Compile Data Set for Download or QSAR
maximum 50k data
Found 22 Enz. Inhib. hit(s) with all data for assayid = 4 entry = 634
TargetRho-associated protein kinase 1(Homo sapiens (Human))
The Regents of The University of Michigan

US Patent
LigandPNGBDBM50173310(CHEMBL3808660 | US10023564, Example 1)
Affinity DataIC50:  11nMAssay Description:Rho-associated coiled-coil kinase (ROCK) assays were performed with the ADP-Glo system using 0.1 μg ROCK1 and 1 μg S6K substrate, and 100 &...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetRho-associated protein kinase 1(Homo sapiens (Human))
The Regents of The University of Michigan

US Patent
LigandPNGBDBM50173307(CHEMBL3809796 | US10023564, Example 8)
Affinity DataIC50:  17nMAssay Description:Rho-associated coiled-coil kinase (ROCK) assays were performed with the ADP-Glo system using 0.1 μg ROCK1 and 1 μg S6K substrate, and 100 &...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetRho-associated protein kinase 1(Homo sapiens (Human))
The Regents of The University of Michigan

US Patent
LigandPNGBDBM50173315(CHEMBL3809100 | US10023564, Example 4)
Affinity DataIC50:  21nMAssay Description:Rho-associated coiled-coil kinase (ROCK) assays were performed with the ADP-Glo system using 0.1 μg ROCK1 and 1 μg S6K substrate, and 100 &...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetRho-associated protein kinase 1(Homo sapiens (Human))
The Regents of The University of Michigan

US Patent
LigandPNGBDBM50173305(CHEMBL3810107 | US10023564, Example 3)
Affinity DataIC50:  23nMAssay Description:Rho-associated coiled-coil kinase (ROCK) assays were performed with the ADP-Glo system using 0.1 μg ROCK1 and 1 μg S6K substrate, and 100 &...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetRho-associated protein kinase 1(Homo sapiens (Human))
The Regents of The University of Michigan

US Patent
LigandPNGBDBM50173311(CHEMBL3810073 | US10023564, Example 6)
Affinity DataIC50:  50nMAssay Description:Rho-associated coiled-coil kinase (ROCK) assays were performed with the ADP-Glo system using 0.1 μg ROCK1 and 1 μg S6K substrate, and 100 &...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetRho-associated protein kinase 1(Homo sapiens (Human))
The Regents of The University of Michigan

US Patent
LigandPNGBDBM50173325(CHEMBL3809965 | US10023564, Example 5)
Affinity DataIC50:  57nMAssay Description:Rho-associated coiled-coil kinase (ROCK) assays were performed with the ADP-Glo system using 0.1 μg ROCK1 and 1 μg S6K substrate, and 100 &...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetRho-associated protein kinase 1(Homo sapiens (Human))
The Regents of The University of Michigan

US Patent
LigandPNGBDBM50173323(CHEMBL3808621 | US10023564, Example 2)
Affinity DataIC50:  61nMAssay Description:Rho-associated coiled-coil kinase (ROCK) assays were performed with the ADP-Glo system using 0.1 μg ROCK1 and 1 μg S6K substrate, and 100 &...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetRho-associated protein kinase 1(Homo sapiens (Human))
The Regents of The University of Michigan

US Patent
LigandPNGBDBM50173314(CHEMBL3808840 | US10023564, Example 16)
Affinity DataIC50:  69nMAssay Description:Rho-associated coiled-coil kinase (ROCK) assays were performed with the ADP-Glo system using 0.1 μg ROCK1 and 1 μg S6K substrate, and 100 &...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetRho-associated protein kinase 1(Homo sapiens (Human))
The Regents of The University of Michigan

US Patent
LigandPNGBDBM50173320(GSK-180736A | GSK180736A | US10023564, Compound GS...)
Affinity DataIC50:  78nMAssay Description:Rho-associated coiled-coil kinase (ROCK) assays were performed with the ADP-Glo system using 0.1 μg ROCK1 and 1 μg S6K substrate, and 100 &...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetRho-associated protein kinase 1(Homo sapiens (Human))
The Regents of The University of Michigan

US Patent
LigandPNGBDBM50173312(CHEMBL3810312 | US10023564, Example 18)
Affinity DataIC50:  97nMAssay Description:Rho-associated coiled-coil kinase (ROCK) assays were performed with the ADP-Glo system using 0.1 μg ROCK1 and 1 μg S6K substrate, and 100 &...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetRho-associated protein kinase 1(Homo sapiens (Human))
The Regents of The University of Michigan

US Patent
LigandPNGBDBM50173329(CHEMBL3809697 | US10023564, Example 15)
Affinity DataIC50:  150nMAssay Description:Rho-associated coiled-coil kinase (ROCK) assays were performed with the ADP-Glo system using 0.1 μg ROCK1 and 1 μg S6K substrate, and 100 &...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetRho-associated protein kinase 1(Homo sapiens (Human))
The Regents of The University of Michigan

US Patent
LigandPNGBDBM50173317(CHEMBL3810349 | US10023564, Example 12)
Affinity DataIC50:  190nMAssay Description:Rho-associated coiled-coil kinase (ROCK) assays were performed with the ADP-Glo system using 0.1 μg ROCK1 and 1 μg S6K substrate, and 100 &...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetRho-associated protein kinase 1(Homo sapiens (Human))
The Regents of The University of Michigan

US Patent
LigandPNGBDBM50173324(CHEMBL3809124 | US10023564, Example 30)
Affinity DataIC50:  200nMAssay Description:Rho-associated coiled-coil kinase (ROCK) assays were performed with the ADP-Glo system using 0.1 μg ROCK1 and 1 μg S6K substrate, and 100 &...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetRho-associated protein kinase 1(Homo sapiens (Human))
The Regents of The University of Michigan

US Patent
LigandPNGBDBM50173328(CHEMBL3808918 | US10023564, Example 14)
Affinity DataIC50:  290nMAssay Description:Rho-associated coiled-coil kinase (ROCK) assays were performed with the ADP-Glo system using 0.1 μg ROCK1 and 1 μg S6K substrate, and 100 &...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetRho-associated protein kinase 1(Homo sapiens (Human))
The Regents of The University of Michigan

US Patent
LigandPNGBDBM50173326(CHEMBL3809604 | US10023564, Example 29)
Affinity DataIC50:  400nMAssay Description:Rho-associated coiled-coil kinase (ROCK) assays were performed with the ADP-Glo system using 0.1 μg ROCK1 and 1 μg S6K substrate, and 100 &...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetRho-associated protein kinase 1(Homo sapiens (Human))
The Regents of The University of Michigan

US Patent
LigandPNGBDBM50173327(CHEMBL3808499 | US10023564, Example 28)
Affinity DataIC50:  450nMAssay Description:Rho-associated coiled-coil kinase (ROCK) assays were performed with the ADP-Glo system using 0.1 μg ROCK1 and 1 μg S6K substrate, and 100 &...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetRho-associated protein kinase 1(Homo sapiens (Human))
The Regents of The University of Michigan

US Patent
LigandPNGBDBM50173330(CHEMBL3808657 | US10023564, Example 13)
Affinity DataIC50:  1.90E+3nMAssay Description:Rho-associated coiled-coil kinase (ROCK) assays were performed with the ADP-Glo system using 0.1 μg ROCK1 and 1 μg S6K substrate, and 100 &...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetRho-associated protein kinase 1(Homo sapiens (Human))
The Regents of The University of Michigan

US Patent
LigandPNGBDBM50173309(CHEMBL3809913 | US10023564, Example 10)
Affinity DataIC50:  5.80E+3nMAssay Description:Rho-associated coiled-coil kinase (ROCK) assays were performed with the ADP-Glo system using 0.1 μg ROCK1 and 1 μg S6K substrate, and 100 &...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetRho-associated protein kinase 1(Homo sapiens (Human))
The Regents of The University of Michigan

US Patent
LigandPNGBDBM50173308(CHEMBL3810271 | US10023564, Example 9)
Affinity DataIC50:  6.70E+3nMAssay Description:Rho-associated coiled-coil kinase (ROCK) assays were performed with the ADP-Glo system using 0.1 μg ROCK1 and 1 μg S6K substrate, and 100 &...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetRho-associated protein kinase 1(Homo sapiens (Human))
The Regents of The University of Michigan

US Patent
LigandPNGBDBM50173319(CHEMBL3809020 | US10023564, Example 11)
Affinity DataIC50: >1.00E+4nMAssay Description:Rho-associated coiled-coil kinase (ROCK) assays were performed with the ADP-Glo system using 0.1 μg ROCK1 and 1 μg S6K substrate, and 100 &...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetRho-associated protein kinase 1(Homo sapiens (Human))
The Regents of The University of Michigan

US Patent
LigandPNGBDBM50173318(CHEMBL3809788 | US10023564, Example 17)
Affinity DataIC50: >1.00E+4nMAssay Description:Rho-associated coiled-coil kinase (ROCK) assays were performed with the ADP-Glo system using 0.1 μg ROCK1 and 1 μg S6K substrate, and 100 &...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetRho-associated protein kinase 1(Homo sapiens (Human))
The Regents of The University of Michigan

US Patent
LigandPNGBDBM50173306(CHEMBL3808565 | US10023564, Example 7)
Affinity DataIC50: >1.00E+5nMAssay Description:Rho-associated coiled-coil kinase (ROCK) assays were performed with the ADP-Glo system using 0.1 μg ROCK1 and 1 μg S6K substrate, and 100 &...More data for this Ligand-Target Pair
In DepthDetails US Patent