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Found 11 Enz. Inhib. hit(s) with all data for assayid = 2 entry = 50048485
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4C(Rattus norvegicus)
Institut De Recherche Jouveinal-Parke Davis

Curated by ChEMBL
LigandPNGBDBM14361((R,S)-Rolipram | 4-(3-cyclopentyloxy-4-methoxy-phe...)
Affinity DataIC50:  5nMAssay Description:Binding affinity against high affinity rolipram binding site (HARBS) was determined by displacing radioactive [3H]rolipram from brain membrane suspen...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4C(Rattus norvegicus)
Institut De Recherche Jouveinal-Parke Davis

Curated by ChEMBL
LigandPNGBDBM50217546(CHEMBL125123)
Affinity DataIC50:  1.09E+3nMAssay Description:Binding affinity against high affinity rolipram binding site (HARBS) was determined by displacing radioactive [3H]rolipram from brain membrane suspen...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4C(Rattus norvegicus)
Institut De Recherche Jouveinal-Parke Davis

Curated by ChEMBL
LigandPNGBDBM50217545(CHEMBL341304)
Affinity DataIC50: >2.00E+3nMAssay Description:Binding affinity against high affinity rolipram binding site (HARBS) was determined by displacing radioactive [3H]rolipram from brain membrane suspen...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4C(Rattus norvegicus)
Institut De Recherche Jouveinal-Parke Davis

Curated by ChEMBL
LigandPNGBDBM50217549(CHEMBL332853)
Affinity DataIC50: >3.00E+3nMAssay Description:Binding affinity against high affinity rolipram binding site (HARBS) was determined by displacing radioactive [3H]rolipram from brain membrane suspen...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4C(Rattus norvegicus)
Institut De Recherche Jouveinal-Parke Davis

Curated by ChEMBL
LigandPNGBDBM50217556(CHEMBL125828)
Affinity DataIC50: >3.00E+3nMAssay Description:Binding affinity against high affinity rolipram binding site (HARBS) was determined by displacing radioactive [3H]rolipram from brain membrane suspen...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4C(Rattus norvegicus)
Institut De Recherche Jouveinal-Parke Davis

Curated by ChEMBL
LigandPNGBDBM50217555(CHEMBL332854)
Affinity DataIC50: >3.00E+3nMAssay Description:Binding affinity against high affinity rolipram binding site (HARBS) was determined by displacing radioactive [3H]rolipram from brain membrane suspen...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4C(Rattus norvegicus)
Institut De Recherche Jouveinal-Parke Davis

Curated by ChEMBL
LigandPNGBDBM50217558(CHEMBL338684)
Affinity DataIC50: >3.00E+3nMAssay Description:Binding affinity against high affinity rolipram binding site (HARBS) was determined by displacing radioactive [3H]rolipram from brain membrane suspen...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4C(Rattus norvegicus)
Institut De Recherche Jouveinal-Parke Davis

Curated by ChEMBL
LigandPNGBDBM50217560(CHEMBL126581)
Affinity DataIC50: >3.00E+3nMAssay Description:Binding affinity against high affinity rolipram binding site (HARBS) was determined by displacing radioactive [3H]rolipram from brain membrane suspen...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4C(Rattus norvegicus)
Institut De Recherche Jouveinal-Parke Davis

Curated by ChEMBL
LigandPNGBDBM50217550(CHEMBL111925 | CI-1018)
Affinity DataIC50: >3.00E+3nMAssay Description:Binding affinity against high affinity rolipram binding site (HARBS) was determined by displacing radioactive [3H]rolipram from brain membrane suspen...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4C(Rattus norvegicus)
Institut De Recherche Jouveinal-Parke Davis

Curated by ChEMBL
LigandPNGBDBM50217551(CHEMBL419791)
Affinity DataIC50: >3.00E+3nMAssay Description:Binding affinity against high affinity rolipram binding site (HARBS) was determined by displacing radioactive [3H]rolipram from brain membrane suspen...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4C(Rattus norvegicus)
Institut De Recherche Jouveinal-Parke Davis

Curated by ChEMBL
LigandPNGBDBM50217553(CHEMBL339749)
Affinity DataIC50: >3.00E+3nMAssay Description:Binding affinity against high affinity rolipram binding site (HARBS) was determined by displacing radioactive [3H]rolipram from brain membrane suspen...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed