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Found 5 Enz. Inhib. hit(s) with all data for assayid = 1 entry = 10819
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Inxmed (Nanjing)

US Patent
LigandPNGBDBM571388(US11440916, HZ10136)
Affinity DataIC50:  1.10nMAssay Description:The IC50 (nM) values of the example compound HZ10126 and several reference compounds against the rat A2A receptor were measured in an in vitro assay,...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Inxmed (Nanjing)

US Patent
LigandPNGBDBM50202993(2-furan-2-yl-7-[2-(4-phenyl-piperazin-1-yl)-ethyl]...)
Affinity DataIC50:  1.20nMAssay Description:The IC50 (nM) values of the example compound HZ10126 and several reference compounds against the rat A2A receptor were measured in an in vitro assay,...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Inxmed (Nanjing)

US Patent
LigandPNGBDBM50048466(2-(furan-2-yl)-7-phenethyl-7H-pyrazolo[4,3-e][1,2,...)
Affinity DataIC50:  1.80nMAssay Description:The IC50 (nM) values of the example compound HZ10126 and several reference compounds against the rat A2A receptor were measured in an in vitro assay,...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Inxmed (Nanjing)

US Patent
LigandPNGBDBM50202986(2-furan-2-yl-7-(2-{4-[4-(2-methoxy-ethoxy)-phenyl]...)
Affinity DataIC50:  2.5nMAssay Description:The IC50 (nM) values of the example compound HZ10126 and several reference compounds against the rat A2A receptor were measured in an in vitro assay,...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Inxmed (Nanjing)

US Patent
LigandPNGBDBM86760(CAS_104924 | CGS 21680 | NSC_104924 | US11440916, ...)
Affinity DataIC50:  66.9nMAssay Description:The IC50 (nM) values of the example compound HZ10126 and several reference compounds against the rat A2A receptor were measured in an in vitro assay,...More data for this Ligand-Target Pair