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Found 124 Enz. Inhib. hit(s) with all data for entry = 50004968
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))TBA
LigandPNGBDBM50118703(CHEMBL109783 | N-[5-(4,5-Dihydro-1H-imidazol-2-yl)...)
Affinity DataKi:  12nMAssay Description:Binding affinity to alpha1A adrenoreceptor in Rattus norvegicus (rat) submaxillary gland by radioligand displacement assayMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))TBA
LigandPNGBDBM50474660(CHEMBL111771)
Affinity DataKi:  22nMAssay Description:Binding affinity to alpha1A adrenoreceptor in Rattus norvegicus (rat) submaxillary gland by radioligand displacement assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50118703(CHEMBL109783 | N-[5-(4,5-Dihydro-1H-imidazol-2-yl)...)
Affinity DataKi:  33nMAssay Description:Binding affinity to Homo sapiens (human) alpha2A receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))TBA
LigandPNGBDBM50474630(CHEMBL108804)
Affinity DataKi:  36nMAssay Description:Binding affinity to alpha1A adrenoreceptor in Rattus norvegicus (rat) submaxillary gland by radioligand displacement assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))TBA
LigandPNGBDBM50487266(CHEMBL2261355)
Affinity DataKi:  47nMAssay Description:Binding affinity to alpha1A adrenoreceptor in Rattus norvegicus (rat) submaxillary gland by radioligand displacement assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))TBA
LigandPNGBDBM50487270(CHEMBL2261347)
Affinity DataKi:  60nMAssay Description:Binding affinity to alpha1A adrenoreceptor in Rattus norvegicus (rat) submaxillary gland by radioligand displacement assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))TBA
LigandPNGBDBM50474635(CHEMBL109827)
Affinity DataKi:  91nMAssay Description:Binding affinity to alpha1A adrenoreceptor in Rattus norvegicus (rat) submaxillary gland by radioligand displacement assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))TBA
LigandPNGBDBM50474633(CHEMBL111496)
Affinity DataKi:  95nMAssay Description:Binding affinity to alpha1A adrenoreceptor in Rattus norvegicus (rat) submaxillary gland by radioligand displacement assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))TBA
LigandPNGBDBM50474654(CHEMBL323402)
Affinity DataKi:  126nMAssay Description:Binding affinity to alpha1A adrenoreceptor in Rattus norvegicus (rat) submaxillary gland by radioligand displacement assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))TBA
LigandPNGBDBM50474643(CHEMBL111734)
Affinity DataKi:  129nMAssay Description:Binding affinity to alpha1A adrenoreceptor in Rattus norvegicus (rat) submaxillary gland by radioligand displacement assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))TBA
LigandPNGBDBM50118705(ABT-866 | CHEMBL326702 | Ethanesulfonic acid [3-(1...)
Affinity DataKi:  135nMAssay Description:Binding affinity to alpha1A adrenoreceptor in Rattus norvegicus (rat) submaxillary gland by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails Article
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50118705(ABT-866 | CHEMBL326702 | Ethanesulfonic acid [3-(1...)
Affinity DataKi:  170nMAssay Description:Binding affinity to Homo sapiens (human) alpha2A receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetAlpha-1D adrenergic receptor(Rattus norvegicus (Rat))TBA
LigandPNGBDBM50474654(CHEMBL323402)
Affinity DataKi:  191nMAssay Description:Binding affinity to Rattus norvegicus (rat) alpha1D adrenoreceptor by radioligand displacement assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))TBA
LigandPNGBDBM50474671(CHEMBL111554)
Affinity DataKi:  195nMAssay Description:Binding affinity to alpha1A adrenoreceptor in Rattus norvegicus (rat) submaxillary gland by radioligand displacement assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
TargetAlpha-2B adrenergic receptor(NEONATAL RAT)TBA
LigandPNGBDBM50118703(CHEMBL109783 | N-[5-(4,5-Dihydro-1H-imidazol-2-yl)...)
Affinity DataKi:  245nMAssay Description:Binding affinity to Rattus norvegicus (rat) alpha2B receptor isolated from neonatal lungMore data for this Ligand-Target Pair
In DepthDetails Article
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))TBA
LigandPNGBDBM50474666(CHEMBL321644)
Affinity DataKi:  251nMAssay Description:Binding affinity to alpha1A adrenoreceptor in Rattus norvegicus (rat) submaxillary gland by radioligand displacement assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
TargetAlpha-1D adrenergic receptor(Rattus norvegicus (Rat))TBA
LigandPNGBDBM50118705(ABT-866 | CHEMBL326702 | Ethanesulfonic acid [3-(1...)
Affinity DataKi:  275nMAssay Description:Binding affinity to Rattus norvegicus (rat) alpha1D adrenoreceptor by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails Article
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))TBA
LigandPNGBDBM50474670(CHEMBL111584)
Affinity DataKi:  275nMAssay Description:Binding affinity to alpha1A adrenoreceptor in Rattus norvegicus (rat) submaxillary gland by radioligand displacement assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))TBA
LigandPNGBDBM50487271(CHEMBL2261351)
Affinity DataKi:  288nMAssay Description:Binding affinity to alpha1A adrenoreceptor in Rattus norvegicus (rat) submaxillary gland by radioligand displacement assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))TBA
LigandPNGBDBM50474653(CHEMBL109755)
Affinity DataKi:  457nMAssay Description:Binding affinity to alpha1A adrenoreceptor in Rattus norvegicus (rat) submaxillary gland by radioligand displacement assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
LigandPNGBDBM50474654(CHEMBL323402)
Affinity DataKi:  525nMAssay Description:Binding affinity to Cricetinae (hamster) alpha1B adrenoreceptor by radioligand displacement assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))TBA
LigandPNGBDBM50474648(CHEMBL109848)
Affinity DataKi:  525nMAssay Description:Binding affinity to alpha1A adrenoreceptor in Rattus norvegicus (rat) submaxillary gland by radioligand displacement assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))TBA
LigandPNGBDBM50474652(CHEMBL325897)
Affinity DataKi:  537nMAssay Description:Binding affinity to alpha1A adrenoreceptor in Rattus norvegicus (rat) submaxillary gland by radioligand displacement assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))TBA
LigandPNGBDBM50487268(CHEMBL2261353)
Affinity DataKi:  617nMAssay Description:Binding affinity to alpha1A adrenoreceptor in Rattus norvegicus (rat) submaxillary gland by radioligand displacement assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))TBA
LigandPNGBDBM50487263(CHEMBL2261348)
Affinity DataKi:  776nMAssay Description:Binding affinity to alpha1A adrenoreceptor in Rattus norvegicus (rat) submaxillary gland by radioligand displacement assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))TBA
LigandPNGBDBM50474661(CHEMBL320765)
Affinity DataKi:  794nMAssay Description:Binding affinity to alpha1A adrenoreceptor in Rattus norvegicus (rat) submaxillary gland by radioligand displacement assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
LigandPNGBDBM50118705(ABT-866 | CHEMBL326702 | Ethanesulfonic acid [3-(1...)
Affinity DataKi:  891nMAssay Description:Binding affinity to Cricetinae (hamster) alpha1B adrenoreceptor by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails Article
TargetAlpha-2B adrenergic receptor(NEONATAL RAT)TBA
LigandPNGBDBM50118705(ABT-866 | CHEMBL326702 | Ethanesulfonic acid [3-(1...)
Affinity DataKi:  977nMAssay Description:Binding affinity to Rattus norvegicus (rat) alpha2B receptor isolated from neonatal lungMore data for this Ligand-Target Pair
In DepthDetails Article
TargetAlpha-1D adrenergic receptor(Rattus norvegicus (Rat))TBA
LigandPNGBDBM50474660(CHEMBL111771)
Affinity DataKi:  977nMAssay Description:Binding affinity to Rattus norvegicus (rat) alpha1D adrenoreceptor by radioligand displacement assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
TargetAlpha-1D adrenergic receptor(Rattus norvegicus (Rat))TBA
LigandPNGBDBM50474643(CHEMBL111734)
Affinity DataKi:  1.00E+3nMAssay Description:Binding affinity to Rattus norvegicus (rat) alpha1D adrenoreceptor by radioligand displacement assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
LigandPNGBDBM50474670(CHEMBL111584)
Affinity DataKi:  1.05E+3nMAssay Description:Binding affinity to Cricetinae (hamster) alpha1B adrenoreceptor by radioligand displacement assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
TargetAlpha-1D adrenergic receptor(Rattus norvegicus (Rat))TBA
LigandPNGBDBM50487266(CHEMBL2261355)
Affinity DataKi:  1.07E+3nMAssay Description:Binding affinity to Rattus norvegicus (rat) alpha1D adrenoreceptor by radioligand displacement assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))TBA
LigandPNGBDBM50474650(CHEMBL111537)
Affinity DataKi:  1.15E+3nMAssay Description:Binding affinity to alpha1A adrenoreceptor in Rattus norvegicus (rat) submaxillary gland by radioligand displacement assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
TargetAlpha-1D adrenergic receptor(Rattus norvegicus (Rat))TBA
LigandPNGBDBM50474630(CHEMBL108804)
Affinity DataKi:  1.26E+3nMAssay Description:Binding affinity to Rattus norvegicus (rat) alpha1D adrenoreceptor by radioligand displacement assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
LigandPNGBDBM50487266(CHEMBL2261355)
Affinity DataKi:  1.32E+3nMAssay Description:Binding affinity to Cricetinae (hamster) alpha1B adrenoreceptor by radioligand displacement assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))TBA
LigandPNGBDBM50474634(CHEMBL322492)
Affinity DataKi:  1.35E+3nMAssay Description:Binding affinity to alpha1A adrenoreceptor in Rattus norvegicus (rat) submaxillary gland by radioligand displacement assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
TargetAlpha-1D adrenergic receptor(Rattus norvegicus (Rat))TBA
LigandPNGBDBM50118703(CHEMBL109783 | N-[5-(4,5-Dihydro-1H-imidazol-2-yl)...)
Affinity DataKi:  1.48E+3nMAssay Description:Binding affinity to Rattus norvegicus (rat) alpha1D adrenoreceptor by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails Article
TargetAlpha-1D adrenergic receptor(Rattus norvegicus (Rat))TBA
LigandPNGBDBM50487268(CHEMBL2261353)
Affinity DataKi:  1.55E+3nMAssay Description:Binding affinity to Rattus norvegicus (rat) alpha1D adrenoreceptor by radioligand displacement assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
TargetAlpha-1D adrenergic receptor(Rattus norvegicus (Rat))TBA
LigandPNGBDBM50474671(CHEMBL111554)
Affinity DataKi:  1.59E+3nMAssay Description:Binding affinity to Rattus norvegicus (rat) alpha1D adrenoreceptor by radioligand displacement assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
TargetAlpha-1D adrenergic receptor(Rattus norvegicus (Rat))TBA
LigandPNGBDBM50474633(CHEMBL111496)
Affinity DataKi:  1.66E+3nMAssay Description:Binding affinity to Rattus norvegicus (rat) alpha1D adrenoreceptor by radioligand displacement assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
TargetAlpha-1D adrenergic receptor(Rattus norvegicus (Rat))TBA
LigandPNGBDBM50118702(2-Amino-1-(2,5-dimethoxy-phenyl)-ethanol | CHEMBL1...)
Affinity DataKi:  1.66E+3nMAssay Description:Binding affinity to Rattus norvegicus (rat) alpha1D adrenoreceptor by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails Article
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))TBA
LigandPNGBDBM50474647(CHEMBL111391)
Affinity DataKi:  1.70E+3nMAssay Description:Binding affinity to alpha1A adrenoreceptor in Rattus norvegicus (rat) submaxillary gland by radioligand displacement assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
TargetAlpha-1D adrenergic receptor(Rattus norvegicus (Rat))TBA
LigandPNGBDBM50487263(CHEMBL2261348)
Affinity DataKi:  1.86E+3nMAssay Description:Binding affinity to Rattus norvegicus (rat) alpha1D adrenoreceptor by radioligand displacement assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
LigandPNGBDBM50474660(CHEMBL111771)
Affinity DataKi:  2.00E+3nMAssay Description:Binding affinity to Cricetinae (hamster) alpha1B adrenoreceptor by radioligand displacement assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))TBA
LigandPNGBDBM50118702(2-Amino-1-(2,5-dimethoxy-phenyl)-ethanol | CHEMBL1...)
Affinity DataKi:  2.00E+3nMAssay Description:Binding affinity to alpha1A adrenoreceptor in Rattus norvegicus (rat) submaxillary gland by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails Article
TargetAlpha-1D adrenergic receptor(Rattus norvegicus (Rat))TBA
LigandPNGBDBM50474650(CHEMBL111537)
Affinity DataKi:  2.04E+3nMAssay Description:Binding affinity to Rattus norvegicus (rat) alpha1D adrenoreceptor by radioligand displacement assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
TargetAlpha-1D adrenergic receptor(Rattus norvegicus (Rat))TBA
LigandPNGBDBM50487270(CHEMBL2261347)
Affinity DataKi:  2.19E+3nMAssay Description:Binding affinity to Rattus norvegicus (rat) alpha1D adrenoreceptor by radioligand displacement assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
LigandPNGBDBM50474630(CHEMBL108804)
Affinity DataKi:  2.51E+3nMAssay Description:Binding affinity to Cricetinae (hamster) alpha1B adrenoreceptor by radioligand displacement assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
TargetAlpha-1D adrenergic receptor(Rattus norvegicus (Rat))TBA
LigandPNGBDBM50474634(CHEMBL322492)
Affinity DataKi:  2.51E+3nMAssay Description:Binding affinity to Rattus norvegicus (rat) alpha1D adrenoreceptor by radioligand displacement assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
TargetAlpha-1D adrenergic receptor(Rattus norvegicus (Rat))TBA
LigandPNGBDBM50474652(CHEMBL325897)
Affinity DataKi:  2.69E+3nMAssay Description:Binding affinity to Rattus norvegicus (rat) alpha1D adrenoreceptor by radioligand displacement assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
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