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Found 8 Enz. Inhib. hit(s) with all data for assayid = 2 entry = 50047632
TargetCholinesterase(Equus caballus (Horse))
Universiti Putra Malaysia

Curated by ChEMBL
LigandPNGBDBM8961(1,2,3,4-tetrahydro-9-acridinamine | 1,2,3,4-tetrah...)
Affinity DataIC50:  10nMAssay Description:Inhibition of equine serum BChE preincubated for 15 mins followed by addition of S-butyrylthiocholine iodide as substrate measured after 30 mins by E...More data for this Ligand-Target Pair
TargetCholinesterase(Equus caballus (Horse))
Universiti Putra Malaysia

Curated by ChEMBL
LigandPNGBDBM50180622(CHEMBL3814519)
Affinity DataIC50:  600nMAssay Description:Inhibition of equine serum BChE preincubated for 15 mins followed by addition of S-butyrylthiocholine iodide as substrate measured after 30 mins by E...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
Universiti Putra Malaysia

Curated by ChEMBL
LigandPNGBDBM50180620(CHEMBL3814587)
Affinity DataIC50:  1.40E+3nMAssay Description:Inhibition of equine serum BChE preincubated for 15 mins followed by addition of S-butyrylthiocholine iodide as substrate measured after 30 mins by E...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
Universiti Putra Malaysia

Curated by ChEMBL
LigandPNGBDBM50180623(CHEMBL3814100)
Affinity DataIC50:  2.30E+3nMAssay Description:Inhibition of equine serum BChE preincubated for 15 mins followed by addition of S-butyrylthiocholine iodide as substrate measured after 30 mins by E...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
Universiti Putra Malaysia

Curated by ChEMBL
LigandPNGBDBM50180621(CHEMBL3814621)
Affinity DataIC50:  2.70E+3nMAssay Description:Inhibition of equine serum BChE preincubated for 15 mins followed by addition of S-butyrylthiocholine iodide as substrate measured after 30 mins by E...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
Universiti Putra Malaysia

Curated by ChEMBL
LigandPNGBDBM50180626(CHEMBL3601745)
Affinity DataIC50:  4.70E+3nMAssay Description:Inhibition of equine serum BChE preincubated for 15 mins followed by addition of S-butyrylthiocholine iodide as substrate measured after 30 mins by E...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
Universiti Putra Malaysia

Curated by ChEMBL
LigandPNGBDBM50180624(CHEMBL3601736)
Affinity DataIC50:  6.50E+3nMAssay Description:Inhibition of equine serum BChE preincubated for 15 mins followed by addition of S-butyrylthiocholine iodide as substrate measured after 30 mins by E...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
Universiti Putra Malaysia

Curated by ChEMBL
LigandPNGBDBM50180625(CHEMBL3601744)
Affinity DataIC50:  1.06E+4nMAssay Description:Inhibition of equine serum BChE preincubated for 15 mins followed by addition of S-butyrylthiocholine iodide as substrate measured after 30 mins by E...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed