4-((5-(6-ethylpyridin-2-yl)-4-(quinoxalin-6-yl)-1H...)
Affinity DataIC50:  92nMAssay Description:Antagonistic activity at TGFBR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTGF-beta receptor type-1(Homo sapiens (Human))
Northeastern Ohio Universities Colleges Of Medicine And Pharmacy

Curated by ChEMBL
LigandPNGBDBM50110208(4-(4-(benzo[d][1,3]dioxol-5-yl)-5-(pyridin-2-yl)-1...)
Affinity DataIC50:  94nMAssay Description:Antagonistic activity at TGFBR1More data for this Ligand-Target Pair
TargetTGF-beta receptor type-1(Homo sapiens (Human))
Northeastern Ohio Universities Colleges Of Medicine And Pharmacy

Curated by ChEMBL
LigandPNGBDBM50214854(3-((5-(6-ethylpyridin-2-yl)-4-(quinoxalin-6-yl)-1H...)
Affinity DataIC50:  119nMAssay Description:Antagonistic activity at TGFBR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTGF-beta receptor type-1(Homo sapiens (Human))
Northeastern Ohio Universities Colleges Of Medicine And Pharmacy

Curated by ChEMBL
LigandPNGBDBM50214858(4-((4-(benzo[d][1,3]dioxol-5-yl)-5-(6-methylpyridi...)
Affinity DataIC50:  153nMAssay Description:Antagonistic activity at TGFBR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTGF-beta receptor type-1(Homo sapiens (Human))
Northeastern Ohio Universities Colleges Of Medicine And Pharmacy

Curated by ChEMBL
LigandPNGBDBM50110205(4-(4-(benzo[d][1,3]dioxol-5-yl)-5-(pyridin-2-yl)-1...)
Affinity DataIC50:  170nMAssay Description:Antagonistic activity at TGFBR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTGF-beta receptor type-1(Homo sapiens (Human))
Northeastern Ohio Universities Colleges Of Medicine And Pharmacy

Curated by ChEMBL
LigandPNGBDBM50214860(4-((4-(benzo[d][1,3]dioxol-5-yl)-5-(6-methylpyridi...)
Affinity DataIC50:  171nMAssay Description:Antagonistic activity at TGFBR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTGF-beta receptor type-1(Homo sapiens (Human))
Northeastern Ohio Universities Colleges Of Medicine And Pharmacy

Curated by ChEMBL
LigandPNGBDBM50110202((4-(4-(benzo[d][1,3]dioxol-5-yl)-5-(pyridin-2-yl)-...)
Affinity DataIC50:  260nMAssay Description:Antagonistic activity at TGFBR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTGF-beta receptor type-1(Homo sapiens (Human))
Northeastern Ohio Universities Colleges Of Medicine And Pharmacy

Curated by ChEMBL
LigandPNGBDBM50214869(4-((4-(benzo[d][1,3]dioxol-5-yl)-5-(6-methylpyridi...)
Affinity DataIC50:  262nMAssay Description:Antagonistic activity at TGFBR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTGF-beta receptor type-1(Homo sapiens (Human))
Northeastern Ohio Universities Colleges Of Medicine And Pharmacy

Curated by ChEMBL
LigandPNGBDBM50214855(4-((4-(benzo[d][1,3]dioxol-5-yl)-5-(6-ethylpyridin...)
Affinity DataIC50:  360nMAssay Description:Antagonistic activity at TGFBR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTGF-beta receptor type-1(Homo sapiens (Human))
Northeastern Ohio Universities Colleges Of Medicine And Pharmacy

Curated by ChEMBL
LigandPNGBDBM50214852(4-((4-(benzo[d][1,3]dioxol-5-yl)-5-(6-ethylpyridin...)
Affinity DataIC50:  385nMAssay Description:Antagonistic activity at TGFBR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTGF-beta receptor type-1(Homo sapiens (Human))
Northeastern Ohio Universities Colleges Of Medicine And Pharmacy

Curated by ChEMBL
LigandPNGBDBM50110199(4-(4-(4-fluorophenyl)-5-(pyridin-2-yl)-1H-imidazol...)
Affinity DataIC50:  1.50E+3nMAssay Description:Antagonistic activity at TGFBR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTGF-beta receptor type-1(Homo sapiens (Human))
Northeastern Ohio Universities Colleges Of Medicine And Pharmacy

Curated by ChEMBL
LigandPNGBDBM50110197(4-(4-(benzo[d][1,3]dioxol-5-yl)-5-(pyridin-2-yl)-1...)
Affinity DataIC50:  2.95E+3nMAssay Description:Antagonistic activity at TGFBR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed