Compile Data Set for Download or QSAR
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Found 9 Enz. Inhib. hit(s) with all data for assayid = 3 entry = 1132
TargetChromatin remodeling regulator CECR2 [424-538](Homo sapiens (Human))
Genentech

US Patent
LigandPNGBDBM310905(2-methyl-7-(6-methyl-7-oxo-1H-pyrrolo[2,3-c]pyridi...)
Affinity DataIC50:  36nMAssay Description:His/Flag epitope tagged CECR2424-538 was cloned, expressed, and purified to homogeneity. CECR2 binding and inhibition was assessed by monitoring the ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetChromatin remodeling regulator CECR2 [424-538](Homo sapiens (Human))
Genentech

US Patent
LigandPNGBDBM310911(6-methyl-4-(2-methyl-3,4-dihydro-1H-isoquinolin-6-...)
Affinity DataIC50:  54nMAssay Description:His/Flag epitope tagged CECR2424-538 was cloned, expressed, and purified to homogeneity. CECR2 binding and inhibition was assessed by monitoring the ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetChromatin remodeling regulator CECR2 [424-538](Homo sapiens (Human))
Genentech

US Patent
LigandPNGBDBM310910(4-(6-methyl-7-oxo-1H-pyrrolo[2,3-c]pyridin-4-yl)-N...)
Affinity DataIC50:  75nMAssay Description:His/Flag epitope tagged CECR2424-538 was cloned, expressed, and purified to homogeneity. CECR2 binding and inhibition was assessed by monitoring the ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetChromatin remodeling regulator CECR2 [424-538](Homo sapiens (Human))
Genentech

US Patent
LigandPNGBDBM310912(3-(2,6-dimethyl-7-oxo-1H-pyrrolo[2,3-c]pyridin-4-y...)
Affinity DataIC50:  130nMAssay Description:His/Flag epitope tagged CECR2424-538 was cloned, expressed, and purified to homogeneity. CECR2 binding and inhibition was assessed by monitoring the ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetChromatin remodeling regulator CECR2 [424-538](Homo sapiens (Human))
Genentech

US Patent
LigandPNGBDBM310909(4-[4-(3,3-difluoroazetidine-1-carbonyl)phenyl]-6-m...)
Affinity DataIC50:  130nMAssay Description:His/Flag epitope tagged CECR2424-538 was cloned, expressed, and purified to homogeneity. CECR2 binding and inhibition was assessed by monitoring the ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetChromatin remodeling regulator CECR2 [424-538](Homo sapiens (Human))
Genentech

US Patent
LigandPNGBDBM310904(3-methoxy-N-[4-(6-methyl-7-oxo-1H-pyrrolo[2,3-c]py...)
Affinity DataIC50:  170nMAssay Description:His/Flag epitope tagged CECR2424-538 was cloned, expressed, and purified to homogeneity. CECR2 binding and inhibition was assessed by monitoring the ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetChromatin remodeling regulator CECR2 [424-538](Homo sapiens (Human))
Genentech

US Patent
LigandPNGBDBM310908(6-methyl-4-(4-(4-methyl-3-oxopiperazine-1-carbonyl...)
Affinity DataIC50:  240nMAssay Description:His/Flag epitope tagged CECR2424-538 was cloned, expressed, and purified to homogeneity. CECR2 binding and inhibition was assessed by monitoring the ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetChromatin remodeling regulator CECR2 [424-538](Homo sapiens (Human))
Genentech

US Patent
LigandPNGBDBM310906(N,N-dimethyl-4-(6-methyl-7-oxo-1H-pyrrolo[2,3-c]py...)
Affinity DataIC50:  730nMAssay Description:His/Flag epitope tagged CECR2424-538 was cloned, expressed, and purified to homogeneity. CECR2 binding and inhibition was assessed by monitoring the ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetChromatin remodeling regulator CECR2 [424-538](Homo sapiens (Human))
Genentech

US Patent
LigandPNGBDBM310907(3-(6-ethyl-7-oxo-1H-pyrrolo[2,3-c]pyridin-4-yl)-N,...)
Affinity DataIC50:  1.30E+3nMAssay Description:His/Flag epitope tagged CECR2424-538 was cloned, expressed, and purified to homogeneity. CECR2 binding and inhibition was assessed by monitoring the ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent