Affinity DataKi: 1.40nMAssay Description:Inhibition of [3H]DSLET binding to delta 1 opioid receptors in rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 2.20nMAssay Description:Inhibition of [3H]DSLET binding to delta 1 opioid receptors in rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 2.20nMAssay Description:Inhibition of [3H]DAGO binding to mu 1 opioid receptor in rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 2.70nMAssay Description:Inhibition of [3H]DSLET binding to delta 1 opioid receptors in rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 3.90nMAssay Description:Inhibition of [3H]DAGO binding to mu 1 opioid receptor in rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 4.20nMAssay Description:Inhibition of [3H]DSLET binding to delta 1 opioid receptors in rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 4.80nMAssay Description:Inhibition of [3H]DSLET binding to delta 1 opioid receptors in rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 5.60nMAssay Description:Inhibition of [3H]DSLET binding to delta 1 opioid receptors in rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 7.30nMAssay Description:Inhibition of [3H]DSLET binding to delta 1 opioid receptors in rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 7.60nMAssay Description:Inhibition of [3H]DSLET binding to delta 1 opioid receptors in rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 7.70nMAssay Description:Inhibition of [3H]DSLET binding to delta 1 opioid receptors in rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 8.40nMAssay Description:Ability to inhibit the binding of [3H]-DAGO to Opioid receptor mu 1 in rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 9.10nMAssay Description:Inhibition of [3H]DSLET binding to delta 1 opioid receptors in rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 9.20nMAssay Description:Inhibition of [3H]DAGO binding to mu 1 opioid receptor in rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Inhibition of [3H]DAGO binding to mu 1 opioid receptor in rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:Inhibition of [3H]DSLET binding to delta 1 opioid receptors in rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 14nMAssay Description:Inhibition of [3H]DAGO binding to mu 1 opioid receptor in rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 15nMAssay Description:Inhibition of [3H]DAGO binding to mu 1 opioid receptor in rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 16nMAssay Description:Inhibition of [3H]DAGO binding to mu 1 opioid receptor in rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 17nMAssay Description:Inhibition of [3H]DAGO binding to mu 1 opioid receptor in rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 25nMAssay Description:Inhibition of [3H]DAGO binding to mu 1 opioid receptor in rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 28nMAssay Description:Inhibition of [3H]DAGO binding to mu 1 opioid receptor in rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 30nMAssay Description:Inhibition of [3H]DSLET binding to delta 1 opioid receptors in rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 31nMAssay Description:Inhibition of [3H]DAGO binding to mu 1 opioid receptor in rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 31nMAssay Description:Inhibition of [3H]DSLET binding to delta 1 opioid receptors in rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 36nMAssay Description:Inhibition of [3H]DAGO binding to mu 1 opioid receptor in rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 38nMAssay Description:Inhibition of [3H]DAGO binding to mu 1 opioid receptor in rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 39nMAssay Description:Inhibition of [3H]DSLET binding to delta 1 opioid receptors in rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 42nMAssay Description:Inhibition of [3H]DAGO binding to mu 1 opioid receptor in rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 43nMAssay Description:Inhibition of [3H]DAGO binding to mu 1 opioid receptor in rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 43nMAssay Description:Inhibition of [3H]DSLET binding to delta 1 opioid receptors in rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 44nMAssay Description:Inhibition of [3H]DAGO binding to mu 1 opioid receptor in rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 61nMAssay Description:Inhibition of [3H]DAGO binding to mu 1 opioid receptor in rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 116nMAssay Description:Inhibition of [3H]DAGO binding to mu 1 opioid receptor in rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 157nMAssay Description:Inhibition of [3H]DAGO binding to mu 1 opioid receptor in rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 158nMAssay Description:Inhibition of [3H]DAGO binding to mu 1 opioid receptor in rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 171nMAssay Description:Inhibition of [3H]DAGO binding to mu 1 opioid receptor in rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 280nMAssay Description:Inhibition of [3H]DSLET binding to delta 1 opioid receptors in rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 395nMAssay Description:Inhibition of [3H]DSLET binding to delta 1 opioid receptors in rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 480nMAssay Description:Inhibition of [3H]DSLET binding to delta 1 opioid receptors in rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 600nMAssay Description:Inhibition of [3H]DSLET binding to delta 1 opioid receptors in rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 700nMAssay Description:Ability to inhibit the binding of [3H]DSLET to Opioid receptor delta 1 in rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 873nMAssay Description:Inhibition of [3H]DAGO binding to mu 1 opioid receptor in rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 1.02E+3nMAssay Description:Inhibition of [3H]DSLET binding to delta 1 opioid receptors in rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 3.45E+3nMAssay Description:Inhibition of [3H]DSLET binding to delta 1 opioid receptors in rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 3.81E+3nMAssay Description:Inhibition of [3H]DSLET binding to delta 1 opioid receptors in rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 6.88E+3nMAssay Description:Inhibition of [3H]DSLET binding to delta 1 opioid receptors in rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 9.79E+3nMAssay Description:Inhibition of [3H]DAGO binding to mu 1 opioid receptor in rat brain membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 12nMAssay Description:Inhibition of electrically evoked contraction of guinea pig ileum (myenteric plexus:longitudinal muscle preparation) by antagonist action at mu 1 opi...More data for this Ligand-Target Pair
Affinity DataIC50: 21nMAssay Description:Inhibition of electrically evoked contraction of guinea pig ileum (myenteric plexus:longitudinal muscle preparation) by antagonist action at mu 1 opi...More data for this Ligand-Target Pair