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Found 37 Enz. Inhib. hit(s) with all data for entry = 50005215
TargetDipeptidyl peptidase 4(Homo sapiens (Human))TBA
LigandPNGBDBM50489030(CHEMBL1230804)
Affinity DataKi:  0.820nMAssay Description:Inhibition of dipeptidyl peptidase 4 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetDipeptidyl peptidase 4(Homo sapiens (Human))TBA
LigandPNGBDBM50324517((6-(aminomethyl)-5-(2,4-dichlorophenyl)-7-methylim...)
Affinity DataKi:  2.20nMAssay Description:Inhibition of dipeptidyl peptidase 4 (unknown origin)More data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Homo sapiens (Human))TBA
LigandPNGBDBM15510((4R,5R)-5-amino-1-(2-(benzo[d][1,3]dioxol-5-yl)eth...)
Affinity DataKi:  3.20nMAssay Description:Inhibition of dipeptidyl peptidase 4 (unknown origin)More data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Homo sapiens (Human))TBA
LigandPNGBDBM15526(N-{[(3S,5S)-5-(1,3-thiazolidin-3-ylcarbonyl)pyrrol...)
Affinity DataKi:  3.40nMAssay Description:Inhibition of dipeptidyl peptidase 4 (unknown origin)More data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Homo sapiens (Human))TBA
LigandPNGBDBM50489031(CHEMBL1230826)
Affinity DataKi:  3.80nMAssay Description:Inhibition of dipeptidyl peptidase 4 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetDipeptidyl peptidase 4(Homo sapiens (Human))TBA
LigandPNGBDBM15518((3R,4R)-1-(6-(3-(methylsulfonyl)phenyl)pyrimidin-4...)
Affinity DataKi:  4nMAssay Description:Inhibition of dipeptidyl peptidase 4 (unknown origin)More data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Homo sapiens (Human))TBA
LigandPNGBDBM15498((3R,4S)-1-[6-(3-methanesulfonylphenyl)pyrimidin-4-...)
Affinity DataKi:  5.30nMAssay Description:Inhibition of dipeptidyl peptidase 4 (unknown origin)More data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Homo sapiens (Human))TBA
LigandPNGBDBM50489029(CHEMBL1230763)
Affinity DataKi:  6.70nMAssay Description:Inhibition of dipeptidyl peptidase 4 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetDipeptidyl peptidase 4(Homo sapiens (Human))TBA
LigandPNGBDBM11593(5-(aminomethyl)-6-(2,4-dichlorophenyl)-2-(3,5-dime...)
Affinity DataIC50:  0.100nMAssay Description:Inhibition of dipeptidyl peptidase 4 (unknown origin)More data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Homo sapiens (Human))TBA
LigandPNGBDBM50489026(CHEMBL1229820)
Affinity DataIC50:  0.5nMAssay Description:Inhibition of dipeptidyl peptidase 4 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetDipeptidyl peptidase 4(Homo sapiens (Human))TBA
LigandPNGBDBM50228403((R)-8-(3-aminopiperidin-1-yl)-7-(but-2-ynyl)-3-met...)
Affinity DataIC50:  1nMAssay Description:Inhibition of dipeptidyl peptidase 4 (unknown origin)More data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Homo sapiens (Human))TBA
LigandPNGBDBM50221979((2S,3S)-2-((1r,4S)-4-([1,2,4]triazolo[1,5-a]pyridi...)
Affinity DataIC50:  2.30nMAssay Description:Inhibition of dipeptidyl peptidase 4 (unknown origin)More data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Homo sapiens (Human))TBA
LigandPNGBDBM50221972((2S,3S)-2-(4-([1,2,4]triazolo[1,5-a]pyridin-6-yl)p...)
Affinity DataIC50:  4.30nMAssay Description:Inhibition of dipeptidyl peptidase 4 (unknown origin)More data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Homo sapiens (Human))TBA
LigandPNGBDBM50221968((2S,3S)-2-((1r,4S)-4-([1,2,4]triazolo[1,5-a]pyridi...)
Affinity DataIC50:  4.80nMAssay Description:Inhibition of dipeptidyl peptidase 4 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
TargetDipeptidyl peptidase 4(Homo sapiens (Human))TBA
LigandPNGBDBM50208877(2-amino-6-chloropurine | 6-Cl-purine (1) | 6-chlor...)
Affinity DataIC50:  5nMAssay Description:Inhibition of dipeptidyl peptidase 4 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
TargetDipeptidyl peptidase 4(Homo sapiens (Human))TBA
LigandPNGBDBM50309470((4S)-1-[(2S,3S,11bS)-2-amino-9,10-dimethoxy-1,3,4,...)
Affinity DataIC50:  6.80nMAssay Description:Inhibition of dipeptidyl peptidase 4 (unknown origin)More data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Homo sapiens (Human))TBA
LigandPNGBDBM50489028(CHEMBL1233461)
Affinity DataIC50:  7nMAssay Description:Inhibition of dipeptidyl peptidase 4 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
TargetDipeptidyl peptidase 4(Homo sapiens (Human))TBA
LigandPNGBDBM50375237(CHEMBL272114)
Affinity DataIC50:  8nMAssay Description:Inhibition of dipeptidyl peptidase 4 (unknown origin)More data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Homo sapiens (Human))TBA
LigandPNGBDBM50374938(CHEMBL402163)
Affinity DataIC50:  12nMAssay Description:Inhibition of dipeptidyl peptidase 4 (unknown origin)More data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Homo sapiens (Human))TBA
LigandPNGBDBM16272(2-({2-[(3R)-3-aminopiperidin-1-yl]-4-oxo-3,4-dihyd...)
Affinity DataIC50:  13nMAssay Description:Inhibition of dipeptidyl peptidase 4 (unknown origin)More data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Homo sapiens (Human))TBA
LigandPNGBDBM50249479(2-(4-{(3S,5S)-5-[(3,3-difluoropyrrolidin-1-yl)carb...)
Affinity DataIC50:  13nMAssay Description:Inhibition of dipeptidyl peptidase 4 (unknown origin)More data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Homo sapiens (Human))TBA
LigandPNGBDBM50489033(CHEMBL1229855)
Affinity DataIC50:  16nMAssay Description:Inhibition of dipeptidyl peptidase 4 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
TargetDipeptidyl peptidase 4(Homo sapiens (Human))TBA
LigandPNGBDBM50489024(CHEMBL1230015)
Affinity DataIC50:  19nMAssay Description:Inhibition of dipeptidyl peptidase 4 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetDipeptidyl peptidase 4(Homo sapiens (Human))TBA
LigandPNGBDBM50212927((1S,2R,5S)-5-(3-(trifluoromethyl)-5,6-dihydro-[1,2...)
Affinity DataIC50:  21nMAssay Description:Inhibition of dipeptidyl peptidase 4 (unknown origin)More data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Homo sapiens (Human))TBA
LigandPNGBDBM50489032(CHEMBL1229644)
Affinity DataIC50:  22nMAssay Description:Inhibition of dipeptidyl peptidase 4 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetDipeptidyl peptidase 4(Homo sapiens (Human))TBA
LigandPNGBDBM50489025(CHEMBL2298396)
Affinity DataIC50:  23nMAssay Description:Inhibition of dipeptidyl peptidase 4 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
TargetDipeptidyl peptidase 4(Homo sapiens (Human))TBA
LigandPNGBDBM50221443((2R)-4-[(8R)-8-METHYL-2-(TRIFLUOROMETHYL)-5,6-DIHY...)
Affinity DataIC50:  25nMAssay Description:Inhibition of dipeptidyl peptidase 4 (unknown origin)More data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Homo sapiens (Human))TBA
LigandPNGBDBM50244011(4'-[(1R)-1-amino-2-(2,5-difluorophenyl)ethyl]biphe...)
Affinity DataIC50:  32nMAssay Description:Inhibition of dipeptidyl peptidase 4 (unknown origin)More data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Homo sapiens (Human))TBA
LigandPNGBDBM50489022(CHEMBL1197118)
Affinity DataIC50:  42nMAssay Description:Inhibition of dipeptidyl peptidase 4 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetDipeptidyl peptidase 4(Homo sapiens (Human))TBA
LigandPNGBDBM50489023(CHEMBL1230044)
Affinity DataIC50:  65nMAssay Description:Inhibition of dipeptidyl peptidase 4 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetDipeptidyl peptidase 4(Homo sapiens (Human))TBA
LigandPNGBDBM50296490((7R,8R)-8-(2,4,5-Trifluoro-phenyl)-6,7,8,9-tetrahy...)
Affinity DataIC50:  67nMAssay Description:Inhibition of dipeptidyl peptidase 4 (unknown origin)More data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Homo sapiens (Human))TBA
LigandPNGBDBM50256266((2R)-4-(2-BENZOYL-1,2-DIAZEPAN-1-YL)-4-OXO-1-(2,4,...)
Affinity DataIC50:  70nMAssay Description:Inhibition of dipeptidyl peptidase 4 (unknown origin)More data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Homo sapiens (Human))TBA
LigandPNGBDBM15464(4-[(3R)-3-{[2-(4-fluorophenyl)-2-oxoethyl]amino}bu...)
Affinity DataIC50:  84nMAssay Description:Inhibition of dipeptidyl peptidase 4 (unknown origin)More data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Homo sapiens (Human))TBA
LigandPNGBDBM11559(N-({(2S)-1-[(3R)-3-amino-4-(2-fluorophenyl)butanoy...)
Affinity DataIC50:  90nMAssay Description:Inhibition of dipeptidyl peptidase 4 (unknown origin)More data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Homo sapiens (Human))TBA
LigandPNGBDBM50256569((R)-4-(4-(3-amino-4-(2,4,5-trifluorophenyl)butanoy...)
Affinity DataIC50:  223nMAssay Description:Inhibition of dipeptidyl peptidase 4 (unknown origin)More data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Homo sapiens (Human))TBA
LigandPNGBDBM50489027(CHEMBL1236897)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of dipeptidyl peptidase 4 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails Article
TargetDipeptidyl peptidase 4(Homo sapiens (Human))TBA
LigandPNGBDBM50375239(CHEMBL257036)
Affinity DataIC50:  3.00E+4nMAssay Description:Inhibition of dipeptidyl peptidase 4 (unknown origin)More data for this Ligand-Target Pair