Compile Data Set for Download or QSAR
maximum 50k data
Found 14 Enz. Inhib. hit(s) with all data for assayid = 1 entry = 50032604
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Frosst Centre For Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50331795(1,1,1-trifluoro-2-(1-((2-(2-hydroxypropan-2-yl)-3-...)
Affinity DataKi:  2.60E+3nMAssay Description:Displacement of labeled MK-499 from human ERGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Frosst Centre For Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50331796(1,1,1-trifluoro-2-(1-((2-(1-hydroxyethyl)-3-phenyl...)
Affinity DataKi:  3.80E+3nMAssay Description:Displacement of labeled MK-499 from human ERGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Frosst Centre For Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50331797(1-(3-phenyl-6-((4-(1,1,1-trifluoro-2-hydroxybutan-...)
Affinity DataKi:  4.40E+3nMAssay Description:Displacement of labeled MK-499 from human ERGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Frosst Centre For Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50331806(CHEMBL1290649 | methyl 3-phenyl-6-((4-(1,1,1-trifl...)
Affinity DataKi:  6.30E+3nMAssay Description:Displacement of labeled MK-499 from human ERGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Frosst Centre For Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50331804((R)-3-(4-fluorophenyl)-6-((4-(1,1,1-trifluoro-2-hy...)
Affinity DataKi:  1.10E+4nMAssay Description:Displacement of labeled MK-499 from human ERGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Frosst Centre For Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50331794(1,1,1-trifluoro-2-(1-((2-(hydroxymethyl)-3-phenylb...)
Affinity DataKi:  1.30E+4nMAssay Description:Displacement of labeled MK-499 from human ERGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Frosst Centre For Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50331803((S)-3-(4-fluorophenyl)-6-((4-(1,1,1-trifluoro-2-hy...)
Affinity DataKi:  1.30E+4nMAssay Description:Displacement of labeled MK-499 from human ERGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Frosst Centre For Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50331802((S)-3-(3-fluorophenyl)-6-((4-(1,1,1-trifluoro-2-hy...)
Affinity DataKi:  1.40E+4nMAssay Description:Displacement of labeled MK-499 from human ERGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Frosst Centre For Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50331801((S)-3-phenyl-6-((4-(1,1,1-trifluoro-2-hydroxybutan...)
Affinity DataKi:  1.60E+4nMAssay Description:Displacement of labeled MK-499 from human ERGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Frosst Centre For Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50331800(3-phenyl-6-((4-(1,1,1-trifluoro-2-hydroxybutan-2-y...)
Affinity DataKi:  1.70E+4nMAssay Description:Displacement of labeled MK-499 from human ERGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Frosst Centre For Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50331805((S)-3-(4-fluorophenyl)-6-((4-(1,1,1-trifluoro-2-hy...)
Affinity DataKi: >2.00E+4nMAssay Description:Displacement of labeled MK-499 from human ERGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Frosst Centre For Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50331798(CHEMBL1289328 | N,N-dimethyl-3-phenyl-6-((4-(1,1,1...)
Affinity DataKi: >2.00E+4nMAssay Description:Displacement of labeled MK-499 from human ERGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Frosst Centre For Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50331793(3-phenyl-6-((4-(1,1,1-trifluoro-2-hydroxybutan-2-y...)
Affinity DataKi: >2.00E+4nMAssay Description:Displacement of labeled MK-499 from human ERGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Frosst Centre For Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50331799(CHEMBL1289329 | N-methyl-3-phenyl-6-((4-(1,1,1-tri...)
Affinity DataKi: >2.00E+4nMAssay Description:Displacement of labeled MK-499 from human ERGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed