Compile Data Set for Download or QSAR
maximum 50k data
Found 28 Enz. Inhib. hit(s) with all data for entry = 50032020
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50323394(5-(2,3,5-trifluorophenyl)-1,4,5,6-tetrahydrocyclop...)
Affinity DataIC50:  20nMAssay Description:Displacement of [3H]nicotinic acid from human GPR10a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Mus musculus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50323394(5-(2,3,5-trifluorophenyl)-1,4,5,6-tetrahydrocyclop...)
Affinity DataIC50:  30nMAssay Description:Displacement of [3H]nicotinic acid from mouse GPR10a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Mus musculus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50277789(3-(1H-tetrazol-5-yl)-5-(2,3,5-trifluorophenyl)-1,4...)
Affinity DataIC50:  70nMAssay Description:Displacement of [3H]nicotinic acid from mouse GPR10a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Mus musculus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50323396(5-(thiophen-3-yl)-1,4,5,6-tetrahydrocyclopenta[c]p...)
Affinity DataIC50:  80nMAssay Description:Displacement of [3H]nicotinic acid from mouse GPR10a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50277789(3-(1H-tetrazol-5-yl)-5-(2,3,5-trifluorophenyl)-1,4...)
Affinity DataIC50:  80nMAssay Description:Displacement of [3H]nicotinic acid from human GPR10a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50323396(5-(thiophen-3-yl)-1,4,5,6-tetrahydrocyclopenta[c]p...)
Affinity DataIC50:  90nMAssay Description:Displacement of [3H]nicotinic acid from human GPR10a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Mus musculus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM23515(CHEMBL573 | Niacin | Nicotinic Acid | [5, 6-3H]-ni...)
Affinity DataIC50:  140nMAssay Description:Displacement of [3H]nicotinic acid from mouse GPR10a receptorMore data for this Ligand-Target Pair
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM23515(CHEMBL573 | Niacin | Nicotinic Acid | [5, 6-3H]-ni...)
Affinity DataIC50:  140nMAssay Description:Displacement of [3H]nicotinic acid from human GPR10a receptorMore data for this Ligand-Target Pair
TargetHydroxycarboxylic acid receptor 2(Mus musculus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50323393(5-phenyl-1,4,5,6-tetrahydrocyclopenta[c]pyrazole-3...)
Affinity DataIC50:  150nMAssay Description:Displacement of [3H]nicotinic acid from mouse GPR10a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50323393(5-phenyl-1,4,5,6-tetrahydrocyclopenta[c]pyrazole-3...)
Affinity DataIC50:  200nMAssay Description:Displacement of [3H]nicotinic acid from human GPR10a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50323395(5-(thiophen-2-yl)-1,4,5,6-tetrahydrocyclopenta[c]p...)
Affinity DataIC50:  240nMAssay Description:Displacement of [3H]nicotinic acid from human GPR10a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Mus musculus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50323390(5-propyl-1,4,5,6-tetrahydrocyclopenta[c]pyrazole-3...)
Affinity DataIC50:  250nMAssay Description:Displacement of [3H]nicotinic acid from mouse GPR10a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Mus musculus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50323395(5-(thiophen-2-yl)-1,4,5,6-tetrahydrocyclopenta[c]p...)
Affinity DataIC50:  250nMAssay Description:Displacement of [3H]nicotinic acid from mouse GPR10a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50323390(5-propyl-1,4,5,6-tetrahydrocyclopenta[c]pyrazole-3...)
Affinity DataIC50:  380nMAssay Description:Displacement of [3H]nicotinic acid from human GPR10a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50323398(5-(1-methyl-1H-pyrazol-5-yl)-1,4,5,6-tetrahydrocyc...)
Affinity DataIC50:  390nMAssay Description:Displacement of [3H]nicotinic acid from human GPR10a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Mus musculus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50323398(5-(1-methyl-1H-pyrazol-5-yl)-1,4,5,6-tetrahydrocyc...)
Affinity DataIC50:  450nMAssay Description:Displacement of [3H]nicotinic acid from mouse GPR10a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Mus musculus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50323391(5-isopropyl-1,4,5,6-tetrahydrocyclopenta[c]pyrazol...)
Affinity DataIC50:  990nMAssay Description:Displacement of [3H]nicotinic acid from mouse GPR10a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Mus musculus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50323392(5-sec-butyl-1,4,5,6-tetrahydrocyclopenta[c]pyrazol...)
Affinity DataIC50:  1.10E+3nMAssay Description:Displacement of [3H]nicotinic acid from mouse GPR10a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Mus musculus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50273099(3-(1H-tetrazol-5-yl)-1,4,5,6-tetrahydrocyclopenta[...)
Affinity DataIC50:  1.20E+3nMAssay Description:Displacement of [3H]nicotinic acid from mouse GPR10a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50323392(5-sec-butyl-1,4,5,6-tetrahydrocyclopenta[c]pyrazol...)
Affinity DataIC50:  1.30E+3nMAssay Description:Displacement of [3H]nicotinic acid from human GPR10a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50273099(3-(1H-tetrazol-5-yl)-1,4,5,6-tetrahydrocyclopenta[...)
Affinity DataIC50:  1.50E+3nMAssay Description:Displacement of [3H]nicotinic acid from human GPR10a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Mus musculus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50323397(5-(1-methyl-1H-pyrazol-4-yl)-1,4,5,6-tetrahydrocyc...)
Affinity DataIC50:  1.60E+3nMAssay Description:Displacement of [3H]nicotinic acid from mouse GPR10a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50323391(5-isopropyl-1,4,5,6-tetrahydrocyclopenta[c]pyrazol...)
Affinity DataIC50:  1.70E+3nMAssay Description:Displacement of [3H]nicotinic acid from human GPR10a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50323399(5-(1H-pyrazol-1-yl)-1,4,5,6-tetrahydrocyclopenta[c...)
Affinity DataIC50:  1.90E+3nMAssay Description:Displacement of [3H]nicotinic acid from human GPR10a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50323397(5-(1-methyl-1H-pyrazol-4-yl)-1,4,5,6-tetrahydrocyc...)
Affinity DataIC50:  2.10E+3nMAssay Description:Displacement of [3H]nicotinic acid from human GPR10a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Mus musculus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50323399(5-(1H-pyrazol-1-yl)-1,4,5,6-tetrahydrocyclopenta[c...)
Affinity DataIC50:  3.40E+3nMAssay Description:Displacement of [3H]nicotinic acid from mouse GPR10a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50323400(5-(1H-1,2,3-triazol-1-yl)-1,4,5,6-tetrahydrocyclop...)
Affinity DataIC50:  4.00E+3nMAssay Description:Displacement of [3H]nicotinic acid from human GPR10a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Mus musculus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50323400(5-(1H-1,2,3-triazol-1-yl)-1,4,5,6-tetrahydrocyclop...)
Affinity DataIC50:  5.20E+3nMAssay Description:Displacement of [3H]nicotinic acid from mouse GPR10a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed