Compile Data Set for Download or QSAR
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Found 6 Enz. Inhib. hit(s) with all data for assayid = 7 entry = 50043769
TargetP2X purinoceptor 4(Mus musculus)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50446060(CHEMBL3103385)
Affinity DataIC50:  1.49E+4nMAssay Description:Antagonist activity at mouse P2X4 receptor assessed as inhibition of ATP-induced cytosolic calcium influx preincubated for 30 mins followed by ATP ad...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 4(Mus musculus)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50446072(CHEMBL3103369)
Affinity DataIC50:  9.84E+4nMAssay Description:Antagonist activity at mouse P2X4 receptor assessed as inhibition of ATP-induced cytosolic calcium influx preincubated for 30 mins followed by ATP ad...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 4(Mus musculus)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50446068(CHEMBL3103375)
Affinity DataIC50: >1.00E+5nMAssay Description:Antagonist activity at mouse P2X4 receptor assessed as inhibition of ATP-induced cytosolic calcium influx preincubated for 30 mins followed by ATP ad...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 4(Mus musculus)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50446076(CHEMBL1483754)
Affinity DataIC50: >1.00E+5nMAssay Description:Antagonist activity at mouse P2X4 receptor assessed as inhibition of ATP-induced cytosolic calcium influx preincubated for 30 mins followed by ATP ad...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 4(Mus musculus)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50446070(CHEMBL3103371)
Affinity DataIC50:  1.02E+5nMAssay Description:Antagonist activity at mouse P2X4 receptor assessed as inhibition of ATP-induced cytosolic calcium influx preincubated for 30 mins followed by ATP ad...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 4(Mus musculus)
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50446069(CHEMBL3103372)
Affinity DataIC50:  1.23E+5nMAssay Description:Antagonist activity at mouse P2X4 receptor assessed as inhibition of ATP-induced cytosolic calcium influx preincubated for 30 mins followed by ATP ad...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed