Compile Data Set for Download or QSAR
maximum 50k data
Found 4 Enz. Inhib. hit(s) with all data for assayid = 2 entry = 50002786
TargetEstrogen receptor(Homo sapiens (Human))
Peking University Shenzhen Graduate School

Curated by ChEMBL
LigandPNGBDBM50462974(CHEMBL4240100)
Affinity DataKi:  0.0700nMAssay Description:Antagonist activity at full length recombinant human ERalpha expressed in baculovirus expression system assessed as inhibition of estradiol-induced E...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Peking University Shenzhen Graduate School

Curated by ChEMBL
LigandPNGBDBM50462976(CHEMBL4250447)
Affinity DataKi:  6.90nMAssay Description:Antagonist activity at full length recombinant human ERalpha expressed in baculovirus expression system assessed as inhibition of estradiol-induced E...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Peking University Shenzhen Graduate School

Curated by ChEMBL
LigandPNGBDBM50462987(CHEMBL4250610)
Affinity DataKi:  11nMAssay Description:Antagonist activity at full length recombinant human ERalpha expressed in baculovirus expression system assessed as inhibition of estradiol-induced E...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Peking University Shenzhen Graduate School

Curated by ChEMBL
LigandPNGBDBM50462973(CHEMBL4246022)
Affinity DataKi:  25nMAssay Description:Antagonist activity at full length recombinant human ERalpha expressed in baculovirus expression system assessed as inhibition of estradiol-induced E...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed